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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • CP19

    CAS:
    CP19 blocks histamine receptors; inhibits EBOV and MARV with IC50s of 3.4 μM and 29.5 μM, respectively; antiviral [1].
    Formula:C26H30N2O5
    Color and Shape:Solid
    Molecular weight:450.53

    Ref: TM-T73571

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AB-MECA

    CAS:
    AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.
    Formula:C18H21N7O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.4

    Ref: TM-T14082

    1mg
    239.00€
    5mg
    1,018.00€
    10mg
    1,783.00€
  • Povafonidine

    CAS:
    Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.
    Formula:C11H13N5
    Color and Shape:Solid
    Molecular weight:215.25

    Ref: TM-T60263

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A1/A3 AR antagonist 2

    CAS:
    The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.
    Formula:C22H16N2O3S
    Color and Shape:Solid
    Molecular weight:388.44

    Ref: TM-T61744

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BAY-27-9955

    CAS:
    BAY-27-9955 is a glucagon receptor antagonist.
    Formula:C23H31FO
    Color and Shape:Solid
    Molecular weight:342.49

    Ref: TM-T30299

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • GPR183-IN-2

    CAS:
    GPR183-IN-2 (compound 23) is an effective, orally active inhibitor of GPR183, displaying an IC50 value of 39.45 nM in Ca2+ mobilization assays. This compound has potential applications in research related to cancer, autoimmune diseases, pain, and osteoporosis.
    Formula:C19H23BrN2O3
    Color and Shape:Solid
    Molecular weight:407.3

    Ref: TM-T88500

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ATC0065

    CAS:
    ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.
    Formula:C25H29BrF3N5O
    Color and Shape:Solid
    Molecular weight:552.43

    Ref: TM-T26676

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Org-12962

    CAS:
    Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).
    Formula:C10H11ClF3N3
    Purity:98.34%
    Color and Shape:Solid
    Molecular weight:265.66

    Ref: TM-T16401

    5mg
    46.00€
    1mL*10mM (DMSO)
    49.00€
    10mg
    58.00€
    25mg
    86.00€
    50mg
    105.00€
    100mg
    150.00€
  • O-2093

    CAS:
    anandamide uptake inhibitor
    Formula:C34H43Cl2NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:584.62

    Ref: TM-T23100

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • BMS-193884

    CAS:
    BMS-193884 is an oral endothelin antagonist for the treatment of congestive heart failure (CHF) and pulmonary arterial hypertension.
    Formula:C20H17N3O4S
    Color and Shape:Solid
    Molecular weight:395.43

    Ref: TM-T30501

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5-HT6/5-HT2A receptor ligand-2

    CAS:
    Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.
    Formula:C20H18FN3O2
    Color and Shape:Solid
    Molecular weight:351.37

    Ref: TM-T61220

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 2-Thio-UTP

    CAS:
    2-ThioUTP tetrasodium salt is a P2Y2 agonist.
    Formula:C9H15N2O14P3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.21

    Ref: TM-T22503

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5-Carboxamidotryptamine maleate

    CAS:
    5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.
    Formula:C15H17N3O5
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:319.31

    Ref: TM-T22520

    1mg
    35.00€
    5mg
    84.00€
    10mg
    119.00€
    25mg
    207.00€
    50mg
    289.00€
    100mg
    399.00€
    200mg
    555.00€
  • Mirisetron

    CAS:
    Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.
    Formula:C24H31N3O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:393.52

    Ref: TM-T70879

    1mg
    285.00€
    5mg
    692.00€
    10mg
    947.00€
    25mg
    1,458.00€
    50mg
    1,839.00€
    100mg
    2,322.00€
  • TSI-01

    CAS:
    TSI-01,Pro-inflammatory phospholipid mediator. Inhibits LPCAT2 (IC50=0.47 μM). Suppresses PAF biosynthesis in macrophages.
    Formula:C14H11Cl2NO4
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:328.15

    Ref: TM-T24904

    1mg
    83.00€
    5mg
    175.00€
    1mL*10mM (DMSO)
    193.00€
    10mg
    305.00€
    25mg
    659.00€
    50mg
    1,046.00€
    100mg
    1,607.00€
    200mg
    2,164.00€
  • Cirazoline hydrochloride

    CAS:
    Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.
    Formula:C13H17ClN2O
    Purity:99.863%
    Color and Shape:Solid
    Molecular weight:252.74

    Ref: TM-T14972

    1mg
    60.00€
    5mg
    130.00€
    10mg
    192.00€
    25mg
    324.00€
    50mg
    480.00€
    100mg
    683.00€
    200mg
    888.00€
  • GR 113808

    CAS:
    GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.
    Formula:C19H27N3O4S
    Purity:98.16% - 99.96%
    Color and Shape:Solid
    Molecular weight:393.5

    Ref: TM-T15414

    1mg
    35.00€
    5mg
    79.00€
  • A-123189

    CAS:
    A-123189 is a potent, alpha1D-selective antagonist.
    Formula:C26H28N4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:476.59

    Ref: TM-T26466

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Nivasorexant

    CAS:
    Nivasorexant is a potent antagonist of the orexin receptor.
    Formula:C23H23N7O2
    Color and Shape:Solid
    Molecular weight:429.47

    Ref: TM-T62370

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Lu AA 47070

    CAS:
    adenosine A2A receptor antagonist
    Formula:C17H20F2N3O6PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:463.39

    Ref: TM-T22934

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€