
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,025 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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CP19
CAS:CP19 blocks histamine receptors; inhibits EBOV and MARV with IC50s of 3.4 μM and 29.5 μM, respectively; antiviral [1].Formula:C26H30N2O5Color and Shape:SolidMolecular weight:450.53AB-MECA
CAS:AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.Formula:C18H21N7O4Purity:98%Color and Shape:SolidMolecular weight:399.4Povafonidine
CAS:Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.Formula:C11H13N5Color and Shape:SolidMolecular weight:215.25A1/A3 AR antagonist 2
CAS:The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.Formula:C22H16N2O3SColor and Shape:SolidMolecular weight:388.44BAY-27-9955
CAS:BAY-27-9955 is a glucagon receptor antagonist.Formula:C23H31FOColor and Shape:SolidMolecular weight:342.49GPR183-IN-2
CAS:GPR183-IN-2 (compound 23) is an effective, orally active inhibitor of GPR183, displaying an IC50 value of 39.45 nM in Ca2+ mobilization assays. This compound has potential applications in research related to cancer, autoimmune diseases, pain, and osteoporosis.Formula:C19H23BrN2O3Color and Shape:SolidMolecular weight:407.3ATC0065
CAS:ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.Formula:C25H29BrF3N5OColor and Shape:SolidMolecular weight:552.43Org-12962
CAS:Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).Formula:C10H11ClF3N3Purity:98.34%Color and Shape:SolidMolecular weight:265.66O-2093
CAS:anandamide uptake inhibitorFormula:C34H43Cl2NO3Purity:98%Color and Shape:SolidMolecular weight:584.62BMS-193884
CAS:BMS-193884 is an oral endothelin antagonist for the treatment of congestive heart failure (CHF) and pulmonary arterial hypertension.Formula:C20H17N3O4SColor and Shape:SolidMolecular weight:395.435-HT6/5-HT2A receptor ligand-2
CAS:Compound 42: brain-penetrant, dual 5-HT6/5-HT2A antagonist, Ki of 25 nM/32 nM, pro-cognitive.Formula:C20H18FN3O2Color and Shape:SolidMolecular weight:351.372-Thio-UTP
CAS:2-ThioUTP tetrasodium salt is a P2Y2 agonist.Formula:C9H15N2O14P3SPurity:98%Color and Shape:SolidMolecular weight:500.215-Carboxamidotryptamine maleate
CAS:5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.Formula:C15H17N3O5Purity:99.88%Color and Shape:SolidMolecular weight:319.31Mirisetron
CAS:Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.Formula:C24H31N3O2Purity:99.88%Color and Shape:SolidMolecular weight:393.52TSI-01
CAS:TSI-01,Pro-inflammatory phospholipid mediator. Inhibits LPCAT2 (IC50=0.47 μM). Suppresses PAF biosynthesis in macrophages.Formula:C14H11Cl2NO4Purity:99.87%Color and Shape:SolidMolecular weight:328.15Ref: TM-T24904
1mg83.00€5mg175.00€1mL*10mM (DMSO)193.00€10mg305.00€25mg659.00€50mg1,046.00€100mg1,607.00€200mg2,164.00€Cirazoline hydrochloride
CAS:Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.Formula:C13H17ClN2OPurity:99.863%Color and Shape:SolidMolecular weight:252.74GR 113808
CAS:GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.Formula:C19H27N3O4SPurity:98.16% - 99.96%Color and Shape:SolidMolecular weight:393.5A-123189
CAS:A-123189 is a potent, alpha1D-selective antagonist.Formula:C26H28N4O3SPurity:98%Color and Shape:SolidMolecular weight:476.59Nivasorexant
CAS:Nivasorexant is a potent antagonist of the orexin receptor.Formula:C23H23N7O2Color and Shape:SolidMolecular weight:429.47Lu AA 47070
CAS:adenosine A2A receptor antagonistFormula:C17H20F2N3O6PSPurity:98%Color and Shape:SolidMolecular weight:463.39
