
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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ST1936
CAS:ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.Formula:C13H17ClN2Purity:98%Color and Shape:SolidMolecular weight:236.74Ref: TM-T23396
1mg44.00€5mg111.00€1mL*10mM (DMSO)123.00€10mg178.00€25mg316.00€50mg470.00€100mg682.00€200mg954.00€EP1-antagonist-1
CAS:EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).Formula:C19H15BrCl2N2O3Purity:97.06%Color and Shape:SolidMolecular weight:470.14COR167
CAS:COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.Formula:C28H38N2O2Color and Shape:SolidMolecular weight:434.61Phenyltoloxamine
CAS:Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).Formula:C17H21NOColor and Shape:SolidMolecular weight:255.35Immepip
CAS:Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.Formula:C9H15N3Color and Shape:SolidMolecular weight:165.24Adatanserin
CAS:Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.Formula:C21H31N5OPurity:99.33%Color and Shape:SolidMolecular weight:369.5CAY10680
CAS:CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.Formula:C18H16N2O2SColor and Shape:SolidMolecular weight:324.4LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Formula:C27H38ClN3OSPurity:98.06%Color and Shape:SolidMolecular weight:488.13AM404
CAS:AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.Formula:C26H37NO2Color and Shape:SolidMolecular weight:395.58FR 64822
CAS:FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.Formula:C11H14N4OColor and Shape:SolidMolecular weight:218.26N-0861 racemate
CAS:N-0861 racemate is the racemate of N-0861.Formula:C13H17N5Purity:98%Color and Shape:SolidMolecular weight:243.31TC-2153
CAS:TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.Formula:C7H5ClF3NS5Color and Shape:SolidMolecular weight:355.89JNJ-26070109
CAS:JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat.Formula:C23H17BrF2N4O3SPurity:98%Color and Shape:SolidMolecular weight:547.37MRS 1523
CAS:MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels & inhibits action potentials in rat DRG neurons.Formula:C23H29NO3SPurity:98%Color and Shape:SolidMolecular weight:399.55COR 170
CAS:inverse agonist of CB2 receptorsFormula:C31H36N2O2Purity:98%Color and Shape:SolidMolecular weight:468.63Dapiprazole
CAS:Dapiprazole, an alpha blocker, is used to reverse mydriasis after eye examination.Formula:C19H27N5Purity:98%Color and Shape:SolidMolecular weight:325.45SK1-IN-1
CAS:SK1-IN-1 is a SPHK1 inhibitor (IC50: 58 nM), with potential anticancer activity, and can be used to study cancer and neurodegenerative diseases.Formula:C22H30N4O3Purity:98.72%Color and Shape:SolidMolecular weight:398.5Tedatioxetine hydrobromide
CAS:Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.Formula:C18H22BrNSPurity:99.65%Color and Shape:SolidMolecular weight:364.34(S)-Terazosin
CAS:(S)-Terazosin is an active S-enantiomer of Terazosin.Formula:C19H25N5O4Color and Shape:SolidMolecular weight:387.43Licogliflozin
CAS:Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).Formula:C23H28O7Purity:98%Color and Shape:SolidMolecular weight:416.46
