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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • ST1936

    CAS:
    ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.
    Formula:C13H17ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:236.74

    Ref: TM-T23396

    1mg
    44.00€
    5mg
    111.00€
    1mL*10mM (DMSO)
    123.00€
    10mg
    178.00€
    25mg
    316.00€
    50mg
    470.00€
    100mg
    682.00€
    200mg
    954.00€
  • EP1-antagonist-1

    CAS:
    EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).
    Formula:C19H15BrCl2N2O3
    Purity:97.06%
    Color and Shape:Solid
    Molecular weight:470.14

    Ref: TM-T10031

    1mg
    109.00€
    5mg
    215.00€
    1mL*10mM (DMSO)
    243.00€
    10mg
    313.00€
    25mg
    492.00€
  • COR167

    CAS:
    COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.
    Formula:C28H38N2O2
    Color and Shape:Solid
    Molecular weight:434.61

    Ref: TM-T72007

    5mg
    304.00€
    10mg
    575.00€
    50mg
    2,367.00€
  • Phenyltoloxamine

    CAS:
    Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).
    Formula:C17H21NO
    Color and Shape:Solid
    Molecular weight:255.35

    Ref: TM-T60391

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Immepip

    CAS:
    Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.
    Formula:C9H15N3
    Color and Shape:Solid
    Molecular weight:165.24

    Ref: TM-T73408

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Adatanserin

    CAS:
    Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.
    Formula:C21H31N5O
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:369.5

    Ref: TM-T23631

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • CAY10680

    CAS:
    CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.
    Formula:C18H16N2O2S
    Color and Shape:Solid
    Molecular weight:324.4

    Ref: TM-T37354

    5mg
    239.00€
    10mg
    421.00€
    25mg
    945.00€
    50mg
    1,701.00€
  • LP44 hydrochloride

    CAS:
    LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.
    Formula:C27H38ClN3OS
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:488.13

    Ref: TM-T22931

    1mg
    37.00€
  • AM404

    CAS:
    AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.
    Formula:C26H37NO2
    Color and Shape:Solid
    Molecular weight:395.58

    Ref: TM-T39281

    5mg
    65.00€
    10mg
    105.00€
    50mg
    419.00€
    100mg
    713.00€
  • FR 64822

    CAS:
    FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.
    Formula:C11H14N4O
    Color and Shape:Solid
    Molecular weight:218.26

    Ref: TM-T27363

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • N-0861 racemate

    CAS:
    N-0861 racemate is the racemate of N-0861.
    Formula:C13H17N5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:243.31

    Ref: TM-T12136

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TC-2153

    CAS:
    TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.
    Formula:C7H5ClF3NS5
    Color and Shape:Solid
    Molecular weight:355.89

    Ref: TM-T70818

    25mg
    513.00€
    50mg
    853.00€
    100mg
    1,420.00€
  • JNJ-26070109

    CAS:
    JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat.
    Formula:C23H17BrF2N4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:547.37

    Ref: TM-T27669

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS 1523

    CAS:
    MRS 1523: selective adenosine A3 antagonist, Ki 18.9/113 nM (human/rat), blocks N-type Ca channels & inhibits action potentials in rat DRG neurons.
    Formula:C23H29NO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.55

    Ref: TM-T16135

    1mg
    178.00€
    5mg
    610.00€
  • COR 170

    CAS:
    inverse agonist of CB2 receptors
    Formula:C31H36N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.63

    Ref: TM-T22679

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dapiprazole

    CAS:
    Dapiprazole, an alpha blocker, is used to reverse mydriasis after eye examination.
    Formula:C19H27N5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:325.45

    Ref: TM-T21381

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SK1-IN-1

    CAS:
    SK1-IN-1 is a SPHK1 inhibitor (IC50: 58 nM), with potential anticancer activity, and can be used to study cancer and neurodegenerative diseases.
    Formula:C22H30N4O3
    Purity:98.72%
    Color and Shape:Solid
    Molecular weight:398.5

    Ref: TM-T12927

    1mg
    180.00€
  • Tedatioxetine hydrobromide

    CAS:
    Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.
    Formula:C18H22BrNS
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:364.34

    Ref: TM-T13110

    1mL*10mM (DMSO)
    44.00€
    1mg
    130.00€
    5mg
    313.00€
    10mg
    497.00€
    25mg
    1,044.00€
    50mg
    1,665.00€
  • (S)-Terazosin

    CAS:
    (S)-Terazosin is an active S-enantiomer of Terazosin.
    Formula:C19H25N5O4
    Color and Shape:Solid
    Molecular weight:387.43

    Ref: TM-T12815

    2mg
    111.00€
    5mg
    178.00€
    1mL*10mM (DMSO)
    203.00€
    50mg
    710.00€
    100mg
    1,116.00€
  • Licogliflozin

    CAS:
    Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).
    Formula:C23H28O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:416.46

    Ref: TM-T15752

    25mg
    775.00€
    50mg
    1,009.00€
    100mg
    1,674.00€