
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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L-775,606
CAS:L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.Formula:C25H29FN6Purity:98%Color and Shape:SolidMolecular weight:432.54VUF 5681 dihydrobromide
CAS:histamine H3 receptor silent antagonistFormula:C11H21Br2N3Purity:98%Color and Shape:SolidMolecular weight:355.11Verlukast
CAS:Verlukast (MK-0679) is a selective, orally active leukotriene D4 receptor antagonist for use in bronchial asthma research.Formula:C26H27ClN2O3S2Purity:98%Color and Shape:SolidMolecular weight:515.09JNJ-27141491
CAS:JNJ-27141491 is a potent, noncompetitive antagonist of human CCR2.Formula:C17H15F2N3O3SPurity:98%Color and Shape:SolidMolecular weight:379.38Metazosin
CAS:Metazosin is an antihypertensive agent that replaces 3H-prazosin from its bond to alpha-1 receptors of the cerebral cortex.Formula:C18H25N5O4Purity:98%Color and Shape:SolidMolecular weight:375.42LY 203647
CAS:LY 203647 is a antagonist of leukotriene D4 and E4 receptor.Formula:C21H30N8O3Purity:98%Color and Shape:SolidMolecular weight:442.51A 61603
CAS:Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.Formula:C14H20BrN3O3SColor and Shape:SolidMolecular weight:390.3DH97
CAS:MT2 melatonin receptor antagonistFormula:C22H26N2OPurity:98%Color and Shape:SolidMolecular weight:334.45A68930
CAS:A 68930 is a dopamine D-1 receptor antagonist. A 68930 inhibits NLRP3 inflammasome activity.Formula:C16H17NO3Color and Shape:SolidMolecular weight:271.31LY 225910
CAS:LY 225910 is a CCK2 receptor antagonist.Formula:C27H24BrN3O2Purity:98%Color and Shape:SolidMolecular weight:502.4MS 245 oxalate
CAS:MS 245 oxalate is a 5-HT6 antagonist.Formula:C21H24N2O7SPurity:98%Color and Shape:SolidMolecular weight:448.49CAY10535
CAS:CAY10535 is a selective TPβ antagonist (IC50 = 99 nM for TPβ vs 1970 nM for TPα), weakly affects platelets (IC50 = 985 nM).Formula:C18H21N3O7SColor and Shape:SolidMolecular weight:423.44N-Salicyloyltryptamine
CAS:N-Salicyloyltryptamine (STP): a tryptamine with anticonvulsant, anti-inflammatory, analgesic effects; inhibits Na+, Ca2+, K+ channels (IC50 34.6 μM).Formula:C17H16N2O2Color and Shape:SolidMolecular weight:280.32SB 235375
CAS:SB 235375 is a potent and selective antagonist of neurokinin-3 receptor with a low central nervous system-penetrant.Formula:C27H24N2O4Purity:98%Color and Shape:SolidMolecular weight:440.49A1AR antagonist 6
CAS:A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].Formula:C17H15N3O2Color and Shape:SolidMolecular weight:293.32SKF-83566 hydrobromide
CAS:D1-like dopamine receptor antagonistFormula:C17H19BrClNOPurity:98%Color and Shape:SolidMolecular weight:368.7Lu AA41063
CAS:Lu AA41063 is a potent and selective antagonist of the hA2A receptor.Formula:C16H17F2N3O2SColor and Shape:SolidMolecular weight:353.39Todralazine
CAS:Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.Formula:C11H12N4O2Purity:98%Color and Shape:SolidMolecular weight:232.24Lexipafant
CAS:Lexipafant is a platelet-activating factor (PAF) receptor antagonist.Formula:C23H30N4O4SColor and Shape:SolidMolecular weight:458.57T 82
CAS:T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.Formula:C56H62N6O8Purity:98%Color and Shape:SolidMolecular weight:947.146
