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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • L-775,606

    CAS:
    L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.
    Formula:C25H29FN6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.54

    Ref: TM-T27782

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • VUF 5681 dihydrobromide

    CAS:
    histamine H3 receptor silent antagonist
    Formula:C11H21Br2N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.11

    Ref: TM-T23519

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Verlukast

    CAS:
    Verlukast (MK-0679) is a selective, orally active leukotriene D4 receptor antagonist for use in bronchial asthma research.
    Formula:C26H27ClN2O3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.09

    Ref: TM-T19674

    50mg
    723.00€
    100mg
    1,094.00€
  • JNJ-27141491

    CAS:
    JNJ-27141491 is a potent, noncompetitive antagonist of human CCR2.
    Formula:C17H15F2N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:379.38

    Ref: TM-T27674

    25mg
    1,369.00€
  • Metazosin

    CAS:
    Metazosin is an antihypertensive agent that replaces 3H-prazosin from its bond to alpha-1 receptors of the cerebral cortex.
    Formula:C18H25N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:375.42

    Ref: TM-T25793

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LY 203647

    CAS:
    LY 203647 is a antagonist of leukotriene D4 and E4 receptor.
    Formula:C21H30N8O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:442.51

    Ref: TM-T27893

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A 61603

    CAS:
    Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.
    Formula:C14H20BrN3O3S
    Color and Shape:Solid
    Molecular weight:390.3

    Ref: TM-T21927

    1mg
    105.00€
    5mg
    325.00€
    10mg
    444.00€
  • DH97

    CAS:
    MT2 melatonin receptor antagonist
    Formula:C22H26N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:334.45

    Ref: TM-T22721

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A68930

    CAS:
    A 68930 is a dopamine D-1 receptor antagonist. A 68930 inhibits NLRP3 inflammasome activity.
    Formula:C16H17NO3
    Color and Shape:Solid
    Molecular weight:271.31

    Ref: TM-T26432

    25mg
    3,492.00€
    50mg
    5,239.00€
    100mg
    7,857.00€
  • LY 225910

    CAS:
    LY 225910 is a CCK2 receptor antagonist.
    Formula:C27H24BrN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:502.4

    Ref: TM-T22941

    10mg
    470.00€
    50mg
    1,918.00€
  • MS 245 oxalate

    CAS:
    MS 245 oxalate is a 5-HT6 antagonist.
    Formula:C21H24N2O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.49

    Ref: TM-T23029

    1mg
    124.00€
    5mg
    462.00€
    10mg
    695.00€
  • CAY10535

    CAS:
    CAY10535 is a selective TPβ antagonist (IC50 = 99 nM for TPβ vs 1970 nM for TPα), weakly affects platelets (IC50 = 985 nM).
    Formula:C18H21N3O7S
    Color and Shape:Solid
    Molecular weight:423.44

    Ref: TM-T36550

    1mg
    118.00€
    5mg
    515.00€
    10mg
    888.00€
    25mg
    1,882.00€
  • N-Salicyloyltryptamine

    CAS:
    N-Salicyloyltryptamine (STP): a tryptamine with anticonvulsant, anti-inflammatory, analgesic effects; inhibits Na+, Ca2+, K+ channels (IC50 34.6 μM).
    Formula:C17H16N2O2
    Color and Shape:Solid
    Molecular weight:280.32

    Ref: TM-T60526

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB 235375

    CAS:
    SB 235375 is a potent and selective antagonist of neurokinin-3 receptor with a low central nervous system-penetrant.
    Formula:C27H24N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.49

    Ref: TM-T28676

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A1AR antagonist 6

    CAS:
    A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].
    Formula:C17H15N3O2
    Color and Shape:Solid
    Molecular weight:293.32

    Ref: TM-T60615

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SKF-83566 hydrobromide

    CAS:
    D1-like dopamine receptor antagonist
    Formula:C17H19BrClNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.7

    Ref: TM-T23362

    5mg
    200.00€
    10mg
    314.00€
    25mg
    620.00€
  • Lu AA41063

    CAS:
    Lu AA41063 is a potent and selective antagonist of the hA2A receptor.
    Formula:C16H17F2N3O2S
    Color and Shape:Solid
    Molecular weight:353.39

    Ref: TM-T24418

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Todralazine

    CAS:
    Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.
    Formula:C11H12N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:232.24

    Ref: TM-T17112

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Lexipafant

    CAS:
    Lexipafant is a platelet-activating factor (PAF) receptor antagonist.
    Formula:C23H30N4O4S
    Color and Shape:Solid
    Molecular weight:458.57

    Ref: TM-T27821

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • T 82

    CAS:
    T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.
    Formula:C56H62N6O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:947.146

    Ref: TM-T13239

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€