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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • Tei 6472

    CAS:
    Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.
    Formula:C32H39N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:545.67

    Ref: TM-T26255

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PGlu-3-methyl-His-Pro-NH2 TFA


    PGlu-3-methyl-His-Pro-NH2 TFA boosts TRH receptor binding & TSH release.
    Formula:C19H25F3N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:490.43

    Ref: TM-T19511

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bepafant

    CAS:
    Bepafant: a PAF antagonist with anti-inflammatory properties; induces apoptosis in PTEN-positive NB4, KG1, NB4-MR4 cells, not in PTEN-negative THP1, U937.
    Formula:C23H22ClN5O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:467.97

    Ref: TM-T26775

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KSCM-5

    CAS:
    KSCM-5 is a sigma receptor ligand.
    Formula:C24H28N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.49

    Ref: TM-T25586

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CI-1015

    CAS:
    CI-1015 is a CCK-B receptor antagonist with oral activity.
    Formula:C29H39N3O4
    Color and Shape:Solid
    Molecular weight:493.64

    Ref: TM-T27014

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • hGPR91 antagonist 3

    CAS:
    hGPR91 antagonist 3 is an hGPR91 antagonist. hGPR91 antagonist 3 can be used to study diseases in hypertension and retinal angiogenesis.
    Formula:C23H18F4N4O2
    Purity:98.82% - 99.347%
    Color and Shape:Solid
    Molecular weight:458.41

    Ref: TM-T62858

    1mg
    123.00€
    5mg
    295.00€
    1mL*10mM (DMSO)
    299.00€
    10mg
    490.00€
    25mg
    792.00€
    50mg
    1,071.00€
    100mg
    1,468.00€
    200mg
    1,972.00€
  • CV-3988

    CAS:
    CV-3988 is a specific antagonist of PAF-R (platelet-activating factor receptor)(Ki = 0.872 μM).
    Formula:C28H53N2O7PS
    Color and Shape:Solid
    Molecular weight:592.77

    Ref: TM-T27101

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • 5-Nonyloxytryptamine oxalate

    CAS:
    5-HT1B agonist
    Formula:C21H32N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.49

    Ref: TM-T22524

    1mg
    112.00€
    5mg
    314.00€
    10mg
    421.00€
  • Flutonidine

    CAS:
    Flutonidine is an agonist of alpha2-Adrenergic receptor.
    Formula:C10H12FN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:193.22

    Ref: TM-T25433

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Gastrazole free acid

    CAS:
    Gastrazole is a CCK2 receptor antagonist potentially. It also used for the treatment of pancreatic cancer.
    Formula:C34H34FN5O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:643.66

    Ref: TM-T24085

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RP5063 Hydrochloride

    CAS:
    RP5063 Hydrochloride is a modulator of multimodal serotonin receptors.
    Formula:C22H26Cl3N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:486.82

    Ref: TM-T24736

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dacemazine hydrochloride

    CAS:
    Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.
    Formula:C16H17ClN2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:320.84

    Ref: TM-T23949

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dacopafant

    CAS:
    Dacopafant is an antagonist of platlet activationg factor receptor.
    Formula:C12H11N3OS
    Color and Shape:Solid
    Molecular weight:245.3

    Ref: TM-T23951

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EP3 antagonist 3

    CAS:
    EP3 antagonist 3, potent and selective oral, inhibited GR63799- or acetic acid-induced reduction in bladder capacity and PGE2-induced overactive bladder model.
    Formula:C21H18N2O4
    Color and Shape:Solid
    Molecular weight:362.38

    Ref: TM-T61357

    25mg
    915.00€
    50mg
    1,190.00€
    100mg
    1,848.00€
  • BN 50341

    CAS:
    BN 50341 is an inhibitor of antithrombotic platelet activating factor.
    Formula:C32H41ClN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.13

    Ref: TM-T26874

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • SKF 86466 hydrochloride

    CAS:
    SKF 86466 hydrochloride is an α2-adrenoceptor antagonist.
    Formula:C11H15Cl2N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:232.15

    Ref: TM-T23366

    1mg
    105.00€
    5mg
    355.00€
    10mg
    500.00€
  • KUL-7211

    CAS:
    KUL-7211 is an β2 and β3 adrenergic receptor agonist. KUL-7211 is a potent ureteral relaxant with a relatively small hypotensive effect.
    Formula:C19H23NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.39

    Ref: TM-T27754

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Embramine

    CAS:
    Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.
    Formula:C18H22BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.28

    Ref: TM-T11180

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cinitapride Hydrogen Tartrate

    CAS:
    Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptors
    Formula:C25H36N4O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:552.581

    Ref: TM-T22294

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB 258585 hydrochloride

    CAS:
    SB 258585 hydrochloride is a 5-HT6 receptor antagonist.
    Formula:C18H23ClIN3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:523.82

    Ref: TM-T23318

    1mg
    105.00€
    5mg
    379.00€
    10mg
    600.00€