
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Tei 6472
CAS:Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.Formula:C32H39N3O5Purity:98%Color and Shape:SolidMolecular weight:545.67PGlu-3-methyl-His-Pro-NH2 TFA
PGlu-3-methyl-His-Pro-NH2 TFA boosts TRH receptor binding & TSH release.Formula:C19H25F3N6O6Purity:98%Color and Shape:SolidMolecular weight:490.43Bepafant
CAS:Bepafant: a PAF antagonist with anti-inflammatory properties; induces apoptosis in PTEN-positive NB4, KG1, NB4-MR4 cells, not in PTEN-negative THP1, U937.Formula:C23H22ClN5O2SPurity:98%Color and Shape:SolidMolecular weight:467.97KSCM-5
CAS:KSCM-5 is a sigma receptor ligand.Formula:C24H28N2O2Purity:98%Color and Shape:SolidMolecular weight:376.49CI-1015
CAS:CI-1015 is a CCK-B receptor antagonist with oral activity.Formula:C29H39N3O4Color and Shape:SolidMolecular weight:493.64hGPR91 antagonist 3
CAS:hGPR91 antagonist 3 is an hGPR91 antagonist. hGPR91 antagonist 3 can be used to study diseases in hypertension and retinal angiogenesis.Formula:C23H18F4N4O2Purity:98.82% - 99.347%Color and Shape:SolidMolecular weight:458.41Ref: TM-T62858
1mg123.00€5mg295.00€1mL*10mM (DMSO)299.00€10mg490.00€25mg792.00€50mg1,071.00€100mg1,468.00€200mg1,972.00€CV-3988
CAS:CV-3988 is a specific antagonist of PAF-R (platelet-activating factor receptor)(Ki = 0.872 μM).Formula:C28H53N2O7PSColor and Shape:SolidMolecular weight:592.775-Nonyloxytryptamine oxalate
CAS:5-HT1B agonistFormula:C21H32N2O5Purity:98%Color and Shape:SolidMolecular weight:392.49Flutonidine
CAS:Flutonidine is an agonist of alpha2-Adrenergic receptor.Formula:C10H12FN3Purity:98%Color and Shape:SolidMolecular weight:193.22Gastrazole free acid
CAS:Gastrazole is a CCK2 receptor antagonist potentially. It also used for the treatment of pancreatic cancer.Formula:C34H34FN5O7Purity:98%Color and Shape:SolidMolecular weight:643.66RP5063 Hydrochloride
CAS:RP5063 Hydrochloride is a modulator of multimodal serotonin receptors.Formula:C22H26Cl3N3O3Purity:98%Color and Shape:SolidMolecular weight:486.82Dacemazine hydrochloride
CAS:Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.Formula:C16H17ClN2OSPurity:98%Color and Shape:SolidMolecular weight:320.84Dacopafant
CAS:Dacopafant is an antagonist of platlet activationg factor receptor.Formula:C12H11N3OSColor and Shape:SolidMolecular weight:245.3EP3 antagonist 3
CAS:EP3 antagonist 3, potent and selective oral, inhibited GR63799- or acetic acid-induced reduction in bladder capacity and PGE2-induced overactive bladder model.Formula:C21H18N2O4Color and Shape:SolidMolecular weight:362.38BN 50341
CAS:BN 50341 is an inhibitor of antithrombotic platelet activating factor.Formula:C32H41ClN2O4Purity:98%Color and Shape:SolidMolecular weight:553.13SKF 86466 hydrochloride
CAS:SKF 86466 hydrochloride is an α2-adrenoceptor antagonist.Formula:C11H15Cl2NPurity:98%Color and Shape:SolidMolecular weight:232.15KUL-7211
CAS:KUL-7211 is an β2 and β3 adrenergic receptor agonist. KUL-7211 is a potent ureteral relaxant with a relatively small hypotensive effect.Formula:C19H23NO5Purity:98%Color and Shape:SolidMolecular weight:345.39Embramine
CAS:Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.Formula:C18H22BrNOPurity:98%Color and Shape:SolidMolecular weight:348.28Cinitapride Hydrogen Tartrate
CAS:Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptorsFormula:C25H36N4O10Purity:98%Color and Shape:SolidMolecular weight:552.581SB 258585 hydrochloride
CAS:SB 258585 hydrochloride is a 5-HT6 receptor antagonist.Formula:C18H23ClIN3O3SPurity:98%Color and Shape:SolidMolecular weight:523.82
