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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • PF-04781340

    CAS:
    PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.
    Formula:C17H21N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.37

    Ref: TM-T24616

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AK-IN-1

    CAS:
    AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.
    Formula:C22H21N3O4
    Color and Shape:Solid
    Molecular weight:391.42

    Ref: TM-T73436

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Sequifenadine

    CAS:
    Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].
    Formula:C22H27NO
    Color and Shape:Solid
    Molecular weight:321.46

    Ref: TM-T60864

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • CCG-271423

    CAS:
    CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.
    Formula:C28H26N4O3
    Color and Shape:Solid
    Molecular weight:466.53

    Ref: TM-T62986

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BMS-193884

    CAS:
    BMS-193884 is an oral endothelin antagonist for the treatment of congestive heart failure (CHF) and pulmonary arterial hypertension.
    Formula:C20H17N3O4S
    Color and Shape:Solid
    Molecular weight:395.43

    Ref: TM-T30501

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ATC0065

    CAS:
    ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.
    Formula:C25H29BrF3N5O
    Color and Shape:Solid
    Molecular weight:552.43

    Ref: TM-T26676

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Acetylaszonalenin

    CAS:
    Acetylaszonalenin, from A. flavipes, is an NK1 receptor antagonist with a Ki of 170 μM, blocking substance P.
    Formula:C25H25N3O3
    Color and Shape:Solid
    Molecular weight:415.48

    Ref: TM-T71833

    500µg
    335.00€
    2500µg
    1,170.00€
  • (R)-(+)-8-Hydroxy-DPAT hydrobromide

    CAS:
    5-HT1A serotonin receptor agonist
    Formula:C16H26BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.29

    Ref: TM-T23218

    10mg
    735.00€
    50mg
    3,052.00€
  • VUF8507

    CAS:
    Vuf8507 is an allosteric regulator of adenosine receptor.
    Formula:C21H15N3O
    Color and Shape:Solid
    Molecular weight:325.36

    Ref: TM-T35086

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PD 81723

    CAS:
    Allosteric potentiator at the adenosine A1 receptor
    Formula:C14H12F3NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.31

    Ref: TM-T23130

    1mg
    To inquire
    5mg
    93.00€
    10mg
    133.00€
    25mg
    295.00€
    50mg
    480.00€
    100mg
    770.00€
  • GAT228

    CAS:
    GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].
    Formula:C22H18N2O2
    Color and Shape:Solid
    Molecular weight:342.39

    Ref: TM-T61105

    1mg
    118.00€
    10mg
    673.00€
  • MRS2179

    CAS:
    MRS2179: P2Y1 antagonist, Kb=100 nM, inactive on P2Y2/4/6 (to 30µM), inhibits ADP-induced platelet changes, prolongs bleeding in rodents.
    Formula:C11H17N5O9P2
    Color and Shape:Solid
    Molecular weight:425.23

    Ref: TM-T28099

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CI 1020

    CAS:
    endothelin-A receptor (ETA) antagonist
    Formula:C28H26O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:506.5

    Ref: TM-T22663

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Idremcinal

    CAS:
    Idremcinal is a motilin receptor agonist.
    Formula:C39H69NO12
    Color and Shape:Solid
    Molecular weight:743.96

    Ref: TM-T27584

    500µg
    304.00€
    1mg
    575.00€
  • CCG-273463

    CAS:
    CCG-273463: Potent GRK5 inhibitor (IC50: 9 nM), used for researching heart failure, hypertrophy, cancer.
    Formula:C26H25BrN4O3
    Color and Shape:Solid
    Molecular weight:521.41

    Ref: TM-T63640

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Lidanserin

    CAS:
    Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.
    Formula:C26H31FN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.53

    Ref: TM-T15754

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • PD-156707

    CAS:
    PD-156707 is a selective antagonist of endothelin A receptor.
    Formula:C28H26NaO9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:529.497

    Ref: TM-T28343

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ASP7657

    CAS:
    ASP7657 is a novel, potent, and selective prostaglandin EP4 receptor antagonist.
    Formula:C28H26F3N3O3
    Color and Shape:Solid
    Molecular weight:509.52

    Ref: TM-T71269

    1mg
    221.00€
    5mg
    982.00€
    10mg
    1,728.00€
    25mg
    3,808.00€
  • ICI 192605

    CAS:
    ICI 192605 is a potent thromboxane A2 receptor (TP receptor) antagonist.
    Formula:C22H23ClO5
    Color and Shape:Solid
    Molecular weight:402.87

    Ref: TM-T27575

    1mg
    105.00€
    5mg
    304.00€
    10mg
    530.00€
    25mg
    1,189.00€
  • AL-3138

    CAS:
    AL-3138 is a prostaglandin F2alpha (PGF2alpha) analogue which antagonizes FP prostanoid receptor-mediated inositol phosphates generation.
    Formula:C20H33FO4
    Color and Shape:Solid
    Molecular weight:356.47

    Ref: TM-T29813

    25mg
    1,369.00€