
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Formula:C17H21N3Purity:98%Color and Shape:SolidMolecular weight:267.37AK-IN-1
CAS:AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.Formula:C22H21N3O4Color and Shape:SolidMolecular weight:391.42Sequifenadine
CAS:Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].Formula:C22H27NOColor and Shape:SolidMolecular weight:321.46CCG-271423
CAS:CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.Formula:C28H26N4O3Color and Shape:SolidMolecular weight:466.53BMS-193884
CAS:BMS-193884 is an oral endothelin antagonist for the treatment of congestive heart failure (CHF) and pulmonary arterial hypertension.Formula:C20H17N3O4SColor and Shape:SolidMolecular weight:395.43ATC0065
CAS:ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.Formula:C25H29BrF3N5OColor and Shape:SolidMolecular weight:552.43Acetylaszonalenin
CAS:Acetylaszonalenin, from A. flavipes, is an NK1 receptor antagonist with a Ki of 170 μM, blocking substance P.Formula:C25H25N3O3Color and Shape:SolidMolecular weight:415.48(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:5-HT1A serotonin receptor agonistFormula:C16H26BrNOPurity:98%Color and Shape:SolidMolecular weight:328.29VUF8507
CAS:Vuf8507 is an allosteric regulator of adenosine receptor.Formula:C21H15N3OColor and Shape:SolidMolecular weight:325.36PD 81723
CAS:Allosteric potentiator at the adenosine A1 receptorFormula:C14H12F3NOSPurity:98%Color and Shape:SolidMolecular weight:299.31GAT228
CAS:GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].Formula:C22H18N2O2Color and Shape:SolidMolecular weight:342.39MRS2179
CAS:MRS2179: P2Y1 antagonist, Kb=100 nM, inactive on P2Y2/4/6 (to 30µM), inhibits ADP-induced platelet changes, prolongs bleeding in rodents.Formula:C11H17N5O9P2Color and Shape:SolidMolecular weight:425.23CI 1020
CAS:endothelin-A receptor (ETA) antagonistFormula:C28H26O9Purity:98%Color and Shape:SolidMolecular weight:506.5Idremcinal
CAS:Idremcinal is a motilin receptor agonist.Formula:C39H69NO12Color and Shape:SolidMolecular weight:743.96CCG-273463
CAS:CCG-273463: Potent GRK5 inhibitor (IC50: 9 nM), used for researching heart failure, hypertrophy, cancer.Formula:C26H25BrN4O3Color and Shape:SolidMolecular weight:521.41Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Formula:C26H31FN2O4Purity:98%Color and Shape:SolidMolecular weight:454.53PD-156707
CAS:PD-156707 is a selective antagonist of endothelin A receptor.Formula:C28H26NaO9Purity:98%Color and Shape:SolidMolecular weight:529.497ASP7657
CAS:ASP7657 is a novel, potent, and selective prostaglandin EP4 receptor antagonist.Formula:C28H26F3N3O3Color and Shape:SolidMolecular weight:509.52ICI 192605
CAS:ICI 192605 is a potent thromboxane A2 receptor (TP receptor) antagonist.Formula:C22H23ClO5Color and Shape:SolidMolecular weight:402.87AL-3138
CAS:AL-3138 is a prostaglandin F2alpha (PGF2alpha) analogue which antagonizes FP prostanoid receptor-mediated inositol phosphates generation.Formula:C20H33FO4Color and Shape:SolidMolecular weight:356.47
