
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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AVN-322
CAS:AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.Formula:C17H20ClN5O2SPurity:>99.99%Color and Shape:SolidMolecular weight:393.89Etrasimod arginine
CAS:Etrasimod arginine is used in the Treatment of Autoimmune and Inflammatory Diseases.Formula:C32H40F3N5O5Color and Shape:SolidMolecular weight:631.69Tilisolol HCl
CAS:Tilisolol, a nonselective beta-blocker, dilates dog coronary arteries via ATP-sensitive K(+) channels.Formula:C17H25ClN2O3Purity:98%Color and Shape:SolidMolecular weight:340.85(R)-PF-06256142
CAS:(R)-PF-06256142: low-activity R enantiomer of a potent, selective D1 agonist reducing receptor desensitization.Formula:C21H16N4O2Color and Shape:SolidMolecular weight:356.38Clopenthixol
CAS:Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.Formula:C22H25ClN2OSColor and Shape:SolidMolecular weight:400.96Elzasonan
CAS:Elzasonan is a selective 5-hydroxytryptamine 1B receptor antagonist used to treat patients with major depressive disorder and obsessive compulsive disorder.Formula:C22H23Cl2N3OSColor and Shape:SolidMolecular weight:448.41MK-0249
CAS:MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
Formula:C23H24F3N3O2Purity:99.90%Color and Shape:SolidMolecular weight:431.45H3 receptor-MO-1
CAS:H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.Formula:C20H27N3O2Purity:99.11%Color and Shape:SolidMolecular weight:341.45Rocastine
CAS:Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.Formula:C13H19N3OSPurity:98.26%Color and Shape:SolidMolecular weight:265.37QF0301B
CAS:QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.Formula:C23H28N2O2Purity:>99.99%Color and Shape:SolidMolecular weight:364.48Tulopafant
CAS:Tulopafant (RP 59227) is a potent platelet-activating factor (PAF) antagonist that increases capillary patency and prolongs allograft heart survival.Formula:C25H19N3O2SPurity:99.38%Color and Shape:SolidMolecular weight:425.5ML179
CAS:ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.Formula:C21H25F3N4O2Purity:99.77%Color and Shape:SolidMolecular weight:422.44Ref: TM-T8954
1mg34.00€5mg75.00€1mL*10mM (DMSO)92.00€10mg110.00€25mg220.00€50mg321.00€100mg469.00€200mg645.00€KY 234
CAS:KY 234 is a thromboxane synthetase antagonist.Formula:C33H35N5O2Color and Shape:SolidMolecular weight:533.676Romifidine
CAS:Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.Formula:C9H9BrFN3Color and Shape:SolidMolecular weight:258.09Paltusotine HCl
CAS:Paltusotine, also known as CRN00808, is a somatostatin receptor agonist.Formula:C27H24Cl2F2N4OColor and Shape:SolidMolecular weight:529.41Isoproterenol-d7 HCl
CAS:Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.Formula:C11H18ClNO3Color and Shape:SolidMolecular weight:254.76CM304
CAS:CM304 is a highly selective sigma-1 receptor antagonist.Formula:C18H26ClFN2OSColor and Shape:SolidMolecular weight:372.93Pd 158771
CAS:Pd 158771 is a D2 and 5-HT1A agonist.Formula:C22H31N5Color and Shape:SolidMolecular weight:365.52SC 51089
CAS:SC 51089 is a somatic PGE2 antagonist with anti-injurious activity and may rescue memory loss.Formula:C22H20Cl2N4O3Purity:98%Color and Shape:SolidMolecular weight:459.33CCK-A receptor inhibitor 1
CAS:CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the studyFormula:C25H35NO6SPurity:99.47%Color and Shape:SolidMolecular weight:477.61
