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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • AVN-322

    CAS:
    AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.
    Formula:C17H20ClN5O2S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:393.89

    Ref: TM-T26691

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • Etrasimod arginine

    CAS:
    Etrasimod arginine is used in the Treatment of Autoimmune and Inflammatory Diseases.
    Formula:C32H40F3N5O5
    Color and Shape:Solid
    Molecular weight:631.69

    Ref: TM-T31726

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
    500mg
    3,137.00€
  • Tilisolol HCl

    CAS:
    Tilisolol, a nonselective beta-blocker, dilates dog coronary arteries via ATP-sensitive K(+) channels.
    Formula:C17H25ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:340.85

    Ref: TM-T28977

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-PF-06256142

    CAS:
    (R)-PF-06256142: low-activity R enantiomer of a potent, selective D1 agonist reducing receptor desensitization.
    Formula:C21H16N4O2
    Color and Shape:Solid
    Molecular weight:356.38

    Ref: TM-T72744

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,250.00€
  • Clopenthixol

    CAS:
    Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
    Formula:C22H25ClN2OS
    Color and Shape:Solid
    Molecular weight:400.96

    Ref: TM-T68193

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Elzasonan

    CAS:
    Elzasonan is a selective 5-hydroxytryptamine 1B receptor antagonist used to treat patients with major depressive disorder and obsessive compulsive disorder.
    Formula:C22H23Cl2N3OS
    Color and Shape:Solid
    Molecular weight:448.41

    Ref: TM-T69364

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MK-0249

    CAS:

    MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).

    Formula:C23H24F3N3O2
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:431.45

    Ref: TM-T12054

    1mg
    227.00€
    5mg
    562.00€
    10mg
    815.00€
    25mg
    1,206.00€
    50mg
    1,605.00€
    100mg
    2,175.00€
    200mg
    2,822.00€
  • H3 receptor-MO-1

    CAS:
    H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.
    Formula:C20H27N3O2
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:341.45

    Ref: TM-T10499

    1mg
    630.00€
    5mg
    1,620.00€
  • Rocastine

    CAS:
    Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.
    Formula:C13H19N3OS
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:265.37

    Ref: TM-T16778

    1mg
    630.00€
    5mg
    1,333.00€
  • QF0301B

    CAS:
    QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.
    Formula:C23H28N2O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:364.48

    Ref: TM-T10100

    1mg
    630.00€
    5mg
    1,620.00€
  • Tulopafant

    CAS:
    Tulopafant (RP 59227) is a potent platelet-activating factor (PAF) antagonist that increases capillary patency and prolongs allograft heart survival.
    Formula:C25H19N3O2S
    Purity:99.38%
    Color and Shape:Solid
    Molecular weight:425.5

    Ref: TM-T17178

    1mg
    630.00€
    5mg
    1,620.00€
  • ML179

    CAS:
    ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.
    Formula:C21H25F3N4O2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:422.44

    Ref: TM-T8954

    1mg
    34.00€
    5mg
    75.00€
    1mL*10mM (DMSO)
    92.00€
    10mg
    110.00€
    25mg
    220.00€
    50mg
    321.00€
    100mg
    469.00€
    200mg
    645.00€
  • KY 234

    CAS:
    KY 234 is a thromboxane synthetase antagonist.
    Formula:C33H35N5O2
    Color and Shape:Solid
    Molecular weight:533.676

    Ref: TM-T70241

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Romifidine

    CAS:
    Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.
    Formula:C9H9BrFN3
    Color and Shape:Solid
    Molecular weight:258.09

    Ref: TM-T26119

    1mg
    63.00€
    5mg
    130.00€
    10mg
    178.00€
    25mg
    305.00€
    50mg
    447.00€
    100mg
    655.00€
    500mg
    1,333.00€
  • Paltusotine HCl

    CAS:
    Paltusotine, also known as CRN00808, is a somatostatin receptor agonist.
    Formula:C27H24Cl2F2N4O
    Color and Shape:Solid
    Molecular weight:529.41

    Ref: TM-T69836

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Isoproterenol-d7 HCl

    CAS:
    Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.
    Formula:C11H18ClNO3
    Color and Shape:Solid
    Molecular weight:254.76

    Ref: TM-T69598

    1mg
    359.00€
  • CM304

    CAS:
    CM304 is a highly selective sigma-1 receptor antagonist.
    Formula:C18H26ClFN2OS
    Color and Shape:Solid
    Molecular weight:372.93

    Ref: TM-T71949

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Pd 158771

    CAS:
    Pd 158771 is a D2 and 5-HT1A agonist.
    Formula:C22H31N5
    Color and Shape:Solid
    Molecular weight:365.52

    Ref: TM-T70081

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SC 51089

    CAS:
    SC 51089 is a somatic PGE2 antagonist with anti-injurious activity and may rescue memory loss.
    Formula:C22H20Cl2N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.33

    Ref: TM-T23331

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CCK-A receptor inhibitor 1

    CAS:
    CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the study
    Formula:C25H35NO6S
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:477.61

    Ref: TM-T12404

    1mg
    630.00€
    5mg
    1,620.00€