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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • CP-195543

    CAS:
    CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.
    Formula:C24H19F3O4
    Color and Shape:Solid
    Molecular weight:428.4

    Ref: TM-T31042

    5mg
    3,445.00€
  • MAT2A-IN-1

    CAS:
    MAT2A-IN-1 suppresses MAT2A, key for MTAP-deficient cancer cell growth; studied for gastric, colon, liver, pancreatic cancers.
    Formula:C29H28F2N6O4
    Color and Shape:Solid
    Molecular weight:562.57

    Ref: TM-T63975

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A 55453

    CAS:
    A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.
    Formula:C25H32N6O3
    Color and Shape:Solid
    Molecular weight:464.56

    Ref: TM-T26421

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS2298

    CAS:
    MRS2298, a potent antagonists of the P2Y 1 receptor, has antiaggregatory activity in human platelets.
    Formula:C10H16ClN5O8P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.66

    Ref: TM-T28100

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • FRG8701

    CAS:
    FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
    Formula:C22H30N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:418.55

    Ref: TM-T11324

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • WB403

    CAS:
    WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.
    Formula:C19H19BrN2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.34

    Ref: TM-T29154

    5mg
    110.00€
    10mg
    168.00€
    25mg
    338.00€
    50mg
    533.00€
    100mg
    2,375.00€
  • MRS1186

    CAS:
    MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).
    Formula:C16H12ClN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:341.75

    Ref: TM-T16138

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PD-135666

    CAS:
    PD-135666 is an antagonist of CCK receptor.
    Formula:C33H39N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:557.68

    Ref: TM-T28340

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • S-777469

    CAS:
    S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.
    Formula:C23H27FN2O4
    Color and Shape:Solid
    Molecular weight:414.47

    Ref: TM-T62132

    25mg
    1,108.00€
    50mg
    1,449.00€
    100mg
    2,385.00€
  • CB2 receptor agonist 3

    CAS:
    GP 2A is a selective agonist of CB2 receptor.
    Formula:C24H23Cl2N3O
    Color and Shape:Solid
    Molecular weight:440.36

    Ref: TM-T24097

    25mg
    690.00€
    50mg
    898.00€
    100mg
    1,566.00€
  • ATL-801

    CAS:
    ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.
    Formula:C24H25N7O3
    Color and Shape:Solid
    Molecular weight:459.5

    Ref: TM-T26680

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Remogliflozin

    CAS:
    Remogliflozin is an effective sodium-glucose transporter 2 inhibitor (Kis = 12.4 and 26 nM for human and rat SGLT2, respectively).
    Formula:C23H34N2O7
    Color and Shape:Solid
    Molecular weight:450.53

    Ref: TM-T24708

    500µg
    157.00€
    1mg
    284.00€
    5mg
    1,288.00€
    10mg
    2,332.00€
  • Benzatropine

    CAS:
    Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.
    Formula:C21H25NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.43

    Ref: TM-T23781

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • γ-Linolenic acid ethyl ester

    CAS:
    γ-Linolenic acid ethyl ester (Ethyl γ-linolenate) is a leukotriene B 4 receptor 4 (LTB 4 ) antagonist which has a potential anti-inflammatory effect[1].
    Formula:C20H34O2
    Color and Shape:Solid
    Molecular weight:306.48

    Ref: TM-T41235

    50mg
    114.00€
    100mg
    208.00€
    250mg
    489.00€
    1g
    1,288.00€
  • MAT2A-IN-3

    CAS:
    MAT2A-IN-3: potent MAT2A inhibitor, hinders MTAP-deficient cancer cell growth, potential for cancer research.
    Formula:C24H16F5N5O3
    Color and Shape:Solid
    Molecular weight:517.41

    Ref: TM-T63603

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5-HT2A receptor agonist-2

    CAS:
    Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.
    Formula:C20H21ClN2O3
    Color and Shape:Solid
    Molecular weight:372.85

    Ref: TM-T61507

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Alaproclate (hydrochloride)

    CAS:
    Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.
    Formula:C13H19Cl2NO2
    Color and Shape:Solid
    Molecular weight:292.2

    Ref: TM-T36521

    5mg
    219.00€
    10mg
    378.00€
  • Edivoxetine

    CAS:
    Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.
    Formula:C18H26FNO4
    Color and Shape:Solid
    Molecular weight:339.4

    Ref: TM-T31604

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ChemR23-IN-1

    CAS:
    ChemR23-IN-1 inhibits human and mouse ChemR23 (IC50: 38 nM, 100 nM) and stops CAL-1 chemotaxis induced by Chemerin in vitro.
    Formula:C28H29N7O2
    Color and Shape:Solid
    Molecular weight:495.58

    Ref: TM-T63347

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • BGC-20-1531 free base

    CAS:
    BGC-20-1531 (PGN 1531) free base is a selective and potent prostaglandin EP4 receptor antagonist (pKB: 7.6) that exhibits potential for migraine research.
    Formula:C26H24N2O6S
    Color and Shape:Solid
    Molecular weight:492.54

    Ref: TM-T63316

    25mg
    1,026.00€
    50mg
    1,341.00€
    100mg
    2,197.00€