
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
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Dipiproverine
CAS:Dipiproverine is an alpha-amino acid ester, an antispasmodic compound. It is used as an anticholinergic drug.Formula:C20H30N2O2Color and Shape:SolidMolecular weight:330.46Ipramidil
CAS:Ipramidil (C80-1324) reveals marked dilator activity in the coronary circulation of isolated working hearts.Formula:C10H16N4O4Purity:98%Color and Shape:SolidMolecular weight:256.26KLS-13019
CAS:KLS-13019 is a highly effective and orally active GPR55 receptor antagonist, neuroprotective can reverse chemotherapy-induced peripheral neuropathy (CIPN).Formula:C22H29NO3Purity:>99.99% - >99.99%Color and Shape:SolidMolecular weight:355.47SKF-82958
CAS:SKF 82958 is a D1/D5 receptor full agonist.Formula:C19H20ClNO2Purity:98%Color and Shape:SolidMolecular weight:329.82MC-4R Agonist 1
CAS:MC-4R Agonist 1 is an agonist of human melanocortin-4 receptor (MC-4R) and can be used in the research of sexual dysfunction, obesity, and diabetes.Formula:C30H38ClF2N3O2Purity:98%Color and Shape:SolidMolecular weight:546.09MRE3008F20
CAS:MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.Formula:C21H20N8O3Purity:97.29%Color and Shape:SolidMolecular weight:432.44GSK1059865
CAS:GSK1059865 is a potent antagonist of the orexin 1 receptor.Formula:C20H23BrFN3O2Color and Shape:SolidMolecular weight:436.32RXFP3 agonist 1
CAS:RXFP3 agonist 1 is a nonpeptide RXFP3 agonist ( EC 50 =6937 nM) [1].Formula:C18H18ClN5Color and Shape:SolidMolecular weight:339.82S-1-Propenyl-L-cysteine
CAS:S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensiveFormula:C6H11NO2SPurity:98%Color and Shape:SolidMolecular weight:161.22MJ 15
CAS:MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.Formula:C23H17Cl3N4OPurity:99.63%Color and Shape:SolidMolecular weight:471.77Ramixotidine
CAS:Ramixotidine is a competitive antagonist of histamine H2-receptor.Formula:C16H21N3O3SPurity:98%Color and Shape:SolidMolecular weight:335.42Blonanserin HCl
CAS:Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.Formula:C23H32Cl2FN3Purity:98%Color and Shape:SolidMolecular weight:440.42CCK-B Receptor Antagonist 2
CAS:CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).Formula:C27H28N6O3Color and Shape:SolidMolecular weight:484.55CI-943
CAS:CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.Formula:C12H17N5Purity:98%Color and Shape:SolidMolecular weight:231.3RUSKI-201 dihydrochloride
CAS:RUSKI-201 dihydrochloride: potent Hhat inhibitor (IC50: 0.20 μM), blocks Hh signaling, and inhibits Hh palmitoylation.Formula:C20H29Cl2N3OSColor and Shape:SolidMolecular weight:430.43PPTN
CAS:PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 pM), with anti-inflammatory and immune activity.Formula:C29H24F3NO2Purity:99.86%Color and Shape:SolidMolecular weight:475.5Clovoxamine
CAS:Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant and anticonvulsant activity.Formula:C14H21ClN2O2Purity:99.44% - 99.75%Color and Shape:SolidMolecular weight:284.78A2ti-2
CAS:A2ti-2: selective A2/S100A10 inhibitor, IC50 230 μM, with antiviral action against HPV16.Formula:C18H18N4O2SPurity:99.98%Color and Shape:SolidMolecular weight:354.43Ref: TM-T36433
1mg92.00€5mg219.00€1mL*10mM (DMSO)241.00€10mg330.00€25mg643.00€50mg888.00€100mg1,224.00€500mg2,457.00€IMMH001
CAS:IMMH001/SYL930: Oral S1P1 receptor agonist; lowers IL-1β, IL-5, IL-18, IP10, CCL3, CCL5; for RA research.Formula:C23H28N2O3Color and Shape:SolidMolecular weight:380.48L 646462
CAS:L 646462 is an antidopaminergic agent.Formula:C27H27N3O4Purity:98%Color and Shape:SolidMolecular weight:457.52
