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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6012 products of "GPCR/G-Protein"

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  • Dipiproverine

    CAS:
    Dipiproverine is an alpha-amino acid ester, an antispasmodic compound. It is used as an anticholinergic drug.
    Formula:C20H30N2O2
    Color and Shape:Solid
    Molecular weight:330.46

    Ref: TM-T25339

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ipramidil

    CAS:
    Ipramidil (C80-1324) reveals marked dilator activity in the coronary circulation of isolated working hearts.
    Formula:C10H16N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:256.26

    Ref: TM-T13588

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KLS-13019

    CAS:
    KLS-13019 is a highly effective and orally active GPR55 receptor antagonist, neuroprotective can reverse chemotherapy-induced peripheral neuropathy (CIPN).
    Formula:C22H29NO3
    Purity:>99.99% - >99.99%
    Color and Shape:Solid
    Molecular weight:355.47

    Ref: TM-T32402

    1mg
    485.00€
    5mg
    1,084.00€
  • SKF-82958

    CAS:
    SKF 82958 is a D1/D5 receptor full agonist.
    Formula:C19H20ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.82

    Ref: TM-T16893

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MC-4R Agonist 1

    CAS:
    MC-4R Agonist 1 is an agonist of human melanocortin-4 receptor (MC-4R) and can be used in the research of sexual dysfunction, obesity, and diabetes.
    Formula:C30H38ClF2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:546.09

    Ref: TM-T10230

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRE3008F20

    CAS:
    MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.
    Formula:C21H20N8O3
    Purity:97.29%
    Color and Shape:Solid
    Molecular weight:432.44

    Ref: TM-T16132

    1mg
    66.00€
    2mg
    96.00€
    5mg
    144.00€
    10mg
    205.00€
    25mg
    349.00€
    50mg
    512.00€
  • GSK1059865

    CAS:
    GSK1059865 is a potent antagonist of the orexin 1 receptor.
    Formula:C20H23BrFN3O2
    Color and Shape:Solid
    Molecular weight:436.32

    Ref: TM-T11477

    1mg
    69.00€
    5mg
    147.00€
    1mL*10mM (DMSO)
    164.00€
    10mg
    230.00€
  • RXFP3 agonist 1

    CAS:
    RXFP3 agonist 1 is a nonpeptide RXFP3 agonist ( EC 50 =6937 nM) [1].
    Formula:C18H18ClN5
    Color and Shape:Solid
    Molecular weight:339.82

    Ref: TM-T61079

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • S-1-Propenyl-L-cysteine

    CAS:
    S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensive
    Formula:C6H11NO2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:161.22

    Ref: TM-T12789

    25mg
    999.00€
    50mg
    1,305.00€
    100mg
    2,088.00€
  • MJ 15

    CAS:
    MJ 15 is a CB1 receptor antagonist with specificity for the study of obesity-induced diseases.
    Formula:C23H17Cl3N4O
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:471.77

    Ref: TM-T22984

    1mg
    34.00€
    5mg
    105.00€
    10mg
    164.00€
    25mg
    334.00€
    50mg
    537.00€
    100mg
    863.00€
    500mg
    1,728.00€
  • Ramixotidine

    CAS:
    Ramixotidine is a competitive antagonist of histamine H2-receptor.
    Formula:C16H21N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:335.42

    Ref: TM-T26039

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Blonanserin HCl

    CAS:
    Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.
    Formula:C23H32Cl2FN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.42

    Ref: TM-T1180L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CCK-B Receptor Antagonist 2

    CAS:
    CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).
    Formula:C27H28N6O3
    Color and Shape:Solid
    Molecular weight:484.55

    Ref: TM-T10707

    5mg
    401.00€
    25mg
    1,288.00€
    50mg
    1,674.00€
    100mg
    2,250.00€
  • CI-943

    CAS:
    CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.
    Formula:C12H17N5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:231.3

    Ref: TM-T14963

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • RUSKI-201 dihydrochloride

    CAS:
    RUSKI-201 dihydrochloride: potent Hhat inhibitor (IC50: 0.20 μM), blocks Hh signaling, and inhibits Hh palmitoylation.
    Formula:C20H29Cl2N3OS
    Color and Shape:Solid
    Molecular weight:430.43

    Ref: TM-T62388

    1mg
    197.00€
    5mg
    862.00€
    10mg
    1,521.00€
  • PPTN

    CAS:
    PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 pM), with anti-inflammatory and immune activity.
    Formula:C29H24F3NO2
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:475.5

    Ref: TM-T12530

    1mg
    47.00€
    5mg
    92.00€
    10mg
    152.00€
    25mg
    289.00€
    50mg
    432.00€
    100mg
    618.00€
    200mg
    859.00€
  • Clovoxamine

    CAS:
    Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant and anticonvulsant activity.
    Formula:C14H21ClN2O2
    Purity:99.44% - 99.75%
    Color and Shape:Solid
    Molecular weight:284.78

    Ref: TM-T27047

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • A2ti-2

    CAS:
    A2ti-2: selective A2/S100A10 inhibitor, IC50 230 μM, with antiviral action against HPV16.
    Formula:C18H18N4O2S
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:354.43

    Ref: TM-T36433

    1mg
    92.00€
    5mg
    219.00€
    1mL*10mM (DMSO)
    241.00€
    10mg
    330.00€
    25mg
    643.00€
    50mg
    888.00€
    100mg
    1,224.00€
    500mg
    2,457.00€
  • IMMH001

    CAS:
    IMMH001/SYL930: Oral S1P1 receptor agonist; lowers IL-1β, IL-5, IL-18, IP10, CCL3, CCL5; for RA research.
    Formula:C23H28N2O3
    Color and Shape:Solid
    Molecular weight:380.48

    Ref: TM-T61621

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L 646462

    CAS:
    L 646462 is an antidopaminergic agent.
    Formula:C27H27N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.52

    Ref: TM-T24302

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€