
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
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PD 119819
CAS:PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.Formula:C21H25Cl2N3O3Purity:98%Color and Shape:SolidMolecular weight:438.35BI-L 239
CAS:BI-L 239 is an inhibition of 5-lipoxygenase products that cause bronchoconstriction.Formula:C16H15FOColor and Shape:SolidMolecular weight:242.29Bifeprunox Mesylate
CAS:Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.Formula:C25H27N3O5SPurity:98%Color and Shape:SolidMolecular weight:481.56Penbutolol
CAS:Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.Formula:C18H29NO2Purity:98%Color and Shape:SolidMolecular weight:291.43DMP 696
CAS:DMP 696 is a selective antagonist of corticotropin-releasing hormone receptor 1. It is used for the treatment of anxiety and depression.Formula:C18H21Cl2N5O2Purity:98%Color and Shape:SolidMolecular weight:410.3IMTPPE
CAS:IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.Formula:C20H27N3O2SColor and Shape:SolidMolecular weight:373.51JMV3002
CAS:JMV3002, a ghrelin receptor foe, blocks hexarelin-induced eating in rats by up to 98% without affecting growth hormone release.Formula:C35H34N6O3Color and Shape:SolidMolecular weight:586.68Tiamenidine
CAS:Tiamenidine is an antagonist of centrally-acting alpha1 adrenergic receptor.Formula:C8H10ClN3SPurity:98%Color and Shape:SolidMolecular weight:215.7Abanoquil
CAS:Abanoquil is an antagonist of alpha-1 adrenoceptor.Formula:C22H25N3O4Color and Shape:SolidMolecular weight:395.45GTS-21
CAS:GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.Formula:C19H20N2O2Purity:98%Color and Shape:SolidMolecular weight:308.37U-101958 Maleate
CAS:U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.Formula:C25H33N3O5Purity:98%Color and Shape:SolidMolecular weight:455.55Zinterol
CAS:Zinterol is a potent and selective agonist of β2-adrenoceptor. Zinterol increases ICa in a concentration-dependent manner(EC50 of 2.2 nM).Formula:C19H26N2O4SPurity:98%Color and Shape:SolidMolecular weight:378.49Prostaglandin D2
CAS:Prostaglandin D2 (PGD2) is one of the major PGs actively produced in the brain of various mammals,and is a potent endogenous sleep promoting substances.Formula:C20H32O5Purity:>99.99%Color and Shape:SolidMolecular weight:352.47(2R,3R)-E1R
CAS:(2R,3R)-E1R is an enantiomer of E1R. (2R,3R)-E1R is a sigma-1 receptor positive allosteric modulator for the treatment of cognition/memory disorders.Formula:C13H16N2O2Purity:98%Color and Shape:SolidMolecular weight:232.28OUP-186
CAS:OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.Formula:C19H30ClN3SColor and Shape:SolidMolecular weight:367.98PF-04628935
CAS:PF-04628935: potent GHS-R1a antagonist/inverse agonist, IC50=4.6 nM, orally bioavailable, brain penetrant.Formula:C24H26ClN7OSPurity:98%Color and Shape:SolidMolecular weight:496.03Clenproperol
CAS:Clenproperol is a β2-adrenergic agonist.Formula:C11H16Cl2N2OColor and Shape:SolidMolecular weight:263.16Benzamide Derivative 1
CAS:Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.Formula:C22H34ClN3O3Purity:>99.99%Color and Shape:SolidMolecular weight:423.98HAMI 3379
CAS:HAMI 3379 (HAMI3379) is a CysLT2 antagonist that attenuates brain damage and inhibits microglia inflammation following focal cerebral ischemia in rats.Formula:C34H45NO8Purity:99.75%Color and Shape:SolidMolecular weight:595.72GR 128107
CAS:GR 128107 is an antagonist of melatonin receptor.Formula:C16H20N2O2Color and Shape:SolidMolecular weight:272.34
