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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6012 products of "GPCR/G-Protein"

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  • PD 119819

    CAS:
    PD 119819 is a heterocyclic piperazine. PD 119819 is an extremely selective DA autoreceptor agonist.
    Formula:C21H25Cl2N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.35

    Ref: TM-T28318

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BI-L 239

    CAS:
    BI-L 239 is an inhibition of 5-lipoxygenase products that cause bronchoconstriction.
    Formula:C16H15FO
    Color and Shape:Solid
    Molecular weight:242.29

    Ref: TM-T26811

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bifeprunox Mesylate

    CAS:
    Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.
    Formula:C25H27N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.56

    Ref: TM-T26807

    1mg
    114.00€
  • Penbutolol

    CAS:
    Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.
    Formula:C18H29NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:291.43

    Ref: TM-T12402L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DMP 696

    CAS:
    DMP 696 is a selective antagonist of corticotropin-releasing hormone receptor 1. It is used for the treatment of anxiety and depression.
    Formula:C18H21Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.3

    Ref: TM-T15145

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • IMTPPE

    CAS:
    IMTPPE inhibits transcriptional activity and protein level of AR in C4-2 prostate cancer cells. It also inhibits AR-target gene expression.
    Formula:C20H27N3O2S
    Color and Shape:Solid
    Molecular weight:373.51

    Ref: TM-T27601

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JMV3002

    CAS:
    JMV3002, a ghrelin receptor foe, blocks hexarelin-induced eating in rats by up to 98% without affecting growth hormone release.
    Formula:C35H34N6O3
    Color and Shape:Solid
    Molecular weight:586.68

    Ref: TM-T35793

    100µg
    195.00€
    500µg
    845.00€
    1mg
    1,485.00€
    5mg
    6,193.00€
  • Tiamenidine

    CAS:
    Tiamenidine is an antagonist of centrally-acting alpha1 adrenergic receptor.
    Formula:C8H10ClN3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:215.7

    Ref: TM-T28970

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Abanoquil

    CAS:
    Abanoquil is an antagonist of alpha-1 adrenoceptor.
    Formula:C22H25N3O4
    Color and Shape:Solid
    Molecular weight:395.45

    Ref: TM-T26507

    25mg
    858.00€
    50mg
    1,116.00€
    100mg
    1,449.00€
  • GTS-21

    CAS:
    GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.
    Formula:C19H20N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:308.37

    Ref: TM-T19933

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • U-101958 Maleate

    CAS:
    U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.
    Formula:C25H33N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:455.55

    Ref: TM-T29030

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Zinterol

    CAS:
    Zinterol is a potent and selective agonist of β2-adrenoceptor. Zinterol increases ICa in a concentration-dependent manner(EC50 of 2.2 nM).
    Formula:C19H26N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:378.49

    Ref: TM-T13399

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Prostaglandin D2

    CAS:
    Prostaglandin D2 (PGD2) is one of the major PGs actively produced in the brain of various mammals,and is a potent endogenous sleep promoting substances.
    Formula:C20H32O5
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:352.47

    Ref: TM-T13831

    100µg
    290.00€
  • (2R,3R)-E1R

    CAS:
    (2R,3R)-E1R is an enantiomer of E1R. (2R,3R)-E1R is a sigma-1 receptor positive allosteric modulator for the treatment of cognition/memory disorders.
    Formula:C13H16N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:232.28

    Ref: TM-T10093

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • OUP-186

    CAS:
    OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.
    Formula:C19H30ClN3S
    Color and Shape:Solid
    Molecular weight:367.98

    Ref: TM-T28275

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-04628935

    CAS:
    PF-04628935: potent GHS-R1a antagonist/inverse agonist, IC50=4.6 nM, orally bioavailable, brain penetrant.
    Formula:C24H26ClN7OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:496.03

    Ref: TM-T28366

    25mg
    1,188.00€
  • Clenproperol

    CAS:
    Clenproperol is a β2-adrenergic agonist.
    Formula:C11H16Cl2N2O
    Color and Shape:Solid
    Molecular weight:263.16

    Ref: TM-T40480

    25mg
    1,369.00€
  • Benzamide Derivative 1

    CAS:
    Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.
    Formula:C22H34ClN3O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:423.98

    Ref: TM-T13570

    1mg
    630.00€
    5mg
    1,620.00€
  • HAMI 3379

    CAS:
    HAMI 3379 (HAMI3379) is a CysLT2 antagonist that attenuates brain damage and inhibits microglia inflammation following focal cerebral ischemia in rats.
    Formula:C34H45NO8
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:595.72

    Ref: TM-T64205

    1mg
    139.00€
    2mg
    225.00€
    5mg
    449.00€
  • GR 128107

    CAS:
    GR 128107 is an antagonist of melatonin receptor.
    Formula:C16H20N2O2
    Color and Shape:Solid
    Molecular weight:272.34

    Ref: TM-T27429

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€