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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6012 products of "GPCR/G-Protein"

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  • Isoetharine

    CAS:
    Isoetharine is a selective agonist of β2-adrenergic receptor used as a bronchodilator for emphysema, bronchitis, and asthma.
    Formula:C13H21NO3
    Color and Shape:Solid
    Molecular weight:239.31

    Ref: TM-T4983L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Sulfisoxazole diethanolamine

    CAS:
    Sulfisoxazole diethanolamine: a sulfonamide antibacterial, endothelin receptors A and B antagonist, inhibits breast cancer exosomes.
    Formula:C15H24N4O5S
    Color and Shape:Solid
    Molecular weight:372.44

    Ref: TM-T61498

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • hBChE-IN-2

    CAS:
    hBChE-IN-2 is a BChE inhibitor and CB2R agonist with neuroprotective activity for the study of Alzheimer's disease-like neurological disorders.
    Formula:C27H36N4O3
    Purity:99.60% - 99.83%
    Color and Shape:Soild
    Molecular weight:464.6

    Ref: TM-T77509

    1mg
    109.00€
    5mg
    261.00€
    10mg
    374.00€
    25mg
    583.00€
  • JTC-017

    CAS:
    JTC-017 is an antagonist of Corticotropin-releasing hormone receptor 1.
    Formula:C20H25Cl2N3O5S
    Color and Shape:Solid
    Molecular weight:490.4

    Ref: TM-T24216

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5-trans-Prostaglandin E2

    CAS:
    5-trans-PGE2 speeds up fibrinolysis, boosts tissue-PA mediated plasminogen activation, and blocks platelet clumping in human PRP.
    Formula:C20H32O5
    Color and Shape:Solid
    Molecular weight:352.47

    Ref: TM-T71851

    1mg
    233.00€
    5mg
    1,035.00€
    10mg
    1,783.00€
  • SEP-363856

    CAS:
    SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.
    Formula:C9H13NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:183.27

    Ref: TM-T12899

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CAD031

    CAS:
    CAD031, a more active derivative of the Alzheimer's disease (AD) targeting agent J147, exhibits neuroprotective and memory-enhancing properties.
    Formula:C18H14F6N2O2
    Color and Shape:Solid
    Molecular weight:404.31

    Ref: TM-T78596

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • HEAT hydrochloride

    CAS:
    HEAT hydrochloride is an α1-adrenoceptor antagonist.
    Formula:C19H22ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.84

    Ref: TM-T22837

    10mg
    577.00€
  • S1P1 Agonist III

    CAS:
    S1P1 Agonist III is an orally active S1P1 receptor agonist (EC₅₀ = 18 nM) with applications in inflammation, immunology, and receptor signaling studies.
    Formula:C21H16F3N3O3
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:415.37

    Ref: TM-T16833

    1mg
    37.00€
    5mg
    72.00€
    1mL*10mM (DMSO)
    79.00€
    10mg
    99.00€
    25mg
    187.00€
    50mg
    309.00€
    100mg
    464.00€
  • ZCZ011

    CAS:
    ZCZ011 enhances CB1 receptor effects, crosses blood-brain barrier, and potentiates cannabimimetic behaviors in mice.
    Formula:C21H18N2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:362.44

    Ref: TM-T29206

    50mg
    35.00€
    100mg
    56.00€
    200mg
    86.00€
    500mg
    140.00€
  • XCC

    CAS:
    XCC is an Adenosine receptor antagonist.
    Formula:C19H22N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.4

    Ref: TM-T23537

    50mg
    2,422.00€
  • Ksg 504

    CAS:
    Ksg 504 has superior selectivity and affinity to CCK-A receptors and derived from proglumide.
    Formula:C31H49N5O8S
    Color and Shape:Solid
    Molecular weight:651.81

    Ref: TM-T32425

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DR4485 hydrochloride

    CAS:
    5-HT7 antagonist
    Formula:C26H29Cl3N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:491.88

    Ref: TM-T22750

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A1AR antagonist 4

    CAS:
    Compound 22: A1AR antagonist, pIC50 5.51, pKi 6.29, potent and selective.
    Formula:C23H25N3O2
    Color and Shape:Solid
    Molecular weight:375.46

    Ref: TM-T61536

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • R-SKF-38393A HCl

    CAS:
    R(+)-SKF-38393A is a D1 dopamine receptor agonist and also is a more active enantiomer of (±)-SKF-38393A.
    Formula:C16H18ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:291.77

    Ref: TM-T26144

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CGP 25454A

    CAS:
    CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor.
    Formula:C15H21Cl2N3O2
    Color and Shape:Solid
    Molecular weight:346.25

    Ref: TM-T10779

    2mg
    125.00€
    5mg
    205.00€
    25mg
    552.00€
    50mg
    717.00€
    100mg
    1,224.00€
  • Org-12962 hydrochloride

    CAS:
    Org-12962 hydrochloride is a 5-HT2C receptor agonist.
    Formula:C10H12Cl2F3N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.12

    Ref: TM-T23110

    5mg
    359.00€
    10mg
    538.00€
    25mg
    1,234.00€
    50mg
    2,277.00€
  • GSK466317A

    CAS:
    GSK466317A is a GRK2 inhibitor.
    Formula:C21H16ClF3N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.83

    Ref: TM-T27479

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Glucagon receptor antagonists-5

    CAS:
    Oral indazole-based glucagon antagonist, Ki: 32 nM, may treat type 2 diabetes.
    Formula:C30H29ClF3N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:572.02

    Ref: TM-T11416

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KUL-7211 racemate

    CAS:
    KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.
    Formula:C19H23NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.39

    Ref: TM-T11786

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€