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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6012 products of "GPCR/G-Protein"

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  • R 75317

    CAS:
    R 75317 is a Platelet-activating factor (PAF) antagonist.
    Formula:C29H50N3O8PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:631.76

    Ref: TM-T26022

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • ANEB-001

    CAS:
    ANEB-001 is an orally active CB1 inhibitor that can be used in studies of acute cannabinoid intoxication.
    Formula:C22H24ClF3N2O2
    Color and Shape:Solid
    Molecular weight:440.89

    Ref: TM-T62551

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Trifluperidol HCl

    CAS:
    Trifluperidol, a dopamine D2-receptor antagonist, is used to treat schizophrenia.
    Formula:C22H24ClF4NO2
    Color and Shape:Solid
    Molecular weight:445.88

    Ref: TM-T29010

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JNJ 10181457 dihydrochloride

    CAS:
    JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.
    Formula:C20H28N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.45

    Ref: TM-T22878

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RBI-257 Maleate

    CAS:
    RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.
    Formula:C25H32IN3O5
    Color and Shape:Solid
    Molecular weight:581.44

    Ref: TM-T28505

    1mg
    221.00€
    5mg
    982.00€
  • MLN3126

    CAS:
    MLN3126: Oral CCR9 blocker, hinders CCL25-triggered chemotaxis/thymocyte calcium influx, IC50 of 6.3 nM.
    Formula:C21H19ClN2O5S
    Color and Shape:Solid
    Molecular weight:446.9

    Ref: TM-T62660

    25mg
    775.00€
    50mg
    1,009.00€
    100mg
    1,449.00€
  • DW-1350

    CAS:
    DW-1350 is an antagonist of LTB4 receptor.
    Formula:C25H31N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.6

    Ref: TM-T15182

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KSCM-1

    CAS:
    KSCM-1 is a selective sigma-1 receptor ligand.
    Formula:C26H32N2O4
    Color and Shape:Solid
    Molecular weight:436.54

    Ref: TM-T25584

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GR-55562 dihydrobromide

    CAS:
    GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.
    Formula:C23H26ClN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.93

    Ref: TM-T27432

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Quinelorane dihydrochloride

    CAS:
    Dopamine D2 and D3 receptor agonist
    Formula:C14H23ClN4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:282.81

    Ref: TM-T23211

    10mg
    1,018.00€
  • Sortilin antagonist 1

    CAS:
    Sortilin antagonist 1 blocks Neurotensin binding with 20 nM IC50, useful in neurological disease research.
    Formula:C20H24N2O4
    Color and Shape:Solid
    Molecular weight:356.42

    Ref: TM-T72410

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Antiplatelet agent 1

    CAS:
    Antiplatelet agent 1 is a ticagrelor analogue that exhibits anti-platelet effects and can be used in platelet agglutination studies.
    Formula:C21H24F2N6O4S
    Color and Shape:Solid
    Molecular weight:494.51

    Ref: TM-T63334

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • CP 59430

    CAS:
    CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.
    Formula:C21H22N8O3
    Color and Shape:Solid
    Molecular weight:434.45

    Ref: TM-T31022

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SDZ 21009

    CAS:
    β-adrenoceptor and 5-HT1A/1B receptor antagonist
    Formula:C19H28N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.44

    Ref: TM-T23343

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Adrenaline sulfate

    CAS:
    Adrenaline sulfate: orally active, α/β-adrenergic agonist, treats anaphylaxis, researched for cardiac arrest.
    Formula:C9H15NO7S
    Color and Shape:Solid
    Molecular weight:281.279

    Ref: TM-T69151

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CL-184005

    CAS:
    CL-184005 is a PAF inhibitor that blocks tumor necrosis factor synthesis and reduces spleen-associated TNF protein.
    Formula:C33H46NO7PS
    Color and Shape:Solid
    Molecular weight:631.76

    Ref: TM-T27035

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PROTAC(H-PGDS)-7

    CAS:
    PROTAC(H-PGDS)-7, a potent H-PGDS degrader, inhibits PGD2 in KU812 cells; DC50 is 17.3 pM. Potential DMD treatment.
    Formula:C40H38N8O7
    Color and Shape:Solid
    Molecular weight:742.78

    Ref: TM-T41267

    500µg
    642.00€
    1mg
    898.00€
  • Anatibant

    CAS:
    Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.
    Formula:C34H36Cl2N6O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:711.66

    Ref: TM-T26627

    500mg
    To inquire
    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • LY 393558

    CAS:
    Dual 5-HT1B/1D receptor antagonist
    Formula:C26H31FN4O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:546.68

    Ref: TM-T22953

    1mg
    112.00€
    5mg
    294.00€
    10mg
    517.00€
  • SGS518 oxalate

    CAS:
    SGS518 oxalate is a 5-HT6 antagonist.
    Formula:C23H24F2N2O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.51

    Ref: TM-T23350

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€