
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
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R 75317
CAS:R 75317 is a Platelet-activating factor (PAF) antagonist.Formula:C29H50N3O8PSPurity:98%Color and Shape:SolidMolecular weight:631.76ANEB-001
CAS:ANEB-001 is an orally active CB1 inhibitor that can be used in studies of acute cannabinoid intoxication.Formula:C22H24ClF3N2O2Color and Shape:SolidMolecular weight:440.89Trifluperidol HCl
CAS:Trifluperidol, a dopamine D2-receptor antagonist, is used to treat schizophrenia.Formula:C22H24ClF4NO2Color and Shape:SolidMolecular weight:445.88JNJ 10181457 dihydrochloride
CAS:JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.Formula:C20H28N2OPurity:98%Color and Shape:SolidMolecular weight:312.45RBI-257 Maleate
CAS:RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.Formula:C25H32IN3O5Color and Shape:SolidMolecular weight:581.44MLN3126
CAS:MLN3126: Oral CCR9 blocker, hinders CCL25-triggered chemotaxis/thymocyte calcium influx, IC50 of 6.3 nM.Formula:C21H19ClN2O5SColor and Shape:SolidMolecular weight:446.9DW-1350
CAS:DW-1350 is an antagonist of LTB4 receptor.Formula:C25H31N3O3SPurity:98%Color and Shape:SolidMolecular weight:453.6KSCM-1
CAS:KSCM-1 is a selective sigma-1 receptor ligand.Formula:C26H32N2O4Color and Shape:SolidMolecular weight:436.54GR-55562 dihydrobromide
CAS:GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.Formula:C23H26ClN3O2Purity:98%Color and Shape:SolidMolecular weight:411.93Quinelorane dihydrochloride
CAS:Dopamine D2 and D3 receptor agonistFormula:C14H23ClN4Purity:98%Color and Shape:SolidMolecular weight:282.81Sortilin antagonist 1
CAS:Sortilin antagonist 1 blocks Neurotensin binding with 20 nM IC50, useful in neurological disease research.Formula:C20H24N2O4Color and Shape:SolidMolecular weight:356.42Antiplatelet agent 1
CAS:Antiplatelet agent 1 is a ticagrelor analogue that exhibits anti-platelet effects and can be used in platelet agglutination studies.Formula:C21H24F2N6O4SColor and Shape:SolidMolecular weight:494.51CP 59430
CAS:CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.Formula:C21H22N8O3Color and Shape:SolidMolecular weight:434.45SDZ 21009
CAS:β-adrenoceptor and 5-HT1A/1B receptor antagonistFormula:C19H28N2O4Purity:98%Color and Shape:SolidMolecular weight:348.44Adrenaline sulfate
CAS:Adrenaline sulfate: orally active, α/β-adrenergic agonist, treats anaphylaxis, researched for cardiac arrest.Formula:C9H15NO7SColor and Shape:SolidMolecular weight:281.279CL-184005
CAS:CL-184005 is a PAF inhibitor that blocks tumor necrosis factor synthesis and reduces spleen-associated TNF protein.Formula:C33H46NO7PSColor and Shape:SolidMolecular weight:631.76PROTAC(H-PGDS)-7
CAS:PROTAC(H-PGDS)-7, a potent H-PGDS degrader, inhibits PGD2 in KU812 cells; DC50 is 17.3 pM. Potential DMD treatment.Formula:C40H38N8O7Color and Shape:SolidMolecular weight:742.78Anatibant
CAS:Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.Formula:C34H36Cl2N6O5SPurity:98%Color and Shape:SolidMolecular weight:711.66LY 393558
CAS:Dual 5-HT1B/1D receptor antagonistFormula:C26H31FN4O4S2Purity:98%Color and Shape:SolidMolecular weight:546.68SGS518 oxalate
CAS:SGS518 oxalate is a 5-HT6 antagonist.Formula:C23H24F2N2O7SPurity:98%Color and Shape:SolidMolecular weight:510.51
