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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6012 products of "GPCR/G-Protein"

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  • cis-Epoxysuccinic acid

    CAS:
    cis-Epoxysuccinic acid is a potential agonist of Succinate receptor 1 and inhibitor of Isocitrate lyase 1 for use in biochemical experiments.
    Formula:C4H4O5
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:132.07

    Ref: TM-T71921

    50mg
    34.00€
    100mg
    47.00€
    1mL*10mM (DMSO)
    50.00€
    500mg
    77.00€
  • JNJ-28610244

    CAS:
    JNJ-28610244 is a specific agonist of the H4 receptor. It acts by blocking Mac-1-dependent activation of p38 MAPK.
    Formula:C16H21N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:271.36

    Ref: TM-T24207

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Rp-cAMPS sodium

    CAS:
    Rp-cAMPS sodium is a phosphorothioate analog of cAMP, a PKA inhibitor and cAMP antagonist that inhibits cAMP-dependent protein kinases.
    Formula:C10H11N5NaO5PS
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:367.25

    Ref: TM-T36679

    1mg
    269.00€
  • CCR2 antagonist 3

    CAS:
    CCR2 antagonist 3 (AZD-2927) is an antagonist of CCR2.
    Formula:C17H25FN2O2
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:308.39

    Ref: TM-T10712

    1mg
    66.00€
    5mg
    147.00€
    1mL*10mM (DMSO)
    161.00€
    10mg
    225.00€
    25mg
    398.00€
    50mg
    532.00€
    100mg
    745.00€
    200mg
    982.00€
  • SF 11

    CAS:
    SF 11 is a potent and brain penetrant neuropeptide Y Y2 receptor antagonist with IC50 of 199 nM. Antidepressant-like activity
    Formula:C27H30N2O2S
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:446.6

    Ref: TM-T23349

    2mg
    34.00€
    5mg
    52.00€
    10mg
    86.00€
    25mg
    156.00€
    50mg
    264.00€
    100mg
    408.00€
    200mg
    548.00€
  • Iferanserin HCl

    CAS:
    Iferanserin HCl is a selective serotonin receptor antagonist.
    Formula:C23H29ClN2O
    Color and Shape:Solid
    Molecular weight:384.95

    Ref: TM-T69905

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GYKI-13380

    CAS:
    GYKI-13380, also known as LS-79445, is a small molecule with potent bioactivity. Detail information has not been published yet.
    Formula:C16H22N2O3
    Color and Shape:Solid
    Molecular weight:290.36

    Ref: TM-T32027

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Pruvanserin hydrochloride

    CAS:
    Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.
    Formula:C22H22ClFN4O
    Purity:99.6%
    Color and Shape:Solid
    Molecular weight:412.89

    Ref: TM-T22762

    1mg
    205.00€
    5mg
    515.00€
    10mg
    740.00€
    25mg
    1,674.00€
    50mg
    3,052.00€
  • CB2 modulator 1

    CAS:
    CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.
    Formula:C18H19F3N4O2
    Purity:99.6%
    Color and Shape:Solid
    Molecular weight:380.36

    Ref: TM-T10696

    5mg
    34.00€
    1mL*10mM (DMSO)
    39.00€
    10mg
    48.00€
    25mg
    73.00€
    50mg
    105.00€
  • Wy 49051

    CAS:
    Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).
    Formula:C28H33N5O3
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:487.59

    Ref: TM-T13352

    1mg
    99.00€
    5mg
    188.00€
    1mL*10mM (DMSO)
    250.00€
    10mg
    273.00€
    25mg
    427.00€
    50mg
    575.00€
    100mg
    743.00€
    200mg
    990.00€
  • LY 393558

    CAS:
    Dual 5-HT1B/1D receptor antagonist
    Formula:C26H31FN4O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:546.68

    Ref: TM-T22953

    1mg
    112.00€
    5mg
    294.00€
    10mg
    517.00€
  • VER-3323

    CAS:
    VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.
    Formula:C11H15BrN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:255.15

    Ref: TM-T29103

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AGI-41998

    CAS:
    AGI-41998: a potent MAT2A inhibitor that crosses the blood-brain barrier, targeting SAM enzymes for cancer therapy and CNS research.
    Formula:C22H16BrF3N4O2
    Color and Shape:Solid
    Molecular weight:505.29

    Ref: TM-T9730

    25mg
    1,144.00€
    50mg
    1,485.00€
    100mg
    2,385.00€
  • Nexopamil racemate

    CAS:
    Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.
    Formula:C24H40N2O3
    Purity:98.61%
    Color and Shape:Solid
    Molecular weight:404.59

    Ref: TM-T12215

    1mg
    630.00€
    5mg
    1,620.00€
  • (-)-GSK598809

    CAS:
    (-)-GSK598809 is an isomer of GSK598809 that is a potent and selective antagonist of dopamine D3 Receptor.
    Formula:C22H23F4N5OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.51

    Ref: TM-T10062

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Reproterol hydrochloride

    CAS:
    Reproterol hydrochloride, a β2 adrenoreceptor agonist, is used to treat asthma and chronic obstructive pulmonary disease (COPD).
    Formula:C18H24ClN5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.87

    Ref: TM-T28519

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Butanserin

    CAS:
    Butanserin is a 5-hydroxytryptamine S2-antagonist.
    Formula:C24H26FN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:423.48

    Ref: TM-T25185

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Orexin receptor antagonist 3

    CAS:
    Orexin receptor antagonist 3 (example 216) is an orexin receptor antagonist.
    Formula:C21H22N8O3
    Color and Shape:Solid
    Molecular weight:434.45

    Ref: TM-T62453

    25mg
    1,459.00€
    50mg
    1,900.00€
    100mg
    2,690.00€
  • Palmitoyl serinol

    CAS:
    Anticancer agent 110 is an anticancer compound with cytotoxic, antitumor and antileukemic activities.
    Formula:C19H39NO3
    Color and Shape:Solid
    Molecular weight:329.52

    Ref: TM-T60957

    5mg
    132.00€
    10mg
    254.00€
    50mg
    1,018.00€
    100mg
    1,783.00€
  • NIDA 41020

    CAS:
    NIDA 41020 is a CB1 receptor antagonist.
    Formula:C23H24Cl2N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.37

    Ref: TM-T23069

    5mg
    421.00€
    50mg
    2,988.00€