
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
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cis-Epoxysuccinic acid
CAS:cis-Epoxysuccinic acid is a potential agonist of Succinate receptor 1 and inhibitor of Isocitrate lyase 1 for use in biochemical experiments.Formula:C4H4O5Purity:99.81%Color and Shape:SolidMolecular weight:132.07JNJ-28610244
CAS:JNJ-28610244 is a specific agonist of the H4 receptor. It acts by blocking Mac-1-dependent activation of p38 MAPK.Formula:C16H21N3OPurity:98%Color and Shape:SolidMolecular weight:271.36Rp-cAMPS sodium
CAS:Rp-cAMPS sodium is a phosphorothioate analog of cAMP, a PKA inhibitor and cAMP antagonist that inhibits cAMP-dependent protein kinases.Formula:C10H11N5NaO5PSPurity:99.71%Color and Shape:SolidMolecular weight:367.25CCR2 antagonist 3
CAS:CCR2 antagonist 3 (AZD-2927) is an antagonist of CCR2.Formula:C17H25FN2O2Purity:99.87%Color and Shape:SolidMolecular weight:308.39Ref: TM-T10712
1mg66.00€5mg147.00€1mL*10mM (DMSO)161.00€10mg225.00€25mg398.00€50mg532.00€100mg745.00€200mg982.00€SF 11
CAS:SF 11 is a potent and brain penetrant neuropeptide Y Y2 receptor antagonist with IC50 of 199 nM. Antidepressant-like activityFormula:C27H30N2O2SPurity:99.51%Color and Shape:SolidMolecular weight:446.6Iferanserin HCl
CAS:Iferanserin HCl is a selective serotonin receptor antagonist.Formula:C23H29ClN2OColor and Shape:SolidMolecular weight:384.95GYKI-13380
CAS:GYKI-13380, also known as LS-79445, is a small molecule with potent bioactivity. Detail information has not been published yet.Formula:C16H22N2O3Color and Shape:SolidMolecular weight:290.36Pruvanserin hydrochloride
CAS:Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.Formula:C22H22ClFN4OPurity:99.6%Color and Shape:SolidMolecular weight:412.89CB2 modulator 1
CAS:CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.Formula:C18H19F3N4O2Purity:99.6%Color and Shape:SolidMolecular weight:380.36Wy 49051
CAS:Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).Formula:C28H33N5O3Purity:99.89%Color and Shape:SolidMolecular weight:487.59Ref: TM-T13352
1mg99.00€5mg188.00€1mL*10mM (DMSO)250.00€10mg273.00€25mg427.00€50mg575.00€100mg743.00€200mg990.00€LY 393558
CAS:Dual 5-HT1B/1D receptor antagonistFormula:C26H31FN4O4S2Purity:98%Color and Shape:SolidMolecular weight:546.68VER-3323
CAS:VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.Formula:C11H15BrN2Purity:98%Color and Shape:SolidMolecular weight:255.15AGI-41998
CAS:AGI-41998: a potent MAT2A inhibitor that crosses the blood-brain barrier, targeting SAM enzymes for cancer therapy and CNS research.Formula:C22H16BrF3N4O2Color and Shape:SolidMolecular weight:505.29Nexopamil racemate
CAS:Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.Formula:C24H40N2O3Purity:98.61%Color and Shape:SolidMolecular weight:404.59(-)-GSK598809
CAS:(-)-GSK598809 is an isomer of GSK598809 that is a potent and selective antagonist of dopamine D3 Receptor.Formula:C22H23F4N5OSPurity:98%Color and Shape:SolidMolecular weight:481.51Reproterol hydrochloride
CAS:Reproterol hydrochloride, a β2 adrenoreceptor agonist, is used to treat asthma and chronic obstructive pulmonary disease (COPD).Formula:C18H24ClN5O5Purity:98%Color and Shape:SolidMolecular weight:425.87Butanserin
CAS:Butanserin is a 5-hydroxytryptamine S2-antagonist.Formula:C24H26FN3O3Purity:98%Color and Shape:SolidMolecular weight:423.48Orexin receptor antagonist 3
CAS:Orexin receptor antagonist 3 (example 216) is an orexin receptor antagonist.Formula:C21H22N8O3Color and Shape:SolidMolecular weight:434.45Palmitoyl serinol
CAS:Anticancer agent 110 is an anticancer compound with cytotoxic, antitumor and antileukemic activities.Formula:C19H39NO3Color and Shape:SolidMolecular weight:329.52NIDA 41020
CAS:NIDA 41020 is a CB1 receptor antagonist.Formula:C23H24Cl2N4O2Purity:98%Color and Shape:SolidMolecular weight:459.37
