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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6012 products of "GPCR/G-Protein"

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  • CP 59430

    CAS:
    CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.
    Formula:C21H22N8O3
    Color and Shape:Solid
    Molecular weight:434.45

    Ref: TM-T31022

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MHP 133

    CAS:
    MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).
    Formula:C17H20ClN5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.83

    Ref: TM-T13772

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SSTR4 agonist 3

    CAS:
    SSTR4 agonist 3 activates SSTR4 in the hippocampus and neocortex, aiding memory and learning, and shows potent pain relief in rodents.
    Formula:C18H24N4OS
    Color and Shape:Solid
    Molecular weight:344.47

    Ref: TM-T61130

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ATC0065 HCl

    CAS:
    ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.
    Formula:C25H31BrCl2F3N5O
    Color and Shape:Solid
    Molecular weight:625.35

    Ref: TM-T69170

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CL-184005

    CAS:
    CL-184005 is a PAF inhibitor that blocks tumor necrosis factor synthesis and reduces spleen-associated TNF protein.
    Formula:C33H46NO7PS
    Color and Shape:Solid
    Molecular weight:631.76

    Ref: TM-T27035

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-Viloxazine Hydrochloride

    CAS:
    (R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.
    Formula:C13H20ClNO3
    Purity:99.88% - 99.94%
    Color and Shape:Solid
    Molecular weight:273.76

    Ref: TM-T22413

    1mg
    52.00€
    1mL*10mM (DMSO)
    101.00€
    5mg
    111.00€
    10mg
    162.00€
    25mg
    235.00€
    50mg
    330.00€
    100mg
    452.00€
    200mg
    607.00€
  • Fenspiride-d5

    CAS:
    Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.
    Formula:C15H15D5N2O2
    Color and Shape:Solid
    Molecular weight:265.36

    Ref: TM-T71141

    1mg
    1,018.00€
    5mg
    3,312.00€
  • CI-943

    CAS:
    CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.
    Formula:C12H17N5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:231.3

    Ref: TM-T14963

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Mequitamium iodide

    CAS:
    Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.
    Formula:C21H25IN2S
    Color and Shape:Solid
    Molecular weight:464.41

    Ref: TM-T28015

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CV-3988

    CAS:
    CV-3988 is a specific antagonist of PAF-R (platelet-activating factor receptor)(Ki = 0.872 μM).
    Formula:C28H53N2O7PS
    Color and Shape:Solid
    Molecular weight:592.77

    Ref: TM-T27101

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • CAY10397

    CAS:
    CAY10397, a selective inhibitor of 15-hydroxy PGDH, significantly suppresses endogenous 11-oxo-ETE production with a corresponding increase in 11(R)-HETE.
    Formula:C17H16N2O5
    Color and Shape:Solid
    Molecular weight:328.32

    Ref: TM-T26956

    1mg
    192.00€
    5mg
    825.00€
    10mg
    1,459.00€
    25mg
    3,177.00€
  • CI-1015

    CAS:
    CI-1015 is a CCK-B receptor antagonist with oral activity.
    Formula:C29H39N3O4
    Color and Shape:Solid
    Molecular weight:493.64

    Ref: TM-T27014

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KSCM-5

    CAS:
    KSCM-5 is a sigma receptor ligand.
    Formula:C24H28N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.49

    Ref: TM-T25586

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bepafant

    CAS:
    Bepafant: a PAF antagonist with anti-inflammatory properties; induces apoptosis in PTEN-positive NB4, KG1, NB4-MR4 cells, not in PTEN-negative THP1, U937.
    Formula:C23H22ClN5O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:467.97

    Ref: TM-T26775

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • E55888

    CAS:
    E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.
    Formula:C16H23N3
    Color and Shape:Solid
    Molecular weight:257.37

    Ref: TM-T27230

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Etoperidone hydrochloride

    CAS:
    Etoperidone hydrochloride is an antidepressant agent.
    Formula:C19H29Cl2N5O
    Color and Shape:Solid
    Molecular weight:414.37

    Ref: TM-T24048

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS1067

    CAS:
    MRS1067 is an antagonist of A3 adenosine receptor.
    Formula:C19H16Cl2O3
    Color and Shape:Solid
    Molecular weight:363.23

    Ref: TM-T28097

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PGlu-3-methyl-His-Pro-NH2 TFA


    PGlu-3-methyl-His-Pro-NH2 TFA boosts TRH receptor binding & TSH release.
    Formula:C19H25F3N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:490.43

    Ref: TM-T19511

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Oxaprotiline

    CAS:
    Oxaprotiline: an antidepressant, norepinephrine inhibitor, and H1 blocker; studied in hospital depression but not marketed.
    Formula:C20H23NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:293.4

    Ref: TM-T25906

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Butaclamol free base

    CAS:
    Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.
    Formula:C25H31NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.52

    Ref: TM-T23842

    25mg
    1,369.00€