
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
CP 59430
CAS:CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.Formula:C21H22N8O3Color and Shape:SolidMolecular weight:434.45MHP 133
CAS:MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).Formula:C17H20ClN5O3Purity:98%Color and Shape:SolidMolecular weight:377.83SSTR4 agonist 3
CAS:SSTR4 agonist 3 activates SSTR4 in the hippocampus and neocortex, aiding memory and learning, and shows potent pain relief in rodents.Formula:C18H24N4OSColor and Shape:SolidMolecular weight:344.47ATC0065 HCl
CAS:ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.Formula:C25H31BrCl2F3N5OColor and Shape:SolidMolecular weight:625.35CL-184005
CAS:CL-184005 is a PAF inhibitor that blocks tumor necrosis factor synthesis and reduces spleen-associated TNF protein.Formula:C33H46NO7PSColor and Shape:SolidMolecular weight:631.76(R)-Viloxazine Hydrochloride
CAS:(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.Formula:C13H20ClNO3Purity:99.88% - 99.94%Color and Shape:SolidMolecular weight:273.76Ref: TM-T22413
1mg52.00€1mL*10mM (DMSO)101.00€5mg111.00€10mg162.00€25mg235.00€50mg330.00€100mg452.00€200mg607.00€Fenspiride-d5
CAS:Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.Formula:C15H15D5N2O2Color and Shape:SolidMolecular weight:265.36CI-943
CAS:CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.Formula:C12H17N5Purity:98%Color and Shape:SolidMolecular weight:231.3Mequitamium iodide
CAS:Mequitamium iodide is a PAF inhibitor, curbing platelet aggregation and bronchoconstriction without blocking PAF receptors.Formula:C21H25IN2SColor and Shape:SolidMolecular weight:464.41CV-3988
CAS:CV-3988 is a specific antagonist of PAF-R (platelet-activating factor receptor)(Ki = 0.872 μM).Formula:C28H53N2O7PSColor and Shape:SolidMolecular weight:592.77CAY10397
CAS:CAY10397, a selective inhibitor of 15-hydroxy PGDH, significantly suppresses endogenous 11-oxo-ETE production with a corresponding increase in 11(R)-HETE.Formula:C17H16N2O5Color and Shape:SolidMolecular weight:328.32CI-1015
CAS:CI-1015 is a CCK-B receptor antagonist with oral activity.Formula:C29H39N3O4Color and Shape:SolidMolecular weight:493.64KSCM-5
CAS:KSCM-5 is a sigma receptor ligand.Formula:C24H28N2O2Purity:98%Color and Shape:SolidMolecular weight:376.49Bepafant
CAS:Bepafant: a PAF antagonist with anti-inflammatory properties; induces apoptosis in PTEN-positive NB4, KG1, NB4-MR4 cells, not in PTEN-negative THP1, U937.Formula:C23H22ClN5O2SPurity:98%Color and Shape:SolidMolecular weight:467.97E55888
CAS:E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.Formula:C16H23N3Color and Shape:SolidMolecular weight:257.37Etoperidone hydrochloride
CAS:Etoperidone hydrochloride is an antidepressant agent.Formula:C19H29Cl2N5OColor and Shape:SolidMolecular weight:414.37MRS1067
CAS:MRS1067 is an antagonist of A3 adenosine receptor.Formula:C19H16Cl2O3Color and Shape:SolidMolecular weight:363.23PGlu-3-methyl-His-Pro-NH2 TFA
PGlu-3-methyl-His-Pro-NH2 TFA boosts TRH receptor binding & TSH release.Formula:C19H25F3N6O6Purity:98%Color and Shape:SolidMolecular weight:490.43Oxaprotiline
CAS:Oxaprotiline: an antidepressant, norepinephrine inhibitor, and H1 blocker; studied in hospital depression but not marketed.Formula:C20H23NOPurity:98%Color and Shape:SolidMolecular weight:293.4Butaclamol free base
CAS:Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.Formula:C25H31NOPurity:98%Color and Shape:SolidMolecular weight:361.52
