
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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SV-156
CAS:SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).Formula:C21H23BrN2O2Color and Shape:SolidMolecular weight:415.32RPT193
CAS:RPT193 is an oral CCR4 inhibitor reducing Th2 cell migration in atopic dermatitis, asthma, and allergies.Formula:C27H34Cl3N5O2Color and Shape:SolidMolecular weight:566.95Bag-1
CAS:Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.Formula:C22H27N3Color and Shape:SolidMolecular weight:333.47JNJ-17156516
CAS:JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.Formula:C26H22Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:481.37Adenosine receptor antagonist 2
CAS:Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.Formula:C23H21FN8OColor and Shape:SolidMolecular weight:444.46GB-110
CAS:GB-110, a potent PAR2 agonist, triggers Ca2+ release in HT29 cells with a 0.28 μM EC50, is orally active and nonpeptidic.Formula:C33H48N6O5Purity:98%Color and Shape:SolidMolecular weight:608.77GSK334429
CAS:GSK334429 is an antagonist of histamine H3 receptor.Formula:C20H29F3N4OColor and Shape:SolidMolecular weight:398.47Piroheptine HCl
CAS:Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.Formula:C22H26ClNPurity:98%Color and Shape:SolidMolecular weight:339.9Bromerguride
CAS:Bromerguride is a dopamine antagonist with the activity of antipsychotic.Formula:C20H25BrN4OColor and Shape:SolidMolecular weight:417.34CCG-271423
CAS:CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.Formula:C28H26N4O3Color and Shape:SolidMolecular weight:466.532-Thio-UTP
CAS:2-ThioUTP tetrasodium salt is a P2Y2 agonist.Formula:C9H15N2O14P3SPurity:98%Color and Shape:SolidMolecular weight:500.215-HT7 receptor ligand 1
CAS:Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.Formula:C21H23N7Color and Shape:SolidMolecular weight:373.45A-940894
CAS:A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.Formula:C17H21N5Color and Shape:SolidMolecular weight:295.38TH-162
CAS:TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.Formula:C19H23N5O4Color and Shape:SolidMolecular weight:385.42Fonazine
CAS:Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.Formula:C19H25N3O2S2Color and Shape:SolidMolecular weight:391.55Lidanserin
CAS:Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Formula:C26H31FN2O4Purity:98%Color and Shape:SolidMolecular weight:454.53PD-156707
CAS:PD-156707 is a selective antagonist of endothelin A receptor.Formula:C28H26NaO9Purity:98%Color and Shape:SolidMolecular weight:529.497ICI 192605
CAS:ICI 192605 is a potent thromboxane A2 receptor (TP receptor) antagonist.Formula:C22H23ClO5Color and Shape:SolidMolecular weight:402.87AL-3138
CAS:AL-3138 is a prostaglandin F2alpha (PGF2alpha) analogue which antagonizes FP prostanoid receptor-mediated inositol phosphates generation.Formula:C20H33FO4Color and Shape:SolidMolecular weight:356.47Methyldopate hydrochloride
CAS:Methyldopate HCl is an agent of antihypertensive.Formula:C12H18ClNO4Color and Shape:SolidMolecular weight:275.73
