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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • SV-156

    CAS:
    SV-156 is a highly selective antagonist of dopamine receptor 2 (D2).
    Formula:C21H23BrN2O2
    Color and Shape:Solid
    Molecular weight:415.32

    Ref: TM-T28889

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RPT193

    CAS:
    RPT193 is an oral CCR4 inhibitor reducing Th2 cell migration in atopic dermatitis, asthma, and allergies.
    Formula:C27H34Cl3N5O2
    Color and Shape:Solid
    Molecular weight:566.95

    Ref: TM-T64013

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Bag-1

    CAS:
    Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.
    Formula:C22H27N3
    Color and Shape:Solid
    Molecular weight:333.47

    Ref: TM-T71595

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • JNJ-17156516

    CAS:
    JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.
    Formula:C26H22Cl2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.37

    Ref: TM-T27664

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Adenosine receptor antagonist 2

    CAS:
    Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.
    Formula:C23H21FN8O
    Color and Shape:Solid
    Molecular weight:444.46

    Ref: TM-T62611

    25mg
    1,791.00€
    50mg
    3,025.00€
  • GB-110

    CAS:
    GB-110, a potent PAR2 agonist, triggers Ca2+ release in HT29 cells with a 0.28 μM EC50, is orally active and nonpeptidic.
    Formula:C33H48N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:608.77

    Ref: TM-T11369

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GSK334429

    CAS:
    GSK334429 is an antagonist of histamine H3 receptor.
    Formula:C20H29F3N4O
    Color and Shape:Solid
    Molecular weight:398.47

    Ref: TM-T27473

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Piroheptine HCl

    CAS:
    Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.
    Formula:C22H26ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:339.9

    Ref: TM-T24645

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Bromerguride

    CAS:
    Bromerguride is a dopamine antagonist with the activity of antipsychotic.
    Formula:C20H25BrN4O
    Color and Shape:Solid
    Molecular weight:417.34

    Ref: TM-T26909

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • CCG-271423

    CAS:
    CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.
    Formula:C28H26N4O3
    Color and Shape:Solid
    Molecular weight:466.53

    Ref: TM-T62986

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 2-Thio-UTP

    CAS:
    2-ThioUTP tetrasodium salt is a P2Y2 agonist.
    Formula:C9H15N2O14P3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.21

    Ref: TM-T22503

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5-HT7 receptor ligand 1

    CAS:
    Compound 5c: 5-HT7 receptor ligand, K i = 8 nM, not hepatotoxic, moderate CYP3A4/CYP2D6 interaction.
    Formula:C21H23N7
    Color and Shape:Solid
    Molecular weight:373.45

    Ref: TM-T61515

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A-940894

    CAS:
    A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.
    Formula:C17H21N5
    Color and Shape:Solid
    Molecular weight:295.38

    Ref: TM-T23597

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TH-162

    CAS:
    TH-162 (R)-PIA is an A1 adenosine receptor agonist with ~100× higher affinity than its (+)-isomer.
    Formula:C19H23N5O4
    Color and Shape:Solid
    Molecular weight:385.42

    Ref: TM-T26266

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Fonazine

    CAS:
    Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.
    Formula:C19H25N3O2S2
    Color and Shape:Solid
    Molecular weight:391.55

    Ref: TM-T31844

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Lidanserin

    CAS:
    Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.
    Formula:C26H31FN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.53

    Ref: TM-T15754

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • PD-156707

    CAS:
    PD-156707 is a selective antagonist of endothelin A receptor.
    Formula:C28H26NaO9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:529.497

    Ref: TM-T28343

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ICI 192605

    CAS:
    ICI 192605 is a potent thromboxane A2 receptor (TP receptor) antagonist.
    Formula:C22H23ClO5
    Color and Shape:Solid
    Molecular weight:402.87

    Ref: TM-T27575

    1mg
    105.00€
    5mg
    304.00€
    10mg
    530.00€
    25mg
    1,189.00€
  • AL-3138

    CAS:
    AL-3138 is a prostaglandin F2alpha (PGF2alpha) analogue which antagonizes FP prostanoid receptor-mediated inositol phosphates generation.
    Formula:C20H33FO4
    Color and Shape:Solid
    Molecular weight:356.47

    Ref: TM-T29813

    25mg
    1,369.00€
  • Methyldopate hydrochloride

    CAS:
    Methyldopate HCl is an agent of antihypertensive.
    Formula:C12H18ClNO4
    Color and Shape:Solid
    Molecular weight:275.73

    Ref: TM-T20133

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€