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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • Daledalin

    CAS:
    Daledalin, an unmarketed 1970s antidepressant, is a selective norepinephrine reuptake inhibitor without serotonergic or dopaminergic effects.
    Formula:C19H24N2
    Color and Shape:Solid
    Molecular weight:280.41

    Ref: TM-T69788

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Fenspiride-d5

    CAS:
    Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.
    Formula:C15H15D5N2O2
    Color and Shape:Solid
    Molecular weight:265.36

    Ref: TM-T71141

    1mg
    1,018.00€
    5mg
    3,312.00€
  • SGC agonist 2

    CAS:
    SGC agonist 2 is a potent activator for cardiovascular and fibrotic diseases, per patent WO2021219088A1, compound 031.
    Formula:C23H17F2N7O2
    Color and Shape:Solid
    Molecular weight:461.42

    Ref: TM-T62909

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A331440

    CAS:
    A331440 is an modulator of L-histidine and histamine H3 receptor.
    Formula:C22H27N3O
    Color and Shape:Solid
    Molecular weight:349.47

    Ref: TM-T26480

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UP202-56

    CAS:
    UP202-56 is an adenosinergic agonist and is an adenosine analog.
    Formula:C33H37N7O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:595.69

    Ref: TM-T13256

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Spirendolol

    CAS:
    Spirendolol is an antagonist of β adrenergic receptor.
    Formula:C21H31NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.48

    Ref: TM-T16919

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UCSF678

    CAS:
    UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.
    Formula:C15H18N2O2S
    Color and Shape:Solid
    Molecular weight:290.38

    Ref: TM-T60597

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-592379

    CAS:
    PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).
    Formula:C13H21N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:235.33

    Ref: TM-T10080

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • HEMADO

    CAS:
    HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).
    Formula:C17H23N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.4

    Ref: TM-T15468

    1mg
    112.00€
    5mg
    388.00€
  • 6-Chloromelatonin

    CAS:
    6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.
    Formula:C13H15ClN2O2
    Purity:97.26% - 99.25%
    Color and Shape:Solid
    Molecular weight:266.72

    Ref: TM-T22530

    1mg
    315.00€
    5mg
    745.00€
    10mg
    1,018.00€
    25mg
    1,431.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
    500mg
    4,410.00€
  • Phenoprolamine Hydrochloride

    CAS:
    Phenoprolamine HCl: α1 blocker with anti-hypertensive, brain, and heart protection; inhibits CYP2D/3A, crosses the blood-brain barrier.
    Formula:C21H30ClNO3
    Color and Shape:Solid
    Molecular weight:379.92

    Ref: TM-T28400

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GR-203040 HCl

    CAS:
    GR203040 inhibits cyclophosphamide-induced damage in the rat and ferret bladder. GR-203040 is a selective NK1 receptor antagonist.
    Formula:C20H26Cl2N6O
    Color and Shape:Solid
    Molecular weight:437.37

    Ref: TM-T24102

    25mg
    1,738.00€
  • Naxifylline

    CAS:
    Naxifylline is an A1 adenosine receptor blocker that increases urine and protects kidneys during edema treatment in heart failure.
    Formula:C18H24N4O3
    Color and Shape:Solid
    Molecular weight:344.41

    Ref: TM-T33600

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • SUN 1334H

    CAS:
    SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
    Formula:C23H28Cl2F2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.38

    Ref: TM-T13040

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • DV 7028 hydrochloride

    CAS:
    DV 7028 hydrochloride is a 5-HT2A receptor antagonist.
    Formula:C21H26ClFN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.91

    Ref: TM-T22753

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Usmarapride free base

    CAS:
    Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.
    Formula:C21H29N5O2
    Purity:99.91% - 99.91%
    Color and Shape:Solid
    Molecular weight:383.49

    Ref: TM-T34751

    1mg
    194.00€
  • Colterol (free base)

    CAS:
    Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.
    Formula:C12H19NO3
    Color and Shape:Solid
    Molecular weight:225.28

    Ref: TM-T70089

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • S20928

    CAS:
    S20928 is an antagonist of melatonin receptor.
    Formula:C17H19NO
    Color and Shape:Solid
    Molecular weight:253.34

    Ref: TM-T28644

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 2-Methyl-5-HT maleate

    CAS:
    2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.
    Formula:C15H18N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:306.31

    Ref: TM-T10075L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Reversan

    CAS:
    Reversan(CBLC4H10) is a potent, nontoxic, and glioblastoma-associated inhibitor of multidrug resistance-associated protein 1 (MRP1) and P-glycoprotein (Pgp).
    Formula:C26H27N5O2
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:441.53

    Ref: TM-T12714

    1mg
    44.00€
    1mL*10mM (DMSO)
    92.00€
    5mg
    93.00€
    10mg
    130.00€
    25mg
    250.00€
    50mg
    401.00€
    100mg
    640.00€
    200mg
    884.00€