
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Daledalin
CAS:Daledalin, an unmarketed 1970s antidepressant, is a selective norepinephrine reuptake inhibitor without serotonergic or dopaminergic effects.Formula:C19H24N2Color and Shape:SolidMolecular weight:280.41Fenspiride-d5
CAS:Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.Formula:C15H15D5N2O2Color and Shape:SolidMolecular weight:265.36SGC agonist 2
CAS:SGC agonist 2 is a potent activator for cardiovascular and fibrotic diseases, per patent WO2021219088A1, compound 031.Formula:C23H17F2N7O2Color and Shape:SolidMolecular weight:461.42A331440
CAS:A331440 is an modulator of L-histidine and histamine H3 receptor.Formula:C22H27N3OColor and Shape:SolidMolecular weight:349.47UP202-56
CAS:UP202-56 is an adenosinergic agonist and is an adenosine analog.Formula:C33H37N7O4Purity:98%Color and Shape:SolidMolecular weight:595.69Spirendolol
CAS:Spirendolol is an antagonist of β adrenergic receptor.Formula:C21H31NO3Purity:98%Color and Shape:SolidMolecular weight:345.48UCSF678
CAS:UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.Formula:C15H18N2O2SColor and Shape:SolidMolecular weight:290.38PF-592379
CAS:PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).Formula:C13H21N3OPurity:98%Color and Shape:SolidMolecular weight:235.33HEMADO
CAS:HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).Formula:C17H23N5O4Purity:98%Color and Shape:SolidMolecular weight:361.46-Chloromelatonin
CAS:6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.Formula:C13H15ClN2O2Purity:97.26% - 99.25%Color and Shape:SolidMolecular weight:266.72Ref: TM-T22530
1mg315.00€5mg745.00€10mg1,018.00€25mg1,431.00€50mg1,783.00€100mg2,250.00€500mg4,410.00€Phenoprolamine Hydrochloride
CAS:Phenoprolamine HCl: α1 blocker with anti-hypertensive, brain, and heart protection; inhibits CYP2D/3A, crosses the blood-brain barrier.Formula:C21H30ClNO3Color and Shape:SolidMolecular weight:379.92GR-203040 HCl
CAS:GR203040 inhibits cyclophosphamide-induced damage in the rat and ferret bladder. GR-203040 is a selective NK1 receptor antagonist.Formula:C20H26Cl2N6OColor and Shape:SolidMolecular weight:437.37Naxifylline
CAS:Naxifylline is an A1 adenosine receptor blocker that increases urine and protects kidneys during edema treatment in heart failure.Formula:C18H24N4O3Color and Shape:SolidMolecular weight:344.41SUN 1334H
CAS:SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).Formula:C23H28Cl2F2N2O3Purity:98%Color and Shape:SolidMolecular weight:489.38DV 7028 hydrochloride
CAS:DV 7028 hydrochloride is a 5-HT2A receptor antagonist.Formula:C21H26ClFN4O3Purity:98%Color and Shape:SolidMolecular weight:436.91Usmarapride free base
CAS:Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.Formula:C21H29N5O2Purity:99.91% - 99.91%Color and Shape:SolidMolecular weight:383.49Colterol (free base)
CAS:Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.Formula:C12H19NO3Color and Shape:SolidMolecular weight:225.28S20928
CAS:S20928 is an antagonist of melatonin receptor.Formula:C17H19NOColor and Shape:SolidMolecular weight:253.342-Methyl-5-HT maleate
CAS:2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.Formula:C15H18N2O5Purity:98%Color and Shape:SolidMolecular weight:306.31Reversan
CAS:Reversan(CBLC4H10) is a potent, nontoxic, and glioblastoma-associated inhibitor of multidrug resistance-associated protein 1 (MRP1) and P-glycoprotein (Pgp).Formula:C26H27N5O2Purity:99.05%Color and Shape:SolidMolecular weight:441.53Ref: TM-T12714
1mg44.00€1mL*10mM (DMSO)92.00€5mg93.00€10mg130.00€25mg250.00€50mg401.00€100mg640.00€200mg884.00€
