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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • BL 6341A

    CAS:
    BL 6341A is related to Tumor data and H2-antagonists or anti-histamins
    Formula:C9H14N8OS3
    Color and Shape:Solid
    Molecular weight:346.46

    Ref: TM-T68703

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Carbuterol hydrochloride

    CAS:
    Carbuterol hydrochloride is a short-acting β2 adrenoreceptor agonist.
    Formula:C13H22ClN3O3
    Color and Shape:Solid
    Molecular weight:303.79

    Ref: TM-T69394

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cgp 52608

    CAS:
    CGP 52608 is a selective ligand for RAR-associated orphan receptor alpha.
    Formula:C8H12N4OS2
    Color and Shape:Solid
    Molecular weight:244.34

    Ref: TM-T30838

    25mg
    1,369.00€
  • Thromboxane B2

    CAS:
    Thromboxane B2 is a prostaglandin derivative that is released during anaphylaxis. Thromboxane B2 induces platelet aggregation and arterial contraction.
    Formula:C20H34O6
    Color and Shape:Solid
    Molecular weight:370.48

    Ref: TM-T41246

    25mg
    To inquire
    50mg
    To inquire
  • Amosulalol, (+)-

    CAS:
    Amosulalol, (+)-, is an adrenergic agent.
    Formula:C18H24N2O5S
    Color and Shape:Solid
    Molecular weight:380.46

    Ref: TM-T30029

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Z-335 sodium

    CAS:
    Z-335 Salt, a thromboxane A2 receptor antagonist, is used potentially for the treatment of arterial occlusive disease.
    Formula:C18H18ClNNaO4S
    Color and Shape:Solid
    Molecular weight:402.84

    Ref: TM-T29200

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • YM-430

    CAS:
    YM-430: β1 blocker & Ca²⁺ channel antagonist; antianginal & antihypertensive; IC50: 59.2 nM (rhythmic contractions), 36.6 mg/kg in rats (ST depression).
    Formula:C29H35N3O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.6

    Ref: TM-T29183

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Pirepemat fumarate

    CAS:
    Pirepemat fumarate (IRL752), aids Parkinson's research, boosts cognition and cortical catecholamine transmission.
    Formula:C15H17F2NO5
    Color and Shape:Solid
    Molecular weight:329.3

    Ref: TM-T60950

    25mg
    825.00€
    50mg
    1,071.00€
    100mg
    1,674.00€
  • NGD 98-2

    CAS:
    NGD 98-2 is a new generation, topology 2 selective orally active corticotropin releasing factor-1 (CRF-1) receptor antagonist.
    Formula:C19H24F3N3O3
    Color and Shape:Solid
    Molecular weight:399.41

    Ref: TM-T69374

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Trimazosin hydrochloride

    CAS:
    Trimazosin hydrochloride is used in the treatment of hypertensive patients failing to respond to thiazides.
    Formula:C20H32ClN5O7
    Color and Shape:Solid
    Molecular weight:489.95

    Ref: TM-T34945

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • mCPBG

    CAS:
    mCPBG is a potent high affinity agonist of 5-HT3 receptor.
    Formula:C8H10ClN5
    Color and Shape:Solid
    Molecular weight:211.65

    Ref: TM-T27987

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ChemR23-IN-2

    CAS:
    ChemR23-IN-2 is a potent, orally active inhibitor of ChemR23 (IC50: 3.2 nM).
    Formula:C29H26N4O5
    Color and Shape:Solid
    Molecular weight:510.54

    Ref: TM-T63520

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RX821002

    CAS:
    RX821002: potent α2-adrenoceptor antagonist, selective for α2D (pKd 9.7) over α2A (pKd 8.2), low affinity for imidazoline.
    Formula:C12H14N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:234.25

    Ref: TM-T28631

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-Azelastine

    CAS:
    (R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.
    Formula:C22H24ClN3O
    Color and Shape:Solid
    Molecular weight:381.9

    Ref: TM-T70675

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TP-680

    CAS:
    TP-680 is a antagonist of cholecystokininA receptor.
    Formula:C35H33N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:619.73

    Ref: TM-T28998

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Eptapirone fumarate

    CAS:
    Eptapirone (F11440) is a strong 5HT1A agonist with high anxiolytic and antidepressant effects, more potent than buspirone and flesinoxan.
    Formula:C20H27N7O6
    Color and Shape:Solid
    Molecular weight:461.479

    Ref: TM-T70183

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Metitepine

    CAS:
    Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.
    Formula:C20H24N2S2
    Color and Shape:Solid
    Molecular weight:356.55

    Ref: TM-T69988

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SNAP-5089

    CAS:
    SNAP-5089 is a highly selective alpha1A-adrenoceptor antagonist.
    Formula:C36H41ClN4O5
    Color and Shape:Solid
    Molecular weight:645.2

    Ref: TM-T70437

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Amibegron

    CAS:
    Amibegron: oral β3 adrenergic agonist, CNS-penetrating, with antidepressant and anxiolytic properties.
    Formula:C22H26ClNO4
    Color and Shape:Solid
    Molecular weight:403.9

    Ref: TM-T71216

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Mivazerol

    CAS:
    Mivazerol is an alpha 2-adrenoceptor agonist.
    Formula:C11H11N3O2
    Color and Shape:Solid
    Molecular weight:217.22

    Ref: TM-T71114

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€