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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • MRS2603

    CAS:
    MRS2603 is an antagonist of P2Y1 and P2Y13 receptors in 1321N1 human astrocytoma cells.
    Formula:C14H12ClN4O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.69

    Ref: TM-T28103

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CCG-224406

    CAS:
    CCG-22440 is a Highly Selective and Potent Inhibitor of G Protein-Coupled Receptor Kinase 2.
    Formula:C29H27FN6O5
    Color and Shape:Solid
    Molecular weight:558.56

    Ref: TM-T30777

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SLM6031434 HCl

    CAS:
    SLM6031434 HCl (SLM-6031434 HCl) is a SphK2 inhibitor that reduces LPS-induced TNF伪 and IL-1尾 production.
    Formula:C22H31ClF3N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.96

    Ref: TM-T28806

    1mg
    172.00€
    5mg
    533.00€
    10mg
    750.00€
  • A 68930 hydrochloride

    CAS:
    A68930 hydrochloride is a dopamine D1 receptor agonist which can be used for the research of bronchiectasis [1].
    Formula:C16H18ClNO3
    Color and Shape:Off-White Solid
    Molecular weight:307.77

    Ref: TM-T21680

    10mg
    645.00€
  • Usmarapride free base

    CAS:
    Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.
    Formula:C21H29N5O2
    Purity:99.91% - 99.91%
    Color and Shape:Solid
    Molecular weight:383.49

    Ref: TM-T34751

    1mg
    194.00€
  • Orexin receptor antagonist 2

    CAS:
    Compound 30, potent orexin antagonist with pKis of 7.69/9.78, potential for insomnia research.
    Formula:C25H31N5O2
    Color and Shape:Solid
    Molecular weight:433.55

    Ref: TM-T38139

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • SKF-104557

    CAS:
    N-Despropyl ropinirole, a ropinirole metabolite, enhances CHO cell acidification via D2/D3/D4 receptors; also a ropinirole impurity. EC50: 0.63-1.23 µM.
    Formula:C13H18N2O
    Color and Shape:Solid
    Molecular weight:218.29

    Ref: TM-T72003

    5mg
    537.00€
    10mg
    763.00€
    25mg
    1,755.00€
    50mg
    3,222.00€
  • Adenosine receptor antagonist 2

    CAS:
    Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.
    Formula:C23H21FN8O
    Color and Shape:Solid
    Molecular weight:444.46

    Ref: TM-T62611

    25mg
    1,791.00€
    50mg
    3,025.00€
  • JNJ-17156516

    CAS:
    JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.
    Formula:C26H22Cl2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.37

    Ref: TM-T27664

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bag-1

    CAS:
    Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.
    Formula:C22H27N3
    Color and Shape:Solid
    Molecular weight:333.47

    Ref: TM-T71595

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • CP 135807

    CAS:
    CP 135807 is a 5-HT1D receptor agonist.
    Formula:C19H21N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.4

    Ref: TM-T22681

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Fonazine hydrochloride

    CAS:
    Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.
    Formula:C19H26ClN3O2S2
    Color and Shape:Solid
    Molecular weight:428.01

    Ref: TM-T69407

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Reproterol hydrochloride

    CAS:
    Reproterol hydrochloride, a β2 adrenoreceptor agonist, is used to treat asthma and chronic obstructive pulmonary disease (COPD).
    Formula:C18H24ClN5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.87

    Ref: TM-T28519

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Zimelidine

    CAS:
    Zimelidine, a withdrawn antidepressant, posed Guillain-Barre risk.
    Formula:C16H17BrN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:317.22

    Ref: TM-T29216

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RP-72540

    CAS:
    RP-72540: CCKB receptor blocker, 200x more selective for CCKA, binds to stomach gastrin, limits [3H]pCCK-8 in mouse brain, <0.01% reaches forebrain.
    Formula:C28H30N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:518.56

    Ref: TM-T28612

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-Bambuterol

    CAS:
    Bambuterol is a β2-agonist prodrug for asthma and COPD, taken daily, with a good safety profile and reduces plasma LDL-C and cholesterol.
    Formula:C18H29N3O5
    Color and Shape:Solid
    Molecular weight:367.44

    Ref: TM-T68695

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Glucagon Receptor Antagonist I

    CAS:
    Glucagon antagonist I blocks the GCGR (IC50=181 nM), stops glucagon-induced glycogenolysis, and lowers glucose in glucagon-treated humanized mice.
    Formula:C20H30N2OS
    Color and Shape:Solid
    Molecular weight:346.53

    Ref: TM-T37223

    1mg
    430.00€
    5mg
    1,549.00€
  • Opaganib HCl

    CAS:
    ABC294640 (Opaganib) is an SK2 inhibitor with potential anti-cancer effects; it blocks S1P production to induce apoptosis.
    Formula:C23H26Cl2N2O
    Color and Shape:Solid
    Molecular weight:417.37

    Ref: TM-T71301

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-06412154 HCl

    CAS:
    PF-06412154 HCl is a glucagon receptor antagonist.
    Formula:C24H28ClN3O3
    Color and Shape:Solid
    Molecular weight:441.96

    Ref: TM-T70712

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Proxodolol hydrochloride

    CAS:
    Proxodolol, a β-adrenergic receptor antagonist, is used potentially for the treatment of glaucoma, hypertension and angina.
    Formula:C17H26ClN3O4
    Color and Shape:Solid
    Molecular weight:371.86

    Ref: TM-T28457

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€