
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,025 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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AZD-1678
CAS:AZD-1678 is a potent CCR4 receptor antagonist.Formula:C11H8Cl2FN3O3SColor and Shape:SolidMolecular weight:352.17LEI 101 hydrochloride
CAS:LEI 101 hydrochloride is potent and selective CB2 partial agonist.Formula:C23H26ClFN4O4SColor and Shape:SolidMolecular weight:508.99MPCI
CAS:MPCI is a selective melanocortin-4 receptor antagonist.Formula:C25H32BrFN4O2Purity:98%Color and Shape:SolidMolecular weight:519.45(R)-Azelastine
CAS:(R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H24ClN3OColor and Shape:SolidMolecular weight:381.9TP-680
CAS:TP-680 is a antagonist of cholecystokininA receptor.Formula:C35H33N5O4SPurity:98%Color and Shape:SolidMolecular weight:619.73SCH-202676 HBr
CAS:SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.Formula:C15H13N3SPurity:98%Color and Shape:SolidMolecular weight:267.35FR-171113
CAS:Protease-activated receptor 1 antagonistFormula:C19H11Cl3N2O4SPurity:98%Color and Shape:SolidMolecular weight:469.73Piclozotan
CAS:Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)Formula:C23H24ClN3O2Purity:98.59%Color and Shape:SolidMolecular weight:409.91ADR-851 HCl
CAS:ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.Formula:C14H19Cl2N3O2Purity:98%Color and Shape:SolidMolecular weight:332.23VUF8507
CAS:Vuf8507 is an allosteric regulator of adenosine receptor.Formula:C21H15N3OColor and Shape:SolidMolecular weight:325.36A-65186
CAS:A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.Formula:C25H35N3O4Purity:98.85% - 99.94%Color and Shape:SolidMolecular weight:441.56(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:5-HT1A serotonin receptor agonistFormula:C16H26BrNOPurity:98%Color and Shape:SolidMolecular weight:328.29E2508
CAS:E2508 is a selective antagonist of corticotropin-releasing factor 1 receptor.Formula:C36H47N3O7SPurity:98%Color and Shape:SolidMolecular weight:665.84Trimipramine
CAS:Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.Formula:C20H26N2Purity:98%Color and Shape:SolidMolecular weight:294.43Amibegron
CAS:Amibegron: oral β3 adrenergic agonist, CNS-penetrating, with antidepressant and anxiolytic properties.Formula:C22H26ClNO4Color and Shape:SolidMolecular weight:403.9SKF 77434 hydrobromide
CAS:SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.Formula:C19H22BrNO2Purity:98%Color and Shape:SolidMolecular weight:376.29Butopamine
CAS:Butopamine differs from dobutamine in location of only one hydroxyl group, but is no longer a catecholamine.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38R 75317
CAS:R 75317 is a Platelet-activating factor (PAF) antagonist.Formula:C29H50N3O8PSPurity:98%Color and Shape:SolidMolecular weight:631.765-OxoETE methyl ester
CAS:5-OxoETE methyl ester is a 5-oxoETE ester, an OXER1 agonist with stronger β-arrestin response, EC50 = 1.54 μM.Formula:C21H32O3Color and Shape:SolidMolecular weight:332.48FR 139317
CAS:highly potent and selective ETA endothelin receptor antagonistFormula:C33H44N6O5Purity:98%Color and Shape:SolidMolecular weight:604.74
