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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • AZD-1678

    CAS:
    AZD-1678 is a potent CCR4 receptor antagonist.
    Formula:C11H8Cl2FN3O3S
    Color and Shape:Solid
    Molecular weight:352.17

    Ref: TM-T26713

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LEI 101 hydrochloride

    CAS:
    LEI 101 hydrochloride is potent and selective CB2 partial agonist.
    Formula:C23H26ClFN4O4S
    Color and Shape:Solid
    Molecular weight:508.99

    Ref: TM-T69732

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MPCI

    CAS:
    MPCI is a selective melanocortin-4 receptor antagonist.
    Formula:C25H32BrFN4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:519.45

    Ref: TM-T24495

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-Azelastine

    CAS:
    (R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.
    Formula:C22H24ClN3O
    Color and Shape:Solid
    Molecular weight:381.9

    Ref: TM-T70675

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TP-680

    CAS:
    TP-680 is a antagonist of cholecystokininA receptor.
    Formula:C35H33N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:619.73

    Ref: TM-T28998

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SCH-202676 HBr

    CAS:
    SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.
    Formula:C15H13N3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.35

    Ref: TM-T24770

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • FR-171113

    CAS:
    Protease-activated receptor 1 antagonist
    Formula:C19H11Cl3N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:469.73

    Ref: TM-T22792

    10mg
    883.00€
    50mg
    3,718.00€
  • Piclozotan

    CAS:
    Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)
    Formula:C23H24ClN3O2
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:409.91

    Ref: TM-T28414

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ADR-851 HCl

    CAS:
    ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.
    Formula:C14H19Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.23

    Ref: TM-T23642L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • VUF8507

    CAS:
    Vuf8507 is an allosteric regulator of adenosine receptor.
    Formula:C21H15N3O
    Color and Shape:Solid
    Molecular weight:325.36

    Ref: TM-T35086

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A-65186

    CAS:
    A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.
    Formula:C25H35N3O4
    Purity:98.85% - 99.94%
    Color and Shape:Solid
    Molecular weight:441.56

    Ref: TM-T26483

    1mg
    279.00€
    5mg
    685.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€
  • (R)-(+)-8-Hydroxy-DPAT hydrobromide

    CAS:
    5-HT1A serotonin receptor agonist
    Formula:C16H26BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.29

    Ref: TM-T23218

    10mg
    735.00€
    50mg
    3,052.00€
  • E2508

    CAS:
    E2508 is a selective antagonist of corticotropin-releasing factor 1 receptor.
    Formula:C36H47N3O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:665.84

    Ref: TM-T27227

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Trimipramine

    CAS:
    Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.
    Formula:C20H26N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:294.43

    Ref: TM-T21364

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Amibegron

    CAS:
    Amibegron: oral β3 adrenergic agonist, CNS-penetrating, with antidepressant and anxiolytic properties.
    Formula:C22H26ClNO4
    Color and Shape:Solid
    Molecular weight:403.9

    Ref: TM-T71216

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SKF 77434 hydrobromide

    CAS:
    SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.
    Formula:C19H22BrNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.29

    Ref: TM-T23360

    5mg
    233.00€
  • Butopamine

    CAS:
    Butopamine differs from dobutamine in location of only one hydroxyl group, but is no longer a catecholamine.
    Formula:C18H23NO3
    Color and Shape:Solid
    Molecular weight:301.38

    Ref: TM-T30630

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • R 75317

    CAS:
    R 75317 is a Platelet-activating factor (PAF) antagonist.
    Formula:C29H50N3O8PS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:631.76

    Ref: TM-T26022

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • 5-OxoETE methyl ester

    CAS:
    5-OxoETE methyl ester is a 5-oxoETE ester, an OXER1 agonist with stronger β-arrestin response, EC50 = 1.54 μM.
    Formula:C21H32O3
    Color and Shape:Solid
    Molecular weight:332.48

    Ref: TM-T37304

    25µg
    305.00€
    50µg
    577.00€
    100µg
    1,063.00€
    250µg
    2,395.00€
  • FR 139317

    CAS:
    highly potent and selective ETA endothelin receptor antagonist
    Formula:C33H44N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:604.74

    Ref: TM-T22791

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€