
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,025 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Brl 22321
CAS:Brl 22321 is a mast cell stabilizer.Formula:C12H9N3O2Color and Shape:SolidMolecular weight:227.22CP 96345
CAS:CP 96345 is a NK1 receptor antagonist.Formula:C28H32N2OPurity:98%Color and Shape:SolidMolecular weight:412.57KW-8232
CAS:KW-8232, an orally active anti-osteoporotic agent, reduces the biosynthesis of PGE2[1].Formula:C37H41ClN4O6SColor and Shape:SolidMolecular weight:705.27Hexoprenaline
CAS:Hexoprenaline is a stimulant of adrenergic beta 2 receptors used as a bronchodilator, antiasthmatic agent, and tocolytic agent.Formula:C22H32N2O6Color and Shape:SolidMolecular weight:420.5SMANT hydrochloride
CAS:SMANT hydrochloride (N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide hydrochloride) is an antagonist of Smoothened accumulation.Formula:C16H24BrClN2OPurity:99.81%Color and Shape:SolidMolecular weight:375.73CAY10498
CAS:A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.Formula:C18H20N6Color and Shape:SolidMolecular weight:320.39Daledalin
CAS:Daledalin, an unmarketed 1970s antidepressant, is a selective norepinephrine reuptake inhibitor without serotonergic or dopaminergic effects.Formula:C19H24N2Color and Shape:SolidMolecular weight:280.41MRS2603
CAS:MRS2603 is an antagonist of P2Y1 and P2Y13 receptors in 1321N1 human astrocytoma cells.Formula:C14H12ClN4O8PPurity:98%Color and Shape:SolidMolecular weight:430.69Fenspiride-d5
CAS:Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.Formula:C15H15D5N2O2Color and Shape:SolidMolecular weight:265.36Monatepil maleate
CAS:Monatepil maleate (AJ-2615 maleate) is a Ca2+-channel and α1-adrenergic receptor antagonist, and ACAT inhibitor with antihypertensive activity.Formula:C32H34FN3O5SPurity:97.90%Color and Shape:SolidMolecular weight:591.69CCG-224406
CAS:CCG-22440 is a Highly Selective and Potent Inhibitor of G Protein-Coupled Receptor Kinase 2.Formula:C29H27FN6O5Color and Shape:SolidMolecular weight:558.56CCG-271423
CAS:CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.Formula:C28H26N4O3Color and Shape:SolidMolecular weight:466.53AK-IN-1
CAS:AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.Formula:C22H21N3O4Color and Shape:SolidMolecular weight:391.42A 69024
CAS:A 69024 is a highly selective antagonist of dopamine D-1 receptor.Formula:C20H24BrNO4Purity:98%Color and Shape:SolidMolecular weight:422.31Impromidine
CAS:Impromidine is a highly potent and specific agonist of the histamine H2 receptor.Formula:C14H23N7SPurity:98%Color and Shape:SolidMolecular weight:321.44PF-3246799
CAS:PF-3246799 is an effective and selective agonist of the 5-HT2C receptor.Formula:C15H17N3Purity:98%Color and Shape:SolidMolecular weight:239.32CCR1 antagonist 7
CAS:CCR1 antagonist 7 (compound 16r) is an antagonist of chemokine receptor 1 (CCR1) with an IC 50 of 4 nM [1].Formula:C21H24ClN5O3SPurity:98%Color and Shape:SolidMolecular weight:461.96PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Formula:C17H21N3Purity:98%Color and Shape:SolidMolecular weight:267.37S 14506 hydrochloride
CAS:S 14506 hydrochloride is a 5-HT1A receptor full agonist.Formula:C24H27ClFN3O2Purity:99.92%Color and Shape:SolidMolecular weight:443.94UNC9975
CAS:UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.Formula:C23H28Cl2N4O2Purity:98.78% - 98.78%Color and Shape:SolidMolecular weight:463.4
