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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • Brl 22321

    CAS:
    Brl 22321 is a mast cell stabilizer.
    Formula:C12H9N3O2
    Color and Shape:Solid
    Molecular weight:227.22

    Ref: TM-T30587

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CP 96345

    CAS:
    CP 96345 is a NK1 receptor antagonist.
    Formula:C28H32N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.57

    Ref: TM-T22690

    10mg
    888.00€
  • KW-8232

    CAS:
    KW-8232, an orally active anti-osteoporotic agent, reduces the biosynthesis of PGE2[1].
    Formula:C37H41ClN4O6S
    Color and Shape:Solid
    Molecular weight:705.27

    Ref: TM-T36762

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Hexoprenaline

    CAS:
    Hexoprenaline is a stimulant of adrenergic beta 2 receptors used as a bronchodilator, antiasthmatic agent, and tocolytic agent.
    Formula:C22H32N2O6
    Color and Shape:Solid
    Molecular weight:420.5

    Ref: TM-T25499

    25mg
    1,369.00€
  • SMANT hydrochloride

    CAS:
    SMANT hydrochloride (N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide hydrochloride) is an antagonist of Smoothened accumulation.
    Formula:C16H24BrClN2O
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:375.73

    Ref: TM-T23370

    10mg
    42.00€
    25mg
    78.00€
    50mg
    123.00€
    100mg
    202.00€
    200mg
    294.00€
  • CAY10498

    CAS:
    A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.
    Formula:C18H20N6
    Color and Shape:Solid
    Molecular weight:320.39

    Ref: TM-T37669

    500µg
    386.00€
    1mg
    712.00€
    5mg
    3,132.00€
  • Daledalin

    CAS:
    Daledalin, an unmarketed 1970s antidepressant, is a selective norepinephrine reuptake inhibitor without serotonergic or dopaminergic effects.
    Formula:C19H24N2
    Color and Shape:Solid
    Molecular weight:280.41

    Ref: TM-T69788

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS2603

    CAS:
    MRS2603 is an antagonist of P2Y1 and P2Y13 receptors in 1321N1 human astrocytoma cells.
    Formula:C14H12ClN4O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.69

    Ref: TM-T28103

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Fenspiride-d5

    CAS:
    Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.
    Formula:C15H15D5N2O2
    Color and Shape:Solid
    Molecular weight:265.36

    Ref: TM-T71141

    1mg
    1,018.00€
    5mg
    3,312.00€
  • Monatepil maleate

    CAS:
    Monatepil maleate (AJ-2615 maleate) is a Ca2+-channel and α1-adrenergic receptor antagonist, and ACAT inhibitor with antihypertensive activity.
    Formula:C32H34FN3O5S
    Purity:97.90%
    Color and Shape:Solid
    Molecular weight:591.69

    Ref: TM-T25828

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • CCG-224406

    CAS:
    CCG-22440 is a Highly Selective and Potent Inhibitor of G Protein-Coupled Receptor Kinase 2.
    Formula:C29H27FN6O5
    Color and Shape:Solid
    Molecular weight:558.56

    Ref: TM-T30777

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CCG-271423

    CAS:
    CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.
    Formula:C28H26N4O3
    Color and Shape:Solid
    Molecular weight:466.53

    Ref: TM-T62986

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AK-IN-1

    CAS:
    AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.
    Formula:C22H21N3O4
    Color and Shape:Solid
    Molecular weight:391.42

    Ref: TM-T73436

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • A 69024

    CAS:
    A 69024 is a highly selective antagonist of dopamine D-1 receptor.
    Formula:C20H24BrNO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:422.31

    Ref: TM-T26433

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Impromidine

    CAS:
    Impromidine is a highly potent and specific agonist of the histamine H2 receptor.
    Formula:C14H23N7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.44

    Ref: TM-T24162

    25mg
    1,586.00€
    50mg
    2,072.00€
    100mg
    2,660.00€
  • PF-3246799

    CAS:
    PF-3246799 is an effective and selective agonist of the 5-HT2C receptor.
    Formula:C15H17N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:239.32

    Ref: TM-T24627

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • CCR1 antagonist 7

    CAS:
    CCR1 antagonist 7 (compound 16r) is an antagonist of chemokine receptor 1 (CCR1) with an IC 50 of 4 nM [1].
    Formula:C21H24ClN5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:461.96

    Ref: TM-T10709

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-04781340

    CAS:
    PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.
    Formula:C17H21N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.37

    Ref: TM-T24616

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • S 14506 hydrochloride

    CAS:
    S 14506 hydrochloride is a 5-HT1A receptor full agonist.
    Formula:C24H27ClFN3O2
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:443.94

    Ref: TM-T23285

    2mg
    47.00€
    5mg
    67.00€
    10mg
    101.00€
    25mg
    197.00€
    50mg
    304.00€
    100mg
    457.00€
    200mg
    650.00€
  • UNC9975

    CAS:
    UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.
    Formula:C23H28Cl2N4O2
    Purity:98.78% - 98.78%
    Color and Shape:Solid
    Molecular weight:463.4

    Ref: TM-T29064

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€