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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5990 products of "GPCR/G-Protein"

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  • Guanethidine

    CAS:
    Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.
    Formula:C10H22N4
    Color and Shape:Solid
    Molecular weight:198.31

    Ref: TM-T50109

    100mg
    To inquire
    500mg
    To inquire
  • Fonazine mesylate

    CAS:
    Fonazine mesylate is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.
    Formula:C20H29N3O5S3
    Color and Shape:Solid
    Molecular weight:487.65

    Ref: TM-T70997

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • A2AR-agonist-1

    CAS:
    A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).
    Formula:C20H22N6O4
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:410.43

    Ref: TM-T10212

    1mg
    90.00€
    2mg
    127.00€
    5mg
    178.00€
    1mL*10mM (DMSO)
    207.00€
    10mg
    269.00€
    25mg
    427.00€
    50mg
    610.00€
    100mg
    820.00€
    500mg
    1,603.00€
  • Flerobuterol HCl

    CAS:
    "Flerobuterol, a β adrenergic agonist, may treat depression by boosting serotonin synthesis and Trp in the brain."
    Formula:C12H19ClFNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:247.74

    Ref: TM-T27331

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Aminaftone

    CAS:
    Aminaftone, a derivative of 4-aminobenzoic acid, inhibits endothelin-1 (ET-1) production and can be used to study hypertension and systemic sclerosis.
    Formula:C18H15NO4
    Purity:96.31% - 99.39%
    Color and Shape:Solid
    Molecular weight:309.32

    Ref: TM-T14219

    1mg
    190.00€
    5mg
    523.00€
    10mg
    648.00€
    25mg
    858.00€
  • EP4 receptor antagonist 4

    CAS:
    EP4 receptor antagonist 4 is an agonist of EP4 receptor (human pEC 50 = 6.3) [1].
    Formula:C19H14N2OS
    Color and Shape:Solid
    Molecular weight:318.39

    Ref: TM-T60840

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Brl 22321

    CAS:
    Brl 22321 is a mast cell stabilizer.
    Formula:C12H9N3O2
    Color and Shape:Solid
    Molecular weight:227.22

    Ref: TM-T30587

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • FR-171113

    CAS:
    Protease-activated receptor 1 antagonist
    Formula:C19H11Cl3N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:469.73

    Ref: TM-T22792

    10mg
    883.00€
    50mg
    3,718.00€
  • ADR-851 HCl

    CAS:
    ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.
    Formula:C14H19Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.23

    Ref: TM-T23642L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • E2508

    CAS:
    E2508 is a selective antagonist of corticotropin-releasing factor 1 receptor.
    Formula:C36H47N3O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:665.84

    Ref: TM-T27227

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-Bambuterol

    CAS:
    Bambuterol is a β2-agonist prodrug for asthma and COPD, taken daily, with a good safety profile and reduces plasma LDL-C and cholesterol.
    Formula:C18H29N3O5
    Color and Shape:Solid
    Molecular weight:367.44

    Ref: TM-T68695

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cannabicitran

    CAS:
    Cannabicitran is a cannabinoid that can decrease rabbits intraocular pressure [1] [2].
    Formula:C21H30O2
    Color and Shape:Solid
    Molecular weight:314.46

    Ref: TM-T60807

    1mg
    389.00€
  • Trimipramine

    CAS:
    Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.
    Formula:C20H26N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:294.43

    Ref: TM-T21364

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UNC9975

    CAS:
    UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.
    Formula:C23H28Cl2N4O2
    Purity:98.78% - 98.78%
    Color and Shape:Solid
    Molecular weight:463.4

    Ref: TM-T29064

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • VUF8504

    CAS:
    VUF8504 is a novel ligand of adenosine A3 receptor.
    Formula:C22H17N3O2
    Color and Shape:Solid
    Molecular weight:355.39

    Ref: TM-T29148

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB-269970

    CAS:
    SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).
    Formula:C18H28N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.49

    Ref: TM-T12842

    25mg
    2,178.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • FR 139317

    CAS:
    highly potent and selective ETA endothelin receptor antagonist
    Formula:C33H44N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:604.74

    Ref: TM-T22791

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EMD 56551

    CAS:
    EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.
    Formula:C24H31N3O2
    Purity:95.64% - 99.39%
    Color and Shape:Solid
    Molecular weight:393.522

    Ref: TM-T61816

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • EP1-antagonist-1

    CAS:
    EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).
    Formula:C19H15BrCl2N2O3
    Purity:97.06%
    Color and Shape:Solid
    Molecular weight:470.14

    Ref: TM-T10031

    1mg
    109.00€
    5mg
    215.00€
    1mL*10mM (DMSO)
    243.00€
    10mg
    313.00€
    25mg
    492.00€
  • S-22153

    CAS:
    S22153 is an antagonist of melatonin receptor.
    Formula:C14H17NOS
    Color and Shape:Solid
    Molecular weight:247.36

    Ref: TM-T28645

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€