GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
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Captodiame
CAS:Captodiame is an antihistamine agent.Formula:C21H29NS2Purity:98%Color and Shape:SolidMolecular weight:359.59S(-)-8-Hydroxy-DPAT hydrobromide
CAS:S(-)-8-Hydroxy-DPAT hydrobromide is an agonist of 5-HT1A serotonin receptor.Formula:C16H26BrNOPurity:98%Color and Shape:SolidMolecular weight:328.29PD 118440
CAS:PD 118440 is a Dopamine antagonist. PD 118440 is an orally active dopamine (DA) agonists with pronounced central nervous system effects.Formula:C11H17N3SPurity:98%Color and Shape:SolidMolecular weight:223.34NVP-QAV-680
CAS:NVP-QAV-680: Powerful, selective CRTh2 antagonist with nM potency inhibiting eosinophil/Th2 activation.Formula:C18H18N2O4SPurity:98%Color and Shape:SolidMolecular weight:358.41GW-876167
CAS:GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.Formula:C16H21N5O2Purity:98%Color and Shape:SolidMolecular weight:315.37SB 272183
CAS:SB 272183 is a highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drug.Formula:C29H28ClN5OPurity:98%Color and Shape:SolidMolecular weight:498.02Sch 24518
CAS:Sc h24518 is an antagonist of D1 receptor.Formula:C16H17BrClNOPurity:98%Color and Shape:SolidMolecular weight:354.67Tilisolol HCl
CAS:Tilisolol, a nonselective beta-blocker, dilates dog coronary arteries via ATP-sensitive K(+) channels.Formula:C17H25ClN2O3Purity:98%Color and Shape:SolidMolecular weight:340.85MK-0249
CAS:MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
Formula:C23H24F3N3O2Purity:99.90%Color and Shape:SolidMolecular weight:431.45H3 receptor-MO-1
CAS:H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.Formula:C20H27N3O2Purity:99.11%Color and Shape:SolidMolecular weight:341.45Rocastine
CAS:Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.Formula:C13H19N3OSPurity:98.26%Color and Shape:SolidMolecular weight:265.37QF0301B
CAS:QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.Formula:C23H28N2O2Purity:>99.99%Color and Shape:SolidMolecular weight:364.48Tulopafant
CAS:Tulopafant (RP 59227) is a potent platelet-activating factor (PAF) antagonist that increases capillary patency and prolongs allograft heart survival.Formula:C25H19N3O2SPurity:99.38%Color and Shape:SolidMolecular weight:425.5Isoproterenol-d7 HCl
CAS:Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.Formula:C11H18ClNO3Color and Shape:SolidMolecular weight:254.76CCK-A receptor inhibitor 1
CAS:CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the studyFormula:C25H35NO6SPurity:99.47%Color and Shape:SolidMolecular weight:477.61Pamatolol
CAS:Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.Formula:C16H26N2O4Purity:>99.99%Color and Shape:SolidMolecular weight:310.39Cicloprolol hydrochloride
CAS:Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.Formula:C18H30ClNO4Purity:97.26%Color and Shape:SolidMolecular weight:359.89Bamirastine
CAS:Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect onFormula:C31H37N5O3Purity:96.68%Color and Shape:SolidMolecular weight:527.66(4E)-SUN9221
CAS:(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity inFormula:C25H31FN4O3Purity:97.79%Color and Shape:SolidMolecular weight:454.54L-771688
CAS:L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benignFormula:C28H33F2N5O5Purity:94.15%Color and Shape:SolidMolecular weight:557.59
