GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5988 products of "GPCR/G-Protein"
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Lusaperidone
CAS:Kaerophyllin ( (-)-Kaerophylin) inhibits hepatic stellate cell activation and inhibits HSC activation to protect against liver cell damage and fibrosis in rats.Formula:C22H21N3O2Purity:99.75%Color and Shape:SolidMolecular weight:359.42Tecalcet Hydrochloride
CAS:Tecalcet Hydrochloride, an allosteric CaSR modulator, enhances extracellular Ca2+ sensitivity.Formula:C18H23Cl2NOPurity:99.97%Color and Shape:SolidMolecular weight:340.29Ref: TM-T13918
200mgTo inquire2mg34.00€5mg47.00€1mL*10mM (DMSO)52.00€10mg72.00€25mg146.00€50mg230.00€100mg335.00€A2AR-antagonist-1
CAS:Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.Formula:C27H25N5O2Purity:98%Color and Shape:SolidMolecular weight:451.52Moprolol
CAS:Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] [2] [3].Formula:C13H21NO3Purity:98%Color and Shape:SolidMolecular weight:239.31A-77636
CAS:A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective concentration (EC50) of 1.1 nM and a corresponding pEC50Formula:C20H27NO3Purity:98%Color and Shape:SolidMolecular weight:329.43Dicarbine
CAS:Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.Formula:C13H18N2Purity:98%Color and Shape:SolidMolecular weight:202.3NPS ALX Compound 4a dihydrochloride
CAS:NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formula:C25H27Cl2N3O2SPurity:98%Color and Shape:SolidMolecular weight:504.47WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Formula:C14H18N2Purity:98%Color and Shape:SolidMolecular weight:214.31ROS 234 dioxalate
CAS:ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)Formula:C17H19N5O8Purity:98%Color and Shape:SolidMolecular weight:421.37Ipsapirone
CAS:Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.
Formula:C19H23N5O3SPurity:99.51%Color and Shape:SolidMolecular weight:401.48ESI-08
CAS:ESI-08 is an effective antagonist of EPAC2 with an IC50 of 8.4 μM. ESI-08 selectively blocks cAMP-induced EPAC activation but not cAMP-mediated PKA activation.Formula:C20H23N3OSPurity:97.17%Color and Shape:SolidMolecular weight:353.48CP-226269
CAS:CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.
Formula:C18H19FN4Purity:99.08%Color and Shape:SolidMolecular weight:310.37Mianserin
CAS:Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.Formula:C18H20N2Purity:99.85%Color and Shape:SolidMolecular weight:264.36MRE3008F20
CAS:MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.Formula:C21H20N8O3Purity:97.29%Color and Shape:SolidMolecular weight:432.44Wy 49051
CAS:Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).Formula:C28H33N5O3Purity:99.89%Color and Shape:SolidMolecular weight:487.59Ref: TM-T13352
1mg99.00€5mg188.00€1mL*10mM (DMSO)250.00€10mg273.00€25mg427.00€50mg575.00€100mg743.00€200mg990.00€PF-03654746
CAS:PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.Formula:C18H24F2N2OPurity:98.85% - 99.57%Color and Shape:SolidMolecular weight:322.39Cinitapride Hydrogen Tartrate
CAS:Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptorsFormula:C25H36N4O10Purity:98%Color and Shape:SolidMolecular weight:552.581Lintopride
CAS:Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.Formula:C14H19ClN4O2Purity:98%Color and Shape:SolidMolecular weight:310.78Apadenoson
CAS:Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.Formula:C23H30N6O6Purity:98%Color and Shape:SolidMolecular weight:486.52Arbutamine
CAS:Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to study cardiac stress.
Formula:C18H23NO4Purity:95.06%Color and Shape:SolidMolecular weight:317.38
