
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5986 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Pargolol
CAS:Pargolol is a beta adrenergic receptor antagonist.Formula:C16H23NO3Color and Shape:SolidMolecular weight:277.36Colterol (free base)
CAS:Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.Formula:C12H19NO3Color and Shape:SolidMolecular weight:225.28CP 66713
CAS:CP-66713 is an adenosine A2 receptor antagonist.Formula:C15H10ClN5Color and Shape:SolidMolecular weight:295.73AM-211 sodium
CAS:AM-211 sodium: potent DP2 receptor antagonist, active against allergic inflammation, selective, and orally bioavailable in rats and dogs.Formula:C27H26F3N2NaO4Color and Shape:SolidMolecular weight:522.5ST1936
CAS:ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.Formula:C13H17ClN2Purity:98%Color and Shape:SolidMolecular weight:236.74Ref: TM-T23396
1mg44.00€5mg111.00€1mL*10mM (DMSO)123.00€10mg178.00€25mg316.00€50mg470.00€100mg682.00€200mg954.00€BMY-25271
CAS:BMY-25271 is an antagonist of histamine H2 receptor.Formula:C12H19N5O2S2Purity:98%Color and Shape:SolidMolecular weight:329.44Adatanserin
CAS:Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.Formula:C21H31N5OPurity:99.33%Color and Shape:SolidMolecular weight:369.5Savoxepin mesylate
CAS:Savoxepin mesylate, a tetracyclic cyano-dibenzoxepino-azepine derivative, has potent antidopaminergic activity.Formula:C26H30N2O4SPurity:98%Color and Shape:SolidMolecular weight:466.59LEQ-506
CAS:LEQ506, an oral Smoothened antagonist, may inhibit cancer growth by blocking the Hedgehog signaling pathway.Formula:C27H29N5OColor and Shape:SolidMolecular weight:439.55PF-4522654
CAS:PF-4522654 is a potent and selective 5-HT2C receptor agonist.Formula:C16H18F2N4Color and Shape:SolidMolecular weight:304.34Bemesetron
CAS:Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.Formula:C15H17Cl2NO2Purity:99.77%Color and Shape:SolidMolecular weight:314.21NR2F1 agonist 1
CAS:NR2F1 agonist 1 activates cancer cell dormancy, suppresses growth in HNSCC, and inhibits tumor growth in mice.Formula:C28H30N4OSColor and Shape:SolidMolecular weight:470.63Fallypride
CAS:Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.Formula:C20H29FN2O3Purity:98.97% - >99.99%Color and Shape:SolidMolecular weight:364.45Ref: TM-T70302
1mg340.00€1mL*10mM (DMSO)640.00€5mg797.00€10mg982.00€25mg1,575.00€50mg1,963.00€100mg2,520.00€Zelandopam free base
CAS:Zelandopam: dopamine D1 agonist, boosts pancreatic secretion, renal vasodilator, counters renal dysfunction.Formula:C15H15NO4Color and Shape:SolidMolecular weight:273.28Isamoltane
CAS:Isamoltane is a serotonin 5-HT1 Receptor AntagonistFormula:C16H23ClN2O2Color and Shape:SolidMolecular weight:310.82Ro 63-0563
CAS:Ro 63-0563 is a potent, 5-HT6 receptors selective antagonist.Formula:C13H17N5O2SPurity:98%Color and Shape:SolidMolecular weight:307.37cis-Epoxysuccinic acid
CAS:cis-Epoxysuccinic acid is a potential agonist of Succinate receptor 1 and inhibitor of Isocitrate lyase 1 for use in biochemical experiments.Formula:C4H4O5Purity:99.81%Color and Shape:SolidMolecular weight:132.07BRL 44408 Maleate Salt
CAS:BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.Formula:C17H21N3O4Purity:98.71%Color and Shape:SolidMolecular weight:331.372-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
CAS:2-Decenoylaminoethyl cyclohexylethyl sulfide prevents stress ulcers, stabilizes phospholipase A2 and prostaglandin E2.Formula:C20H37NOSPurity:98%Color and Shape:SolidMolecular weight:339.58Etrasimod arginine
CAS:Etrasimod arginine is used in the Treatment of Autoimmune and Inflammatory Diseases.Formula:C32H40F3N5O5Color and Shape:SolidMolecular weight:631.69
