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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5986 products of "GPCR/G-Protein"

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  • Pargolol

    CAS:
    Pargolol is a beta adrenergic receptor antagonist.
    Formula:C16H23NO3
    Color and Shape:Solid
    Molecular weight:277.36

    Ref: TM-T69217

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Colterol (free base)

    CAS:
    Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.
    Formula:C12H19NO3
    Color and Shape:Solid
    Molecular weight:225.28

    Ref: TM-T70089

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CP 66713

    CAS:
    CP-66713 is an adenosine A2 receptor antagonist.
    Formula:C15H10ClN5
    Color and Shape:Solid
    Molecular weight:295.73

    Ref: TM-T31026

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AM-211 sodium

    CAS:
    AM-211 sodium: potent DP2 receptor antagonist, active against allergic inflammation, selective, and orally bioavailable in rats and dogs.
    Formula:C27H26F3N2NaO4
    Color and Shape:Solid
    Molecular weight:522.5

    Ref: TM-T71088

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ST1936

    CAS:
    ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.
    Formula:C13H17ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:236.74

    Ref: TM-T23396

    1mg
    44.00€
    5mg
    111.00€
    1mL*10mM (DMSO)
    123.00€
    10mg
    178.00€
    25mg
    316.00€
    50mg
    470.00€
    100mg
    682.00€
    200mg
    954.00€
  • BMY-25271

    CAS:
    BMY-25271 is an antagonist of histamine H2 receptor.
    Formula:C12H19N5O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.44

    Ref: TM-T10575

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Adatanserin

    CAS:
    Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.
    Formula:C21H31N5O
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:369.5

    Ref: TM-T23631

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • Savoxepin mesylate

    CAS:
    Savoxepin mesylate, a tetracyclic cyano-dibenzoxepino-azepine derivative, has potent antidopaminergic activity.
    Formula:C26H30N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:466.59

    Ref: TM-T28666

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • LEQ-506

    CAS:
    LEQ506, an oral Smoothened antagonist, may inhibit cancer growth by blocking the Hedgehog signaling pathway.
    Formula:C27H29N5O
    Color and Shape:Solid
    Molecular weight:439.55

    Ref: TM-T71520

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-4522654

    CAS:
    PF-4522654 is a potent and selective 5-HT2C receptor agonist.
    Formula:C16H18F2N4
    Color and Shape:Solid
    Molecular weight:304.34

    Ref: TM-T71507

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bemesetron

    CAS:
    Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.
    Formula:C15H17Cl2NO2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:314.21

    Ref: TM-T14526

    10mg
    52.00€
    25mg
    66.00€
    50mg
    89.00€
  • NR2F1 agonist 1

    CAS:
    NR2F1 agonist 1 activates cancer cell dormancy, suppresses growth in HNSCC, and inhibits tumor growth in mice.
    Formula:C28H30N4OS
    Color and Shape:Solid
    Molecular weight:470.63

    Ref: TM-T72776

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Fallypride

    CAS:
    Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.
    Formula:C20H29FN2O3
    Purity:98.97% - >99.99%
    Color and Shape:Solid
    Molecular weight:364.45

    Ref: TM-T70302

    1mg
    340.00€
    1mL*10mM (DMSO)
    640.00€
    5mg
    797.00€
    10mg
    982.00€
    25mg
    1,575.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Zelandopam free base

    CAS:
    Zelandopam: dopamine D1 agonist, boosts pancreatic secretion, renal vasodilator, counters renal dysfunction.
    Formula:C15H15NO4
    Color and Shape:Solid
    Molecular weight:273.28

    Ref: TM-T29213

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Isamoltane

    CAS:
    Isamoltane is a serotonin 5-HT1 Receptor Antagonist
    Formula:C16H23ClN2O2
    Color and Shape:Solid
    Molecular weight:310.82

    Ref: TM-T68176

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ro 63-0563

    CAS:
    Ro 63-0563 is a potent, 5-HT6 receptors selective antagonist.
    Formula:C13H17N5O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.37

    Ref: TM-T28594

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • cis-Epoxysuccinic acid

    CAS:
    cis-Epoxysuccinic acid is a potential agonist of Succinate receptor 1 and inhibitor of Isocitrate lyase 1 for use in biochemical experiments.
    Formula:C4H4O5
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:132.07

    Ref: TM-T71921

    50mg
    34.00€
    100mg
    47.00€
    1mL*10mM (DMSO)
    50.00€
    500mg
    77.00€
  • BRL 44408 Maleate Salt

    CAS:
    BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.
    Formula:C17H21N3O4
    Purity:98.71%
    Color and Shape:Solid
    Molecular weight:331.37

    Ref: TM-T26904

    1mg
    71.00€
    5mg
    155.00€
    10mg
    268.00€
    25mg
    442.00€
    50mg
    645.00€
    100mg
    950.00€
  • 2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide

    CAS:
    2-Decenoylaminoethyl cyclohexylethyl sulfide prevents stress ulcers, stabilizes phospholipase A2 and prostaglandin E2.
    Formula:C20H37NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:339.58

    Ref: TM-T13488

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Etrasimod arginine

    CAS:
    Etrasimod arginine is used in the Treatment of Autoimmune and Inflammatory Diseases.
    Formula:C32H40F3N5O5
    Color and Shape:Solid
    Molecular weight:631.69

    Ref: TM-T31726

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
    500mg
    3,137.00€