GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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EP1-antagonist-1
CAS:EP1-antagonist-1 (EP1 antagonist 1) is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).Formula:C19H15BrCl2N2O3Purity:97.06%Color and Shape:SolidMolecular weight:470.14EMD 56551
CAS:EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.Formula:C24H31N3O2Purity:95.64% - 99.39%Color and Shape:SolidMolecular weight:393.522(S)-(-)-Propranolol hydrochloride
CAS:(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂，具有抗高血压活性和潜在的抗癌活性，对β1，β2，和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后，可用于研究酒精症。Formula:C16H22ClNO2Purity:99.02% - 99.91%Color and Shape:SolidMolecular weight:295.8Befetupitant
CAS:Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.Formula:C29H29F6N3O2Purity:98.72%Color and Shape:SolidMolecular weight:565.55Aminaftone
CAS:Aminaftone, a derivative of 4-aminobenzoic acid, inhibits endothelin-1 (ET-1) production and can be used to study hypertension and systemic sclerosis.Formula:C18H15NO4Purity:96.31% - 99.39%Color and Shape:SolidMolecular weight:309.32AP521
CAS:AP521 is an agonist of the human 5-HT1A receptor (IC50: 94 nM).Formula:C20H19ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:402.89PG 01037 dihydrochloride
CAS:PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.Formula:C26H28Cl4N4OPurity:99.89%Color and Shape:SolidMolecular weight:554.34WAY208466 dihydrochloride
CAS:WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.Formula:C17H20Cl2FN3O2SPurity:98.43% - 99.56%Color and Shape:SolidMolecular weight:420.33AM6545
CAS:AM6545 is a CB1 receptor antagonist used in the study of obesity and diabetes.Formula:C26H23Cl2N5O3SPurity:97.03%Color and Shape:SolidMolecular weight:556.46LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Formula:C27H38ClN3OSPurity:98.06%Color and Shape:SolidMolecular weight:488.13Rp-cAMPS sodium
CAS:Rp-cAMPS sodium is a phosphorothioate analog of cAMP, a PKA inhibitor and cAMP antagonist that inhibits cAMP-dependent protein kinases.Formula:C10H11N5NaO5PSPurity:99.71%Color and Shape:SolidMolecular weight:367.25Aligeron
CAS:Aligeron is a non-selective prostaglandin (PG) antagonist that inhibits PGF2α- and PGE2-induced decreases in blood pressure in cats, and can be used to inhibitFormula:C20H24N2Purity:99.09% - >99.99%Color and Shape:SolidMolecular weight:292.42Vapitadine dihydrochloride
CAS:Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.Formula:C17H22Cl2N4OPurity:98.28% - 99.30%Color and Shape:SolidMolecular weight:369.292-Iodomelatonin
CAS:2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.Formula:C13H15IN2O2Purity:99.7%Color and Shape:SolidMolecular weight:358.17Ref: TM-T10073
10mg43.00€25mg79.00€50mg118.00€100mg178.00€200mg268.00€500mgTo inquire1mL*10mM (DMSO)34.00€TIK-301
CAS:TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM
Formula:C14H17ClN2O2Purity:98%Color and Shape:SolidMolecular weight:280.75GSK-239512
CAS:GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.Formula:C23H27N3O2Purity:99.62% - 99.74%Color and Shape:SolidMolecular weight:377.48GR 113808
CAS:GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.Formula:C19H27N3O4SPurity:98.16% - 99.96%Color and Shape:SolidMolecular weight:393.5ST3932
CAS:ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).Formula:C12H16N8OPurity:98%Color and Shape:SolidMolecular weight:288.31PRX933 hydrochloride
CAS:PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.Formula:C16H22ClN5O2Purity:99.51% - 99.89%Color and Shape:SolidMolecular weight:351.84Ref: TM-T12565
1mg338.00€5mg538.00€10mg858.00€25mg1,269.00€50mg1,720.00€100mg2,305.00€1mL*10mM (DMSO)618.00€H4R antagonist 1
CAS:H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, H3R.Formula:C11H11BrN8Color and Shape:SolidMolecular weight:335.16
