CymitQuimica logo
GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 19 more subcategories

Found 5983 products of "GPCR/G-Protein"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Cirazoline (free base)

    CAS:
    Cirazoline: full α1A agonist, partial α1B/D, nonselective α2 antagonist; potential vasoconstrictor.
    Formula:C13H16N2O
    Color and Shape:Solid
    Molecular weight:216.28

    Ref: TM-T69031

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SLM6031434 HCl

    CAS:
    SLM6031434 HCl (SLM-6031434 HCl) is a SphK2 inhibitor that reduces LPS-induced TNF伪 and IL-1尾 production.
    Formula:C22H31ClF3N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.96

    Ref: TM-T28806

    1mg
    172.00€
    5mg
    533.00€
    10mg
    750.00€
  • ST-836

    CAS:
    ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .
    Formula:C23H34N4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.61

    Ref: TM-T13025

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SNAP-5089

    CAS:
    SNAP-5089 is a highly selective alpha1A-adrenoceptor antagonist.
    Formula:C36H41ClN4O5
    Color and Shape:Solid
    Molecular weight:645.2

    Ref: TM-T70437

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Mivazerol

    CAS:
    Mivazerol is an alpha 2-adrenoceptor agonist.
    Formula:C11H11N3O2
    Color and Shape:Solid
    Molecular weight:217.22

    Ref: TM-T71114

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-Praziquantel

    CAS:
    (R)-Praziquantel is an active enantiomer of praziquantel.
    Formula:C19H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.41

    Ref: TM-T20127

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Butopamine

    CAS:
    Butopamine differs from dobutamine in location of only one hydroxyl group, but is no longer a catecholamine.
    Formula:C18H23NO3
    Color and Shape:Solid
    Molecular weight:301.38

    Ref: TM-T30630

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Pd 158771

    CAS:
    Pd 158771 is a D2 and 5-HT1A agonist.
    Formula:C22H31N5
    Color and Shape:Solid
    Molecular weight:365.52

    Ref: TM-T70081

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ML179

    CAS:
    ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.
    Formula:C21H25F3N4O2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:422.44

    Ref: TM-T8954

    1mg
    34.00€
    5mg
    75.00€
    10mg
    110.00€
    25mg
    220.00€
    50mg
    321.00€
    100mg
    469.00€
    200mg
    645.00€
    1mL*10mM (DMSO)
    92.00€
  • SC 53116 Hydrochloride

    CAS:
    SC 53116 Hydrochloride is selective agonist of the newly identified serotonin 5-HT4 receptor subtype.
    Formula:C16H23Cl2N3O2
    Color and Shape:Solid
    Molecular weight:360.28

    Ref: TM-T28696

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • 4-Chloro Trazodone hydrochloride

    CAS:
    4-Chloro Trazodone HCl is a Trazodone isomer, an antidepressant for anxiety disorders.
    Formula:C19H23Cl2N5O
    Color and Shape:Solid
    Molecular weight:408.32

    Ref: TM-T72119

    1mg
    96.00€
    5mg
    261.00€
    10mg
    480.00€
  • CCG-273220

    CAS:
    CCG-273220 covalently inhibits GRK5 at Cys474 with 220 nM IC50; more selective over GRK2.
    Formula:C26H24ClFN4O3
    Color and Shape:Solid
    Molecular weight:494.95

    Ref: TM-T63340

    25mg
    858.00€
    50mg
    1,116.00€
    100mg
    1,693.00€
  • Mocravimod

    CAS:
    Mocravimod: S1P1 receptor agonist, reduces atherosclerosis in mice. KRP-203 mitigates rat heart disease, extends graft survival.
    Formula:C24H26ClNO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:443.99

    Ref: TM-T28080

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (S)-V-0219


    (S)-V-0219: oral, GLP-1R PAM, boosts calcium in hGLP-1R HEK cells, lowers glucose, curbs hunger in mice.
    Formula:C20H25F3N4O2
    Color and Shape:Solid
    Molecular weight:410.43

    Ref: TM-T73081

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF 10040

    CAS:
    PF 10040 is an antagonist of platelet activating factor (PAF).
    Formula:C20H24ClNO2
    Color and Shape:Solid
    Molecular weight:345.86

    Ref: TM-T28359

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Noberastine maleate

    CAS:
    Noberastine maleate, a fast-acting furan-derived H1 antagonist, peaks at 4 hours with minimal CNS effects and maximal efficacy at 30 mg/day.
    Formula:C25H29N5O9
    Color and Shape:Solid
    Molecular weight:543.53

    Ref: TM-T71425

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cianergoline

    CAS:
    Cianergoline is a dopaminergic agonist.
    Formula:C19H22N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:322.4

    Ref: TM-T25247

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • AUY-954 free base

    CAS:
    AUY-954 is a selective S1P(1) modulator reducing EAN inflammation and demyelination in rats.
    Formula:C25H20F3NO2S
    Color and Shape:Solid
    Molecular weight:455.49

    Ref: TM-T30215

    1mg
    386.00€
    5mg
    1,198.00€
    500µg
    221.00€
  • Q8 hydrochloride

    CAS:
    Q8 is an antagonist of cysteinyl leukotreine receptor. Q8 inhibits VEGF-independent angiogenesis.
    Formula:C17H14ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.75

    Ref: TM-T28481

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tiamenidine hydrochloride

    CAS:
    Tiamenidine hydrochloride is a centrally-acting alpha1 adrenergic receptor antagonist.
    Formula:C8H11Cl2N3S
    Color and Shape:Solid
    Molecular weight:252.16

    Ref: TM-T69169

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€