
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Cirazoline (free base)
CAS:Cirazoline: full α1A agonist, partial α1B/D, nonselective α2 antagonist; potential vasoconstrictor.Formula:C13H16N2OColor and Shape:SolidMolecular weight:216.28SLM6031434 HCl
CAS:SLM6031434 HCl (SLM-6031434 HCl) is a SphK2 inhibitor that reduces LPS-induced TNF伪 and IL-1尾 production.Formula:C22H31ClF3N5O2Purity:98%Color and Shape:SolidMolecular weight:489.96ST-836
CAS:ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .Formula:C23H34N4OSPurity:98%Color and Shape:SolidMolecular weight:414.61SNAP-5089
CAS:SNAP-5089 is a highly selective alpha1A-adrenoceptor antagonist.Formula:C36H41ClN4O5Color and Shape:SolidMolecular weight:645.2Mivazerol
CAS:Mivazerol is an alpha 2-adrenoceptor agonist.Formula:C11H11N3O2Color and Shape:SolidMolecular weight:217.22(R)-Praziquantel
CAS:(R)-Praziquantel is an active enantiomer of praziquantel.Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:312.41Butopamine
CAS:Butopamine differs from dobutamine in location of only one hydroxyl group, but is no longer a catecholamine.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.38Pd 158771
CAS:Pd 158771 is a D2 and 5-HT1A agonist.Formula:C22H31N5Color and Shape:SolidMolecular weight:365.52ML179
CAS:ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.Formula:C21H25F3N4O2Purity:99.77%Color and Shape:SolidMolecular weight:422.44Ref: TM-T8954
1mg34.00€5mg75.00€10mg110.00€25mg220.00€50mg321.00€100mg469.00€200mg645.00€1mL*10mM (DMSO)92.00€SC 53116 Hydrochloride
CAS:SC 53116 Hydrochloride is selective agonist of the newly identified serotonin 5-HT4 receptor subtype.Formula:C16H23Cl2N3O2Color and Shape:SolidMolecular weight:360.284-Chloro Trazodone hydrochloride
CAS:4-Chloro Trazodone HCl is a Trazodone isomer, an antidepressant for anxiety disorders.Formula:C19H23Cl2N5OColor and Shape:SolidMolecular weight:408.32CCG-273220
CAS:CCG-273220 covalently inhibits GRK5 at Cys474 with 220 nM IC50; more selective over GRK2.Formula:C26H24ClFN4O3Color and Shape:SolidMolecular weight:494.95Mocravimod
CAS:Mocravimod: S1P1 receptor agonist, reduces atherosclerosis in mice. KRP-203 mitigates rat heart disease, extends graft survival.Formula:C24H26ClNO3SPurity:98%Color and Shape:SolidMolecular weight:443.99(S)-V-0219
(S)-V-0219: oral, GLP-1R PAM, boosts calcium in hGLP-1R HEK cells, lowers glucose, curbs hunger in mice.Formula:C20H25F3N4O2Color and Shape:SolidMolecular weight:410.43PF 10040
CAS:PF 10040 is an antagonist of platelet activating factor (PAF).Formula:C20H24ClNO2Color and Shape:SolidMolecular weight:345.86Noberastine maleate
CAS:Noberastine maleate, a fast-acting furan-derived H1 antagonist, peaks at 4 hours with minimal CNS effects and maximal efficacy at 30 mg/day.Formula:C25H29N5O9Color and Shape:SolidMolecular weight:543.53Cianergoline
CAS:Cianergoline is a dopaminergic agonist.Formula:C19H22N4OPurity:98%Color and Shape:SolidMolecular weight:322.4AUY-954 free base
CAS:AUY-954 is a selective S1P(1) modulator reducing EAN inflammation and demyelination in rats.Formula:C25H20F3NO2SColor and Shape:SolidMolecular weight:455.49Q8 hydrochloride
CAS:Q8 is an antagonist of cysteinyl leukotreine receptor. Q8 inhibits VEGF-independent angiogenesis.Formula:C17H14ClNO2Purity:98%Color and Shape:SolidMolecular weight:299.75Tiamenidine hydrochloride
CAS:Tiamenidine hydrochloride is a centrally-acting alpha1 adrenergic receptor antagonist.Formula:C8H11Cl2N3SColor and Shape:SolidMolecular weight:252.16
