
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:<p>Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].</p>Formula:C47H75N13O11Purity:98%Color and Shape:SolidMolecular weight:998.18Spns2-IN-1
<p>Spns2-IN-1 is a potent Spns2 inhibitor, effectively impeding Spns2-dependent S1P transport with an IC50 value of 1.4±0.3 μM, crucial for modulating the immune</p>Purity:98%Color and Shape:Odour Solid[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS:<p>[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).</p>Formula:C48H69N13O11S2Purity:98%Color and Shape:SolidMolecular weight:1068.27Prolactin Releasing Peptide (1-31), human
CAS:<p>Human Prolactin Releasing Peptide (1-31) is a potent GPR10 agonist; Ki values are 1.03 nM (human) and 0.33 nM (rat).</p>Formula:C160H252N56O42SPurity:98%Color and Shape:SolidMolecular weight:3664.15(D-Arg8)-Inotocin
CAS:<p>'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM.</p>Formula:C39H68N14O11S2Purity:98%Color and Shape:SolidMolecular weight:973.17Tafluprost acid
CAS:<p>Tafluprost acid is a selective agonist at the prostaglandin F receptor.</p>Formula:C22H28F2O5Color and Shape:SolidMolecular weight:410.46Heterobivalent ligand-1
<p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>Formula:C86H115FN16O21Color and Shape:SolidMolecular weight:1727.93S1R agonist 2
CAS:<p>S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for S2R and 1.1 nM for S1R and is protective against ROS and NMDA-induced neurotoxicity.</p>Formula:C21H27NOPurity:98.85%Color and Shape:SolidMolecular weight:309.45Adrenomedullin (16-31), human
CAS:<p>Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).</p>Formula:C82H129N25O21S2Purity:98%Color and Shape:SolidMolecular weight:1865.19Chir 2279
CAS:<p>CHIR 2279, a peptoid trimer, binds alpha 1-adrenoceptors, blocking epinephrine effects in dogs (pseudo pA2 6.86).</p>Formula:C34H36N4O4Color and Shape:SolidMolecular weight:564.67Eloralintide
CAS:<p>Eloralintide (LY 3841136) is an AMYR agonist, anticipated for research in type 2 diabetes and obesity.</p>Formula:C201H319N49O65S2Color and Shape:SolidMolecular weight:4526.1BAY-6672 hydrochloride
CAS:BAY-6672 hydrochloride is a potent, selective antagonist of the human Prostaglandin F (FP) receptor, exhibiting an IC50 value of 11 nM.Formula:C26H28BrCl2N3O3Color and Shape:SolidMolecular weight:581.3317-TFM-PGF1α
CAS:<p>17-TFM-PGF1α (Compound 8) is a saturated prostaglandin analog. It exhibits a high affinity and receptor selectivity for the human prostaglandin F receptor (hFP receptor), with an EC50 of 85 nM.</p>Formula:C24H35F3O5Color and Shape:SolidMolecular weight:460.538β-Hydroxy-exo-THC
CAS:<p>8β-Hydroxy-exo-THC, a cannabinoid ether analog, exhibits weak affinity for receptor sites with an IC50 of 1.2 μM.</p>Formula:C21H30O3Color and Shape:SolidMolecular weight:330.462,6-DMA hydrochloride
CAS:<p>2,6-DMA hydrochloride is a phenethylamine and acts as an agonist of the serotonin 5-HT2 receptor, with a pA2 value of 5.09.</p>Formula:C11H18ClNO2Color and Shape:SolidMolecular weight:231.72Methylhexanamine hydrochloride
CAS:<p>Methylhexanamine hydrochloride is a fatty amine and vasoconstrictor that functions as a nasal decongestant when inhaled through the nasal mucosa.</p>Formula:C7H18ClNColor and Shape:SolidMolecular weight:151.688-Chloro caffeine
CAS:<p>8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.</p>Formula:C8H9ClN4O2Color and Shape:SolidMolecular weight:228.64UKH-1114
CAS:<p>UKH-1114 is a potent σ2 receptor/Tmem97 agonist with a Ki value of 46 nM, demonstrating antinociceptive effects against mechanical hypersensitivity. This compound alleviates mechanical hypersensitivity in mice caused by nerve injury without inducing motor impairment and is a promising candidate for neuropathic pain research.</p>Formula:C22H24F3NOColor and Shape:SolidMolecular weight:375.43sGC activator 2
<p>sGC activator 2 (Compound 16a) acts as an activator of soluble guanylate cyclase (sGC), enhancing the production of cGMP and exhibiting vasoprotective and anti-inflammatory properties.</p>Formula:C21H21FN8O3Color and Shape:SolidMolecular weight:452.44QWF acetate
<p>QWF acetate is a Substance P antagonist peptide that specifically inhibits the binding to its receptor, NK1, and inhibits the activation of MRGPRX2.</p>Formula:C40H47N5O10Purity:96.65%Color and Shape:SolidMolecular weight:757.84

