
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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MRS2179
CAS:MRS2179: P2Y1 antagonist, Kb=100 nM, inactive on P2Y2/4/6 (to 30µM), inhibits ADP-induced platelet changes, prolongs bleeding in rodents.Formula:C11H17N5O9P2Color and Shape:SolidMolecular weight:425.23GAT228
CAS:GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].Formula:C22H18N2O2Color and Shape:SolidMolecular weight:342.39PD 81723
CAS:Allosteric potentiator at the adenosine A1 receptorFormula:C14H12F3NOSPurity:98%Color and Shape:SolidMolecular weight:299.31SKF 77434 hydrobromide
CAS:SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.Formula:C19H22BrNO2Purity:98%Color and Shape:SolidMolecular weight:376.29Usmarapride
CAS:Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.Formula:C23H31N5O6Color and Shape:SolidMolecular weight:473.53BMS-193884
CAS:BMS-193884 is an oral endothelin antagonist for the treatment of congestive heart failure (CHF) and pulmonary arterial hypertension.Formula:C20H17N3O4SColor and Shape:SolidMolecular weight:395.43MK761
CAS:MK761 combines β-blocker and vasodilator effects, matching timolol and indololol in efficacy; active in cat heart and rat atria studies.Formula:C13H19N3O2Color and Shape:SolidMolecular weight:249.31NPC 17731
CAS:NPC 17731 is a bradykinin receptor antagonist.Formula:C59H95N19O14Color and Shape:SolidMolecular weight:1294.5AK-IN-1
CAS:AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.Formula:C22H21N3O4Color and Shape:SolidMolecular weight:391.42PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Formula:C17H21N3Purity:98%Color and Shape:SolidMolecular weight:267.37Bromerguride
CAS:Bromerguride is a dopamine antagonist with the activity of antipsychotic.Formula:C20H25BrN4OColor and Shape:SolidMolecular weight:417.34Piroheptine HCl
CAS:Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.Formula:C22H26ClNPurity:98%Color and Shape:SolidMolecular weight:339.9GSK334429
CAS:GSK334429 is an antagonist of histamine H3 receptor.Formula:C20H29F3N4OColor and Shape:SolidMolecular weight:398.47GB-110
CAS:GB-110, a potent PAR2 agonist, triggers Ca2+ release in HT29 cells with a 0.28 μM EC50, is orally active and nonpeptidic.Formula:C33H48N6O5Purity:98%Color and Shape:SolidMolecular weight:608.77Adenosine receptor antagonist 2
CAS:Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.Formula:C23H21FN8OColor and Shape:SolidMolecular weight:444.46JNJ-17156516
CAS:JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.Formula:C26H22Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:481.37Bag-1
CAS:Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.Formula:C22H27N3Color and Shape:SolidMolecular weight:333.47ABT-546
CAS:ABT-546 is a potent, selective endothelin ETA receptor antagonist, Ki 0.46 nM for [125I]ET-1 binding.Formula:C30H48N2O6Purity:98%Color and Shape:SolidMolecular weight:532.71MRS2395
CAS:MRS2395, a dipivaloyl P2Y12 receptor blocker, inhibits ADP-induced platelet activation with a Ki of 3.6 μM and boosts TRAP-6-triggered dense granule release.Formula:C20H30ClN5O4Color and Shape:SolidMolecular weight:439.94(RS)-Butyryltimolol
CAS:(RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.Formula:C17H30N4O4SPurity:98%Color and Shape:SolidMolecular weight:386.51
