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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • MRS2179

    CAS:
    MRS2179: P2Y1 antagonist, Kb=100 nM, inactive on P2Y2/4/6 (to 30µM), inhibits ADP-induced platelet changes, prolongs bleeding in rodents.
    Formula:C11H17N5O9P2
    Color and Shape:Solid
    Molecular weight:425.23

    Ref: TM-T28099

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GAT228

    CAS:
    GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].
    Formula:C22H18N2O2
    Color and Shape:Solid
    Molecular weight:342.39

    Ref: TM-T61105

    1mg
    118.00€
    10mg
    673.00€
  • PD 81723

    CAS:
    Allosteric potentiator at the adenosine A1 receptor
    Formula:C14H12F3NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.31

    Ref: TM-T23130

    10mg
    623.00€
    50mg
    2,565.00€
  • SKF 77434 hydrobromide

    CAS:
    SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.
    Formula:C19H22BrNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:376.29

    Ref: TM-T23360

    5mg
    233.00€
  • Usmarapride

    CAS:
    Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.
    Formula:C23H31N5O6
    Color and Shape:Solid
    Molecular weight:473.53

    Ref: TM-T63069

    25mg
    1,080.00€
    50mg
    1,414.00€
    100mg
    2,277.00€
  • BMS-193884

    CAS:
    BMS-193884 is an oral endothelin antagonist for the treatment of congestive heart failure (CHF) and pulmonary arterial hypertension.
    Formula:C20H17N3O4S
    Color and Shape:Solid
    Molecular weight:395.43

    Ref: TM-T30501

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • MK761

    CAS:
    MK761 combines β-blocker and vasodilator effects, matching timolol and indololol in efficacy; active in cat heart and rat atria studies.
    Formula:C13H19N3O2
    Color and Shape:Solid
    Molecular weight:249.31

    Ref: TM-T33437

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NPC 17731

    CAS:
    NPC 17731 is a bradykinin receptor antagonist.
    Formula:C59H95N19O14
    Color and Shape:Solid
    Molecular weight:1294.5

    Ref: TM-T70576

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AK-IN-1

    CAS:
    AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.
    Formula:C22H21N3O4
    Color and Shape:Solid
    Molecular weight:391.42

    Ref: TM-T73436

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • PF-04781340

    CAS:
    PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.
    Formula:C17H21N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.37

    Ref: TM-T24616

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bromerguride

    CAS:
    Bromerguride is a dopamine antagonist with the activity of antipsychotic.
    Formula:C20H25BrN4O
    Color and Shape:Solid
    Molecular weight:417.34

    Ref: TM-T26909

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Piroheptine HCl

    CAS:
    Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.
    Formula:C22H26ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:339.9

    Ref: TM-T24645

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • GSK334429

    CAS:
    GSK334429 is an antagonist of histamine H3 receptor.
    Formula:C20H29F3N4O
    Color and Shape:Solid
    Molecular weight:398.47

    Ref: TM-T27473

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GB-110

    CAS:
    GB-110, a potent PAR2 agonist, triggers Ca2+ release in HT29 cells with a 0.28 μM EC50, is orally active and nonpeptidic.
    Formula:C33H48N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:608.77

    Ref: TM-T11369

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Adenosine receptor antagonist 2

    CAS:
    Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.
    Formula:C23H21FN8O
    Color and Shape:Solid
    Molecular weight:444.46

    Ref: TM-T62611

    25mg
    1,791.00€
    50mg
    3,025.00€
  • JNJ-17156516

    CAS:
    JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.
    Formula:C26H22Cl2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.37

    Ref: TM-T27664

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bag-1

    CAS:
    Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.
    Formula:C22H27N3
    Color and Shape:Solid
    Molecular weight:333.47

    Ref: TM-T71595

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • ABT-546

    CAS:
    ABT-546 is a potent, selective endothelin ETA receptor antagonist, Ki 0.46 nM for [125I]ET-1 binding.
    Formula:C30H48N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:532.71

    Ref: TM-T10225

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS2395

    CAS:
    MRS2395, a dipivaloyl P2Y12 receptor blocker, inhibits ADP-induced platelet activation with a Ki of 3.6 μM and boosts TRAP-6-triggered dense granule release.
    Formula:C20H30ClN5O4
    Color and Shape:Solid
    Molecular weight:439.94

    Ref: TM-T62532

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (RS)-Butyryltimolol

    CAS:
    (RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.
    Formula:C17H30N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.51

    Ref: TM-T13439

    2mg
    63.00€