GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,002 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(192 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5966 products of "GPCR/G-Protein"
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ST 91
CAS:ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.Formula:C13H20ClN3Purity:99.83%Color and Shape:SolidMolecular weight:253.77Ref: TM-T23397
5mg49.00€10mg72.00€25mg142.00€50mg245.00€100mg354.00€200mg497.00€1mL*10mM (DMSO)50.00€Antihistamine-1
CAS:Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。Formula:C23H24FN5Purity:99.69%Color and Shape:SolidMolecular weight:389.47KI-7
CAS:KI-7 is an adenosine A2B receptor positive allosteric modulator.Formula:C23H18N2O2Purity:98.33%Color and Shape:SolidMolecular weight:354.4Ref: TM-T9238
2mg35.00€5mg55.00€10mg95.00€25mg172.00€50mg264.00€100mg399.00€200mg560.00€1mL*10mM (DMSO)62.00€Ecastolol
CAS:Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formula:C26H33N3O6Purity:99.89%Color and Shape:SolidMolecular weight:483.56Ref: TM-T11148
1mg349.00€5mg697.00€10mg888.00€25mg1,395.00€50mg1,783.00€100mg2,530.00€1mL*10mM (DMSO)880.00€Runcaciguat
CAS:Runcaciguat, a soluble guanylate cyclase stimulator, aids in cardiovascular and renal research.Formula:C23H22Cl2F3NO3Purity:99.17%Color and Shape:SolidMolecular weight:488.33PSB-16133 sodium
CAS:PSB-16133 sodium is a selective P2Y purine receptor variant antagonist with an IC of 233 nM.Formula:C28H21N2NaO5S2Purity:98.03% - 98.93%Color and Shape:SolidMolecular weight:552.60Vadocaine
CAS:Vadocaine (Vadocaina) is a novel analgesic compound for local anaesthesia and can be used to study the central nervous system and cardiovascular system.Formula:C18H28N2O2Purity:99.7%Color and Shape:SolidMolecular weight:304.43Ordopidine
CAS:Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.Formula:C14H20FNO2SPurity:97.09%Color and Shape:SolidMolecular weight:285.38Pirmagrel
CAS:pirmagrel is a potent thromboxane synthase inhibitor.Formula:C13H16N2O2Purity:98.02%Color and Shape:SolidMolecular weight:232.285-HT1A modulator 1
CAS:5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).Formula:C21H25N3O2SPurity:99.68%Color and Shape:SolidMolecular weight:383.51N 0861
CAS:N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.Formula:C13H17N5Purity:98.78%Color and Shape:SolidMolecular weight:243.31Ref: TM-T70722
1mg164.00€2mg234.00€5mg389.00€10mg532.00€25mg820.00€50mg1,063.00€100mg1,423.00€200mg1,945.00€Oxyfedrine L-form HCl
CAS:Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.Formula:C19H24ClNO3Purity:99.5% - 99.57%Color and Shape:SolidMolecular weight:349.85Ref: TM-T24579
1mg92.00€5mg178.00€10mg313.00€25mg485.00€50mg700.00€100mg893.00€200mg1,198.00€1mL*10mM (DMSO)203.00€Eclazolast
CAS:Eclazolast (RHC 2871), a lipophilic anti-allergic, inhibits mast cell mediator release by affecting Fc(epsilon)RI-related processes, dose-dependently.Formula:C12H12ClNO4Purity:98.29% - 98.61%Color and Shape:SolidMolecular weight:269.68Ref: TM-T25360
1mg112.00€5mg261.00€10mg396.00€25mg655.00€50mg888.00€100mg1,251.00€500mg2,493.00€1mL*10mM (DMSO)249.00€GW438014A
CAS:GW438014A 是一种有效且具有选择性的 NPY-Y5 受体拮抗剂。GW438014A 对食物摄入并减少肥胖啮齿动物的体重增加具有抑制作用。Formula:C23H23N3O4SPurity:99.94%Color and Shape:SolidMolecular weight:437.51CGRP antagonist 1
CAS:CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for theFormula:C29H26N4O4Purity:99.55%Color and Shape:SolidMolecular weight:494.54Viloxazine
CAS:Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activityFormula:C13H19NO3Purity:99.65%Color and Shape:SolidMolecular weight:237.29Torbafylline
CAS:Torbafylline is a xanthine-based PDE inhibitor reducing protein breakdown via PDE4/cAMP/EPAC/PI3K/Akt in rats with burns, cancer, or sepsis.Formula:C16H26N4O4Purity:99.96% - 99.97%Color and Shape:SoildMolecular weight:338.4Ref: TM-T67965
1mg81.00€5mg172.00€10mg259.00€25mg424.00€50mg583.00€100mg800.00€1mL*10mM (DMSO)178.00€O-1602
CAS:O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatmentFormula:C17H22O2Purity:99.85%Color and Shape:SolidMolecular weight:258.36Ref: TM-T23097
1mg44.00€5mg95.00€10mg137.00€25mg254.00€50mg358.00€100mg537.00€200mg762.00€1mL*10mM (DMSO)95.00€ADR-851 free base
CAS:ADR-851 free base is an antagonist of the HT3 receptor.Formula:C14H18ClN3O2Purity:97.88% - 98.39%Color and Shape:SolidMolecular weight:295.77TASP0390325
CAS:TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in rodents.Formula:C25H30Cl2FN5O4Purity:98.62%Color and Shape:SolidMolecular weight:554.44
