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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5745 products of "GPCR/G-Protein"

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  • SLF1081851
    Targetmol
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    SLF1081851

    CAS:
    <p>SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.</p>
    Formula:C21H33N3O
    Purity:99.26%
    Color and Shape:Solid
    Molecular weight:343.51

    Ref: TM-T61112

  • R 59-022 hydrochloride
    Targetmol
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    R 59-022 hydrochloride

    CAS:
    <p>R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.</p>
    Formula:C27H27ClFN3OS
    Purity:97.7%
    Color and Shape:Solid
    Molecular weight:496.04

    Ref: TM-T72322

  • Remoxipride hydrochloride
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    Remoxipride hydrochloride

    CAS:
    Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-
    Formula:C16H24BrClN2O3
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:407.73

    Ref: TM-T23232

  • Lorglumide sodium salt
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    Lorglumide sodium salt

    CAS:
    Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).
    Formula:C22H31Cl2N2NaO4
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:481.39

    Ref: TM-T11868

  • SB-277011
    Targetmol
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    SB-277011

    CAS:
    <p>SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), &lt;5.2 (5-HT1B).</p>
    Formula:C28H30N4O
    Purity:99.39%
    Color and Shape:Solid
    Molecular weight:438.56

    Ref: TM-T12861

  • Liafensine
    Targetmol
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    Liafensine

    CAS:
    Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.
    Formula:C24H22N4
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:366.46

    Ref: TM-T32737

  • rel-(1R,2R)-Vesamicol Hydrochloride
    Targetmol
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    rel-(1R,2R)-Vesamicol Hydrochloride

    CAS:
    rel-(1R,2R)-Vesamicol Hydrochloride is a acetylcholine transport inhibitor.
    Formula:C17H26ClNO
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:295.85

    Ref: TM-T22486

  • Enerisant hydrochloride
    Targetmol
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    Enerisant hydrochloride

    CAS:
    <p>Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins</p>
    Formula:C22H31ClN4O3
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:434.96

    Ref: TM-T70489

  • Dabelotine
    Targetmol
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    Dabelotine

    CAS:
    <p>Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.</p>
    Formula:C15H22N2O2
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:262.35

    Ref: TM-T31175

  • CCG 203769
    Targetmol
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    CCG 203769

    CAS:
    CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.
    Formula:C8H14N2O2S
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:202.27

    Ref: TM-T10705

  • Tiospirone
    Targetmol
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    Tiospirone

    CAS:
    Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and a dopamine blocker used in the study of neurological disorders such as schizophrenia.
    Formula:C24H32N4O2S
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:440.6

    Ref: TM-T24885

  • Sitaxsentan
    Targetmol
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    Sitaxsentan

    CAS:
    Sitaxsentan (TBC-11251), a selective ETA receptor antagonist, prevents vasoconstriction by blocking endothelin.
    Formula:C18H15ClN2O6S2
    Purity:97.99% - 98.71%
    Color and Shape:Solid
    Molecular weight:454.9

    Ref: TM-T12924

  • Efletirizine
    Targetmol
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    Efletirizine

    CAS:
    <p>Efletirizine (UCB-28754), a histamine blocker and 5-LO inhibitor, aids in topical allergy treatment.</p>
    Formula:C21H24F2N2O3
    Purity:99.39%
    Color and Shape:Solid
    Molecular weight:390.42

    Ref: TM-T27244

  • ABT-080
    Targetmol
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    ABT-080

    CAS:
    <p>ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma.</p>
    Formula:C37H31N2NaO4
    Purity:98.42%
    Color and Shape:Solid
    Molecular weight:590.64

    Ref: TM-T26524

  • Milveterol HCl
    Targetmol
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    Milveterol HCl

    CAS:
    Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).
    Formula:C25H30ClN3O4
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:471.98

    Ref: TM-T33386

  • Antihistamine-1
    Targetmol
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    Antihistamine-1

    CAS:
    Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。
    Formula:C23H24FN5
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:389.47

    Ref: TM-T10335

  • Sergliflozin etabonate
    Targetmol
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    Sergliflozin etabonate

    CAS:
    Sergliflozin etabonate (KGT-1251) is an inhibitor of SGLT2 and can be used in studies about type 2 diabetes and obesity.
    Formula:C23H28O9
    Purity:97.88%
    Color and Shape:Solid
    Molecular weight:448.46

    Ref: TM-T28757

  • K6PC-5
    Targetmol
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    K6PC-5

    CAS:
    <p>K6PC-5 is a ceramide derivative that acts as an activator of sphingosine kinase 1 (SPHK1), inducing a swift and temporary rise in intracellular calcium levels.</p>
    Formula:C19H37NO4
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:343.5

    Ref: TM-T27710

  • Felcisetrag
    Targetmol
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    Felcisetrag

    CAS:
    <p>Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.</p>
    Formula:C25H37N5O3
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:455.59

    Ref: TM-T28934

  • Evodenoson
    Targetmol
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    Evodenoson

    CAS:
    Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.
    Formula:C23H29N7O6
    Purity:99.75% - 99.83%
    Color and Shape:Solid
    Molecular weight:499.52

    Ref: TM-T31731