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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5745 products of "GPCR/G-Protein"

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  • L 674573

    CAS:
    L 674573 is an inhibitor of leukotriene biosynthesis.
    Formula:C28H27NO3S
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:457.58
  • Ticolubant

    CAS:
    Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.
    Formula:C23H19Cl2NO3S
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:460.37
  • Roxindole

    CAS:
    Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.
    Formula:C23H26N2O
    Purity:98.03% - 98.93%
    Color and Shape:Solid
    Molecular weight:346.47
  • SK609 HCl

    CAS:
    <p>SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.</p>
    Formula:C10H15Cl2N
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:220.14
  • ABT-080

    CAS:
    <p>ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma.</p>
    Formula:C37H31N2NaO4
    Purity:98.42%
    Color and Shape:Solid
    Molecular weight:590.64
  • AS-35

    CAS:
    AS-35, an oral selective leukotriene antagonist, counters ileum contractions with IC50: 8 nM (LTC4), 4 nM (LTD4), 3 nM (LTE4); shows antiallergic effects.
    Formula:C21H20N6O4
    Purity:96.69%
    Color and Shape:Solid
    Molecular weight:420.42
  • Runcaciguat

    CAS:
    Runcaciguat, a soluble guanylate cyclase stimulator, aids in cardiovascular and renal research.
    Formula:C23H22Cl2F3NO3
    Purity:99.17%
    Color and Shape:Solid
    Molecular weight:488.33
  • Vadocaine

    CAS:
    Vadocaine (Vadocaina) is a novel analgesic compound for local anaesthesia and can be used to study the central nervous system and cardiovascular system.
    Formula:C18H28N2O2
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:304.43
  • Rezatomidine

    CAS:
    <p>Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.</p>
    Formula:C13H16N2S
    Purity:98.34%
    Color and Shape:Solid
    Molecular weight:232.34
  • (S)-(+)-Niguldipine hydrochloride

    CAS:
    (S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.
    Formula:C36H40ClN3O6
    Purity:98.27%
    Color and Shape:Solid
    Molecular weight:646.17
  • DA-6886

    CAS:
    DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.
    Formula:C19H28Cl2N6O2
    Purity:99.91% - 99.99%
    Color and Shape:Solid
    Molecular weight:443.37
  • Masupirdine free base

    CAS:
    Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.
    Formula:C21H24BrN3O3S
    Purity:98.36% - 99.65%
    Color and Shape:Solid
    Molecular weight:478.4
  • CP 316311

    CAS:
    CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression.
    Formula:C21H29NO2
    Purity:99.71% - >99.99%
    Color and Shape:Solid
    Molecular weight:327.46
  • Pavinetant

    CAS:
    Pavinetant (MLE-4901) is an orally available neurokinin-3 receptor (NK3R) antagonist used to improve menopausal symptoms.
    Formula:C26H25N3O3S
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:459.56
  • Benperidol

    CAS:
    Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.
    Formula:C22H24FN3O2
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:381.44
  • Butofilolol

    CAS:
    <p>Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.</p>
    Formula:C17H26FNO3
    Purity:98.96% - >99.99%
    Color and Shape:Solid
    Molecular weight:311.392
  • JP1302

    CAS:
    JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.
    Formula:C24H24N4
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:368.47
  • S1p receptor agonist 2

    CAS:
    <p>S1P5-selective agonist; less so for S1P1/S1P3; useful for CNS disorders.</p>
    Formula:C24H23ClN2O4
    Color and Shape:Solid
    Molecular weight:438.9
  • Bufuralol (hydrochloride)

    CAS:
    Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.
    Formula:C16H24ClNO2
    Color and Shape:Solid
    Molecular weight:297.82
  • Cipralisant maleate

    CAS:
    Cipralisant maleate is a potent, selective Histamine H3 receptor antagonist.
    Formula:C18H24N2O4
    Color and Shape:Solid
    Molecular weight:332.39