
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(993 products)
- Adenosine Receptor(246 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(212 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(182 products)
- Hedgehog/Smoothened(47 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(310 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5745 products of "GPCR/G-Protein"
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L 674573
CAS:L 674573 is an inhibitor of leukotriene biosynthesis.Formula:C28H27NO3SPurity:99.51%Color and Shape:SolidMolecular weight:457.58Ticolubant
CAS:Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.Formula:C23H19Cl2NO3SPurity:99.5%Color and Shape:SolidMolecular weight:460.37Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formula:C23H26N2OPurity:98.03% - 98.93%Color and Shape:SolidMolecular weight:346.47SK609 HCl
CAS:<p>SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.</p>Formula:C10H15Cl2NPurity:99.02%Color and Shape:SolidMolecular weight:220.14ABT-080
CAS:<p>ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma.</p>Formula:C37H31N2NaO4Purity:98.42%Color and Shape:SolidMolecular weight:590.64AS-35
CAS:AS-35, an oral selective leukotriene antagonist, counters ileum contractions with IC50: 8 nM (LTC4), 4 nM (LTD4), 3 nM (LTE4); shows antiallergic effects.Formula:C21H20N6O4Purity:96.69%Color and Shape:SolidMolecular weight:420.42Runcaciguat
CAS:Runcaciguat, a soluble guanylate cyclase stimulator, aids in cardiovascular and renal research.Formula:C23H22Cl2F3NO3Purity:99.17%Color and Shape:SolidMolecular weight:488.33Vadocaine
CAS:Vadocaine (Vadocaina) is a novel analgesic compound for local anaesthesia and can be used to study the central nervous system and cardiovascular system.Formula:C18H28N2O2Purity:99.7%Color and Shape:SolidMolecular weight:304.43Rezatomidine
CAS:<p>Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.</p>Formula:C13H16N2SPurity:98.34%Color and Shape:SolidMolecular weight:232.34(S)-(+)-Niguldipine hydrochloride
CAS:(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.Formula:C36H40ClN3O6Purity:98.27%Color and Shape:SolidMolecular weight:646.17DA-6886
CAS:DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Formula:C19H28Cl2N6O2Purity:99.91% - 99.99%Color and Shape:SolidMolecular weight:443.37Masupirdine free base
CAS:Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formula:C21H24BrN3O3SPurity:98.36% - 99.65%Color and Shape:SolidMolecular weight:478.4CP 316311
CAS:CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression.Formula:C21H29NO2Purity:99.71% - >99.99%Color and Shape:SolidMolecular weight:327.46Pavinetant
CAS:Pavinetant (MLE-4901) is an orally available neurokinin-3 receptor (NK3R) antagonist used to improve menopausal symptoms.Formula:C26H25N3O3SPurity:99.8%Color and Shape:SolidMolecular weight:459.56Benperidol
CAS:Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.Formula:C22H24FN3O2Purity:99.91%Color and Shape:SolidMolecular weight:381.44Butofilolol
CAS:<p>Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.</p>Formula:C17H26FNO3Purity:98.96% - >99.99%Color and Shape:SolidMolecular weight:311.392JP1302
CAS:JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.Formula:C24H24N4Purity:99.96%Color and Shape:SolidMolecular weight:368.47S1p receptor agonist 2
CAS:<p>S1P5-selective agonist; less so for S1P1/S1P3; useful for CNS disorders.</p>Formula:C24H23ClN2O4Color and Shape:SolidMolecular weight:438.9Bufuralol (hydrochloride)
CAS:Bufuralol hydrochloride is a potent, non-selective, orally active β-blocker with partial agonist effects and a CYP2D6 probe.Formula:C16H24ClNO2Color and Shape:SolidMolecular weight:297.82Cipralisant maleate
CAS:Cipralisant maleate is a potent, selective Histamine H3 receptor antagonist.Formula:C18H24N2O4Color and Shape:SolidMolecular weight:332.39
