
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(993 products)
- Adenosine Receptor(246 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(212 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(182 products)
- Hedgehog/Smoothened(47 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(310 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5745 products of "GPCR/G-Protein"
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RP-23618
CAS:RP-23618 is a non-peptidic antagonist of RANTES.Formula:C30H35N5O3S2Purity:98%Color and Shape:SolidMolecular weight:577.76RO5527239
CAS:RO5527239 is a potent, orally available GPBAR1 agonist agent.Formula:C28H31N3O3Purity:98%Color and Shape:SolidMolecular weight:457.56Leukotriene B4-3-aminopropylamide
CAS:Leukotriene B4 (LTB4)-3-aminopropylamide is an analog of LTB4 that exhibits potent and selective binding to the BLT1 receptor with Ki values of 5.1 nM at BLT1 and 1,227 nM at BLT2, indicating its high affinity for BLT1 over BLT2. This compound's effects are mediated through interactions with two receptors, BLT1 and BLT2.Formula:C23H40N2O3Color and Shape:SolidMolecular weight:392.6YM44778
CAS:YM44778 is a NK1-receptor antagonist for treating restless legs syndrome.Formula:C34H39Cl2N3O5Color and Shape:SolidMolecular weight:640.6Tricosanoyl Ethanolamide
CAS:Tricosanoyl ethanolamide, a fatty N-acyl ethanolamine within the endocannabinoid family, has an ethanolamine metabolite whose significance remains to be established.Formula:C25H51NO2Color and Shape:SolidMolecular weight:397.688TASP0376377
CAS:TASP0376377 is a potent antagonist of CRTH2.Formula:C25H16Cl2N2O4Color and Shape:SolidMolecular weight:479.311-Carboxycyclohexaneacetic Acid
CAS:1-Carboxycyclohexaneacetic acid may be present as a potential impurity in commercial gabapentin, an antiepileptic drug. Furthermore, it serves as a precursor for synthesizing antagonists targeting the serotonin (5-HT) receptor subtype 5-HT2A.Formula:C9H14O4Color and Shape:SolidMolecular weight:186.207Binedaline
CAS:Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.Formula:C19H23N3Purity:98%Color and Shape:SolidMolecular weight:293.41Bufuralol
CAS:Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.Formula:C16H23NO2Purity:98.26%Color and Shape:SolidMolecular weight:261.36RBC10
CAS:RBC10 inhibits the binding of Ral to its effector RALBP1, as well as inhibiting Ral-mediated cell spreading of murine embryonic fibroblasts and anchorage-Formula:C24H25ClN2O2Purity:99.71%Color and Shape:SolidMolecular weight:408.92GPR3 agonist-2
CAS:GPR3 agonist-2 (compound 32) is a potent full agonist of the G protein-coupled receptor 3 (GPR3), exhibiting an IC50 value of 260 nM [1].Formula:C14H7F6IO4SColor and Shape:SolidMolecular weight:512.16Emicerfont
CAS:<p>Emicerfont is an antagonist of the corticotropin-releasing factor type 1 receptor (IC50: 66 nM).</p>Formula:C22H24N6O2Purity:98%Color and Shape:SolidMolecular weight:404.46PD 165929
CAS:PD 165929 is a selective antagonist of Bombesin BB1.Formula:C37H47N5O2Purity:98%Color and Shape:SolidMolecular weight:593.8Quinpirole dihydrochloride
CAS:<p>Quinpirole dihydrochloride is an agonist of the D2-like dopamine receptor.</p>Formula:C13H23Cl2N3Purity:98%Color and Shape:SolidMolecular weight:292.25EP2 receptor agonist 4
CAS:EP2 receptor agonist 4 selectively activates the EP2 receptor with an efficacy concentration (EC50) of 43 nM [1].Formula:C23H36O5Color and Shape:SolidMolecular weight:392.53NBI-35965
CAS:<p>NBI-35965 is a CRF1 receptor antagonist.</p>Formula:C21H22Cl2N4Color and Shape:SolidMolecular weight:401.33SGC agonist 1
CAS:SGC agonist 1 is a potent soluble guanylate cyclase (SGC) agonist. SGC agonist 1 is able to increase solubility and has high cell permeability.Formula:C22H19F2N7OColor and Shape:SolidMolecular weight:435.43Indeloxazine hydrochloride
CAS:Indeloxazine HCl: Serotonin releaser, NE reuptake inhibitor, NMDA antagonist; antidepressant that boosts acetylcholine in rats.Formula:C14H18ClNO2Purity:98%Color and Shape:SolidMolecular weight:267.75[D-Ala6]-LH-RH
CAS:[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32Prostaglandin E1 ethanolamide
CAS:Prostaglandin E1 ethanolamide, an analog of Prostaglandin E1 (PGE1), can potentially inhibit the GLI2-induced expression of target genes such as Gli1 and Ptch1, thereby reducing tumor growth [1].Formula:C22H39NO5Color and Shape:SolidMolecular weight:397.55

