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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5745 products of "GPCR/G-Protein"

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  • RP-23618

    CAS:
    RP-23618 is a non-peptidic antagonist of RANTES.
    Formula:C30H35N5O3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:577.76
  • RO5527239

    CAS:
    RO5527239 is a potent, orally available GPBAR1 agonist agent.
    Formula:C28H31N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.56
  • Leukotriene B4-3-aminopropylamide

    CAS:
    Leukotriene B4 (LTB4)-3-aminopropylamide is an analog of LTB4 that exhibits potent and selective binding to the BLT1 receptor with Ki values of 5.1 nM at BLT1 and 1,227 nM at BLT2, indicating its high affinity for BLT1 over BLT2. This compound's effects are mediated through interactions with two receptors, BLT1 and BLT2.
    Formula:C23H40N2O3
    Color and Shape:Solid
    Molecular weight:392.6
  • YM44778

    CAS:
    YM44778 is a NK1-receptor antagonist for treating restless legs syndrome.
    Formula:C34H39Cl2N3O5
    Color and Shape:Solid
    Molecular weight:640.6
  • Tricosanoyl Ethanolamide

    CAS:
    Tricosanoyl ethanolamide, a fatty N-acyl ethanolamine within the endocannabinoid family, has an ethanolamine metabolite whose significance remains to be established.
    Formula:C25H51NO2
    Color and Shape:Solid
    Molecular weight:397.688
  • TASP0376377

    CAS:
    TASP0376377 is a potent antagonist of CRTH2.
    Formula:C25H16Cl2N2O4
    Color and Shape:Solid
    Molecular weight:479.31
  • 1-Carboxycyclohexaneacetic Acid

    CAS:
    1-Carboxycyclohexaneacetic acid may be present as a potential impurity in commercial gabapentin, an antiepileptic drug. Furthermore, it serves as a precursor for synthesizing antagonists targeting the serotonin (5-HT) receptor subtype 5-HT2A.
    Formula:C9H14O4
    Color and Shape:Solid
    Molecular weight:186.207
  • Binedaline

    CAS:
    Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.
    Formula:C19H23N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:293.41
  • Bufuralol

    CAS:
    Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects and can be used to study cardiovascular diseases.
    Formula:C16H23NO2
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:261.36
  • RBC10

    CAS:
    RBC10 inhibits the binding of Ral to its effector RALBP1, as well as inhibiting Ral-mediated cell spreading of murine embryonic fibroblasts and anchorage-
    Formula:C24H25ClN2O2
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:408.92
  • GPR3 agonist-2

    CAS:
    GPR3 agonist-2 (compound 32) is a potent full agonist of the G protein-coupled receptor 3 (GPR3), exhibiting an IC50 value of 260 nM [1].
    Formula:C14H7F6IO4S
    Color and Shape:Solid
    Molecular weight:512.16
  • Emicerfont

    CAS:
    <p>Emicerfont is an antagonist of the corticotropin-releasing factor type 1 receptor (IC50: 66 nM).</p>
    Formula:C22H24N6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:404.46
  • PD 165929

    CAS:
    PD 165929 is a selective antagonist of Bombesin BB1.
    Formula:C37H47N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:593.8
  • Quinpirole dihydrochloride

    CAS:
    <p>Quinpirole dihydrochloride is an agonist of the D2-like dopamine receptor.</p>
    Formula:C13H23Cl2N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:292.25
  • EP2 receptor agonist 4

    CAS:
    EP2 receptor agonist 4 selectively activates the EP2 receptor with an efficacy concentration (EC50) of 43 nM [1].
    Formula:C23H36O5
    Color and Shape:Solid
    Molecular weight:392.53
  • NBI-35965

    CAS:
    <p>NBI-35965 is a CRF1 receptor antagonist.</p>
    Formula:C21H22Cl2N4
    Color and Shape:Solid
    Molecular weight:401.33
  • SGC agonist 1

    CAS:
    SGC agonist 1 is a potent soluble guanylate cyclase (SGC) agonist. SGC agonist 1 is able to increase solubility and has high cell permeability.
    Formula:C22H19F2N7O
    Color and Shape:Solid
    Molecular weight:435.43
  • Indeloxazine hydrochloride

    CAS:
    Indeloxazine HCl: Serotonin releaser, NE reuptake inhibitor, NMDA antagonist; antidepressant that boosts acetylcholine in rats.
    Formula:C14H18ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.75
  • [D-Ala6]-LH-RH

    CAS:
    [D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].
    Formula:C56H77N17O13
    Color and Shape:Solid
    Molecular weight:1196.32
  • Prostaglandin E1 ethanolamide

    CAS:
    Prostaglandin E1 ethanolamide, an analog of Prostaglandin E1 (PGE1), can potentially inhibit the GLI2-induced expression of target genes such as Gli1 and Ptch1, thereby reducing tumor growth [1].
    Formula:C22H39NO5
    Color and Shape:Solid
    Molecular weight:397.55