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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5838 products of "GPCR/G-Protein"

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  • N-[(4-Aminophenyl)methyl]adenosine
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    N-[(4-Aminophenyl)methyl]adenosine

    CAS:
    N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).
    Formula:C17H20N6O4
    Purity:98.75%
    Color and Shape:Solid
    Molecular weight:372.38

    Ref: TM-T16166

  • Pimethixene maleate
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    Pimethixene maleate

    CAS:
    <p>Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.</p>
    Formula:C23H23NO4S
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:409.5

    Ref: TM-T12489L

  • EP2 receptor antagonist-2
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    EP2 receptor antagonist-2

    CAS:
    <p>CID891729, an EP2 receptor blocker, hinders PGE2 activation and reduces NMDA-induced LDH release.</p>
    Formula:C15H14F3N3O
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:309.29

    Ref: TM-T67946

  • Impromidine hydrochloride
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    Impromidine hydrochloride

    CAS:
    <p>Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.</p>
    Formula:C14H26Cl3N7S
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:430.83

    Ref: TM-T68921

  • Edonentan
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    Edonentan

    CAS:
    <p>Edonentan is A potent endothelin A (ETA) receptor antagonist that can be used to study heart failure.</p>
    Formula:C28H32N4O5S
    Purity:98.07% - 99.6%
    Color and Shape:Solid
    Molecular weight:536.64

    Ref: TM-T31605

  • Nemazoline Free Base
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    Nemazoline Free Base

    CAS:
    Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.
    Formula:C10H11Cl2N3
    Purity:98.06% - 98.83%
    Color and Shape:Solid
    Molecular weight:244.12

    Ref: TM-T71012

  • CP 96021
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    CP 96021

    CAS:
    <p>"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."</p>
    Formula:C29H21FN4OS
    Purity:97.81% - 99.62%
    Color and Shape:Soild
    Molecular weight:492.57

    Ref: TM-T10872L

  • rel-(1R,2R)-Vesamicol Hydrochloride
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    rel-(1R,2R)-Vesamicol Hydrochloride

    CAS:
    rel-(1R,2R)-Vesamicol Hydrochloride is a acetylcholine transport inhibitor.
    Formula:C17H26ClNO
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:295.85

    Ref: TM-T22486

  • GBR 12783 dihydrochloride
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    GBR 12783 dihydrochloride

    CAS:
    <p>GBR 12783 dihydrochloride inhibits dopamine uptake in rats/mice; IC50s: 1.8/1.2 nM. Enhances memory, boosts hippocampal acetylcholine.</p>
    Formula:C28H34Cl2N2O
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:485.49

    Ref: TM-T19337

  • Enerisant hydrochloride
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    Enerisant hydrochloride

    CAS:
    <p>Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteins</p>
    Formula:C22H31ClN4O3
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:434.96

    Ref: TM-T70489

  • JP1302
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    JP1302

    CAS:
    JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.
    Formula:C24H24N4
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:368.47

    Ref: TM-T22882

  • Upacicalcet
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    Upacicalcet

    CAS:
    Upacicalcet (AJT-240) is a calcium mimetic for SHPT in dialysis, reducing PTH by targeting parathyroid receptors.
    Formula:C11H14ClN3O6S
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:351.76

    Ref: TM-T29067

  • SCH-336
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    SCH-336

    CAS:
    <p>SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.</p>
    Formula:C23H25NO8S3
    Purity:95.01%
    Color and Shape:Solid
    Molecular weight:539.64

    Ref: TM-T24771

  • Tiopinac
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    Tiopinac

    CAS:
    Tiopinac: tricyclic with anti-inflammatory, analgesic, antipyretic properties; inhibits prostaglandin synthesis; mild anti-platelet effects in humans.
    Formula:C16H12O3S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:284.33

    Ref: TM-T17101

  • MM 77 dihydrochloride
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    MM 77 dihydrochloride

    CAS:
    <p>MM 77 dihydrochloride is an effecitve 5-HT1A receptor postsynaptic antagonist with anxiolytic-like activity.</p>
    Formula:C19H29Cl2N3O3
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:418.36

    Ref: TM-T23007

  • RO3244794
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    RO3244794

    CAS:
    RO3244794 is a selective prostacyclin (IP) receptor antagonist that can be used to study liver injury.
    Formula:C25H19F2NO5
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:451.42

    Ref: TM-T69360

  • ST-1535
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    ST-1535

    CAS:
    <p>ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.</p>
    Formula:C12H16N8
    Purity:99.64% - 99.69%
    Color and Shape:Solid
    Molecular weight:272.31

    Ref: TM-T28861

  • Lensiprazine
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    Lensiprazine

    CAS:
    Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and
    Formula:C24H27FN4O2
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:422.5

    Ref: TM-T32633

  • RG 7152
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    RG 7152

    CAS:
    RG 7152 is a leukotriene D4 antagonist with anti-asthmatic properties and can be used in the study of asthma.
    Formula:C20H19N5O2
    Purity:98.45%
    Color and Shape:Solid
    Molecular weight:361.4

    Ref: TM-T28529

  • Antihistamine-1
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    Antihistamine-1

    CAS:
    Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。
    Formula:C23H24FN5
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:389.47

    Ref: TM-T10335