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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5980 products of "GPCR/G-Protein"

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  • CCR2 antagonist 5

    CAS:
    JNJ-41443532: oral hCCR2 antagonist, IC50=37 nM, anti-chemotaxis, treats inflammation & diabetes.
    Formula:C22H25F3N4O3S
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:482.52

    Ref: TM-T27682

    1mg
    99.00€
    5mg
    235.00€
    10mg
    354.00€
    25mg
    635.00€
    50mg
    902.00€
    100mg
    1,225.00€
    200mg
    1,644.00€
  • Litoxetine

    CAS:
    Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.
    Formula:C16H19NO
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:241.33

    Ref: TM-T67956

    1mg
    97.00€
    5mg
    217.00€
    10mg
    325.00€
    25mg
    557.00€
    50mg
    797.00€
    100mg
    1,103.00€
    500mg
    2,205.00€
    1mL*10mM (DMSO)
    188.00€
  • Crinecerfont

    CAS:
    Crinecerfont (SSR-125543) is a CRF1 antagonist, useful in congenital adrenal hyperplasia research.
    Formula:C27H28ClFN2OS
    Purity:97.79% - 98.55%
    Color and Shape:Solid
    Molecular weight:483.04

    Ref: TM-T31095

    1mg
    92.00€
    5mg
    219.00€
    10mg
    329.00€
    25mg
    550.00€
  • L-161982

    CAS:
    L-161982 is a selective EP4 receptor antagonist that inhibits PGE2-induced ERK phosphorylation and cell proliferation in HCA-7 cells.Cost-effective and quality-assured.
    Formula:C32H29F3N4O4S2
    Purity:99.58% - 99.6%
    Color and Shape:Solid
    Molecular weight:654.72

    Ref: TM-T15681

    1mg
    70.00€
    5mg
    129.00€
    10mg
    212.00€
    25mg
    447.00€
    50mg
    642.00€
    100mg
    895.00€
    200mg
    1,206.00€
    1mL*10mM (DMSO)
    180.00€
  • Linetastine

    CAS:
    Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.
    Formula:C35H40N2O6
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:584.7

    Ref: TM-T25737

    1mg
    86.00€
    5mg
    182.00€
    10mg
    274.00€
    25mg
    449.00€
    50mg
    655.00€
    100mg
    934.00€
    200mg
    1,264.00€
  • Sonedenoson

    CAS:
    Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.
    Formula:C18H20ClN5O5
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:421.84

    Ref: TM-T34685

    1mg
    279.00€
    5mg
    685.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Tildacerfont

    CAS:
    Tildacerfont inhibits CRF1, lowers ACTH/adrenal androgens, and aids in congenital adrenal hyperplasia research.
    Formula:C20H26ClN5OS
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:419.97

    Ref: TM-T26278

    1mg
    87.00€
    5mg
    183.00€
    10mg
    280.00€
    25mg
    565.00€
    50mg
    895.00€
    100mg
    1,388.00€
  • H-9 dihydrochloride

    CAS:
    H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.
    Formula:C11H15Cl2N3O2S
    Purity:97.3%
    Color and Shape:Solid
    Molecular weight:324.23

    Ref: TM-T22833

    1mg
    35.00€
    5mg
    72.00€
    10mg
    95.00€
    25mg
    156.00€
    50mg
    225.00€
    100mg
    331.00€
  • AZD8542

    CAS:
    AZD8542 is an antagonist of Smoothened (SMO) with potential as an oncology therapeutic.
    Formula:C25H24N4O2
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:412.48

    Ref: TM-T26723

    1mg
    259.00€
    5mg
    612.00€
    10mg
    847.00€
    25mg
    1,311.00€
    50mg
    1,691.00€
    100mg
    2,232.00€
  • ISAM-140

    CAS:
    <p>ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.</p>
    Formula:C19H19N3O3
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:337.37

    Ref: TM-T27629

    1mg
    38.00€
    5mg
    84.00€
    10mg
    108.00€
    25mg
    170.00€
    50mg
    255.00€
    100mg
    363.00€
    200mg
    494.00€
  • 5-HT1A modulator 1

    CAS:
    5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).
    Formula:C21H25N3O2S
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:383.51

    Ref: TM-T10168

    1mg
    250.00€
    5mg
    610.00€
    10mg
    815.00€
    25mg
    1,206.00€
    50mg
    1,644.00€
    100mg
    2,205.00€
  • SLF1081851

    CAS:
    SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.
    Formula:C21H33N3O
    Purity:99.26%
    Color and Shape:Solid
    Molecular weight:343.51

    Ref: TM-T61112

    1mg
    56.00€
    5mg
    119.00€
    10mg
    187.00€
    25mg
    400.00€
    50mg
    597.00€
    100mg
    848.00€
  • RLX-33

    CAS:
    <p>RLX-33 blocks RXFP3 and relaxin 3 effects, controls food intake in rats, and may help study metabolic syndrome.</p>
    Formula:C24H19ClN4O4
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:462.89

    Ref: TM-T62929

    1mg
    82.00€
    5mg
    177.00€
    10mg
    284.00€
    25mg
    452.00€
    50mg
    645.00€
    100mg
    867.00€
    500mg
    1,691.00€
  • Imiloxan

    CAS:
    Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.
    Formula:C14H16N2O2
    Purity:98.13% - 99.8%
    Color and Shape:Solid
    Molecular weight:244.29

    Ref: TM-T27599

    1mg
    235.00€
    5mg
    560.00€
    10mg
    To inquire
    25mg
    1,121.00€
  • Sergliflozin etabonate

    CAS:
    Sergliflozin etabonate (KGT-1251) is an inhibitor of SGLT2 and can be used in studies about type 2 diabetes and obesity.
    Formula:C23H28O9
    Purity:97.88%
    Color and Shape:Solid
    Molecular weight:448.46

    Ref: TM-T28757

    1mg
    87.00€
    5mg
    215.00€
    10mg
    321.00€
    25mg
    518.00€
    50mg
    692.00€
    100mg
    944.00€
    1mL*10mM (DMSO)
    212.00€
  • (S)-(+)-Niguldipine hydrochloride

    CAS:
    (S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.
    Formula:C36H40ClN3O6
    Purity:98.27%
    Color and Shape:Solid
    Molecular weight:646.17

    Ref: TM-T23301

    1mg
    82.00€
    5mg
    170.00€
    10mg
    250.00€
    25mg
    588.00€
    50mg
    1,026.00€
    100mg
    1,378.00€
    500mg
    2,745.00€
  • Anpirtoline hydrochloride

    CAS:
    Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.
    Formula:C10H14Cl2N2S
    Purity:>99.99% - >99.99%
    Color and Shape:Solid
    Molecular weight:265.20

    Ref: TM-T22576

    1mg
    52.00€
    5mg
    111.00€
    10mg
    170.00€
    25mg
    283.00€
    50mg
    430.00€
    100mg
    620.00€
    500mg
    1,283.00€
  • Rilapine

    CAS:
    Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.
    Formula:C22H20ClN3
    Purity:97.76% - 99.20%
    Color and Shape:Solid
    Molecular weight:361.87

    Ref: TM-T26085

    1mg
    279.00€
    5mg
    685.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€
  • Ricasetron

    CAS:
    Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.
    Formula:C19H27N3O
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:313.44

    Ref: TM-T28537

    1mg
    44.00€
    2mg
    To inquire
    5mg
    57.00€
    10mg
    88.00€
    25mg
    156.00€
    50mg
    243.00€
    100mg
    376.00€
    200mg
    873.00€
  • CP 316311

    CAS:
    CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression.
    Formula:C21H29NO2
    Purity:99.71% - >99.99%
    Color and Shape:Solid
    Molecular weight:327.46

    Ref: TM-T15008

    1mg
    279.00€
    5mg
    507.00€
    10mg
    648.00€
    25mg
    882.00€
    50mg
    1,198.00€
    100mg
    1,596.00€