
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(53 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5980 products of "GPCR/G-Protein"
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CCR2 antagonist 5
CAS:JNJ-41443532: oral hCCR2 antagonist, IC50=37 nM, anti-chemotaxis, treats inflammation & diabetes.Formula:C22H25F3N4O3SPurity:99.98%Color and Shape:SolidMolecular weight:482.52Litoxetine
CAS:Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.Formula:C16H19NOPurity:99.68%Color and Shape:SolidMolecular weight:241.33Ref: TM-T67956
1mg97.00€5mg217.00€10mg325.00€25mg557.00€50mg797.00€100mg1,103.00€500mg2,205.00€1mL*10mM (DMSO)188.00€Crinecerfont
CAS:Crinecerfont (SSR-125543) is a CRF1 antagonist, useful in congenital adrenal hyperplasia research.Formula:C27H28ClFN2OSPurity:97.79% - 98.55%Color and Shape:SolidMolecular weight:483.04L-161982
CAS:L-161982 is a selective EP4 receptor antagonist that inhibits PGE2-induced ERK phosphorylation and cell proliferation in HCA-7 cells.Cost-effective and quality-assured.Formula:C32H29F3N4O4S2Purity:99.58% - 99.6%Color and Shape:SolidMolecular weight:654.72Ref: TM-T15681
1mg70.00€5mg129.00€10mg212.00€25mg447.00€50mg642.00€100mg895.00€200mg1,206.00€1mL*10mM (DMSO)180.00€Linetastine
CAS:Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.Formula:C35H40N2O6Purity:99.99%Color and Shape:SolidMolecular weight:584.7Sonedenoson
CAS:Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.Formula:C18H20ClN5O5Purity:99.79%Color and Shape:SolidMolecular weight:421.84Tildacerfont
CAS:Tildacerfont inhibits CRF1, lowers ACTH/adrenal androgens, and aids in congenital adrenal hyperplasia research.Formula:C20H26ClN5OSPurity:>99.99%Color and Shape:SolidMolecular weight:419.97H-9 dihydrochloride
CAS:H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.Formula:C11H15Cl2N3O2SPurity:97.3%Color and Shape:SolidMolecular weight:324.23AZD8542
CAS:AZD8542 is an antagonist of Smoothened (SMO) with potential as an oncology therapeutic.Formula:C25H24N4O2Purity:99.96%Color and Shape:SolidMolecular weight:412.48ISAM-140
CAS:<p>ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.</p>Formula:C19H19N3O3Purity:99.51%Color and Shape:SolidMolecular weight:337.375-HT1A modulator 1
CAS:5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).Formula:C21H25N3O2SPurity:99.68%Color and Shape:SolidMolecular weight:383.51SLF1081851
CAS:SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.Formula:C21H33N3OPurity:99.26%Color and Shape:SolidMolecular weight:343.51RLX-33
CAS:<p>RLX-33 blocks RXFP3 and relaxin 3 effects, controls food intake in rats, and may help study metabolic syndrome.</p>Formula:C24H19ClN4O4Purity:99.89%Color and Shape:SolidMolecular weight:462.89Imiloxan
CAS:Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.Formula:C14H16N2O2Purity:98.13% - 99.8%Color and Shape:SolidMolecular weight:244.29Sergliflozin etabonate
CAS:Sergliflozin etabonate (KGT-1251) is an inhibitor of SGLT2 and can be used in studies about type 2 diabetes and obesity.Formula:C23H28O9Purity:97.88%Color and Shape:SolidMolecular weight:448.46Ref: TM-T28757
1mg87.00€5mg215.00€10mg321.00€25mg518.00€50mg692.00€100mg944.00€1mL*10mM (DMSO)212.00€(S)-(+)-Niguldipine hydrochloride
CAS:(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.Formula:C36H40ClN3O6Purity:98.27%Color and Shape:SolidMolecular weight:646.17Anpirtoline hydrochloride
CAS:Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.Formula:C10H14Cl2N2SPurity:>99.99% - >99.99%Color and Shape:SolidMolecular weight:265.20Rilapine
CAS:Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.Formula:C22H20ClN3Purity:97.76% - 99.20%Color and Shape:SolidMolecular weight:361.87Ricasetron
CAS:Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Formula:C19H27N3OPurity:99.52%Color and Shape:SolidMolecular weight:313.44Ref: TM-T28537
1mg44.00€2mgTo inquire5mg57.00€10mg88.00€25mg156.00€50mg243.00€100mg376.00€200mg873.00€CP 316311
CAS:CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression.Formula:C21H29NO2Purity:99.71% - >99.99%Color and Shape:SolidMolecular weight:327.46
