GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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CCK Octapeptide, non-sulfated acetate
<p>CCK Octapeptide, non-sulfated acetate is a synthetic desulfated peptide of cholecystokinin.</p>Formula:C51H66N10O15S2Purity:98.9700%Color and Shape:SolidMolecular weight:1123.26Cortistatin-14 acetate
<p>Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5).</p>Formula:C83H118N20O20S2Purity:98.24% - 99.63%Color and Shape:SoildMolecular weight:1780.08CGRP antagonist 6
<p>CGRP Antagonist 6 (Compound 23) is a potent CGRP receptor antagonist (Ki: 0.84 nM). It is utilized in the study of migraines.</p>Color and Shape:Odour SolidBMS-753426
CAS:<p>BMS-753426 is a potent and orally bioavailable antagonist of CCR2 .</p>Formula:C25H33F3N6O2Color and Shape:SolidMolecular weight:506.574HAEGTFTSD
CAS:<p>HAEGTFTSD is GLP-1's initial segment; GLP-1 (7-36) amide, tied to food intake, stems from preproglucagon in L-cells.</p>Formula:C40H57N11O17Purity:98%Color and Shape:SolidMolecular weight:963.94Pasireotide
CAS:Pasireotide (SOM 230) is a cyclohexapeptide, mimicking somatostatin with high affinity for sst1/2/3/4/5 receptors (pKi=8.2/9.0/9.1/<7.0/9.9).Formula:C58H66N10O9Purity:98%Color and Shape:SolidMolecular weight:1047.21JKC363
CAS:<p>MC4 receptor antagonist; IC50: 0.5 nM (MC4), 44.9 nM (MC3). Blocks α-MSH, reduces TRH, food intake, and pain.</p>Formula:C69H91N19O16S2Purity:98%Color and Shape:SolidMolecular weight:1506.72Chemerin-9 (149-157) TFA
<p>Chemerin-9 (149-157) TFA is a peptide located at positions 149-157 of chemerin-9, acting as a ChemR23/CMKLR1 agonist.</p>Formula:C56H67F3N10O15Purity:99.77%Color and Shape:SolidMolecular weight:1177.18Linzagolix choline
CAS:<p>Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.</p>Formula:C27H28F3N3O8SPurity:99.64%Color and Shape:SolidMolecular weight:611.59SGLT1/2-IN-2
CAS:<p>SGLT1/2-IN-2 is a chemical compound with robust dual inhibitory properties, exhibiting potent activities against SGLT1 (IC50 = 96 nM) and SGLT2 (IC50 = 1.3 nM).</p>Formula:C23H26F2O7Color and Shape:SolidMolecular weight:452.451A71378
CAS:<p>A71378 is a high potency, selectivity CCK-A receptors agonist.</p>Formula:C48H62N8O13SPurity:98%Color and Shape:SolidMolecular weight:991.12Enuvaptan
CAS:<p>Enuvaptan is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.</p>Formula:C21H15ClF6N8O3Color and Shape:SolidMolecular weight:576.84MCUF-651
CAS:<p>MCUF-651 is a guanylyl cyclase A receptor positive allosteric modulators, EC50=0.45 μM.</p>Formula:C17H22F2N4OSPurity:99.83%Color and Shape:SoildMolecular weight:368.44(R)-Preclamol hydrochloride
CAS:<p>(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.</p>Formula:C14H22ClNOColor and Shape:SolidMolecular weight:255.78cAC 253 acetate
<p>cAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin binding, with an IC50 of 25 nM.</p>Formula:C128H206N42O42S2Purity:98.16% - 99.99%Color and Shape:SoildMolecular weight:3069.39{Val1}-Exendin-3/4
{Val1}- exendin-3/4 is the first n-terminal 1-28 residue of exendin-4 peptide.Formula:NAPurity:98%Color and Shape:SolidMolecular weight:3241.7Upidosin
CAS:<p>Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.</p>Formula:C31H33N3O4Purity:99.66%Color and Shape:SolidMolecular weight:511.61I-BOP
CAS:<p>I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).</p>Formula:C23H29IO5Color and Shape:SolidMolecular weight:512.384Y1 receptor antagonist 1 formic
<p>H 409-22 isomer formic, a formate salt of Y1 receptor antagonist 1, is an antagonist of the neuropeptide Y1 receptor (neuropeptide Y1 receptor). This compound effectively blocks the actions of the receptor, playing a crucial role in modulating physiological responses.</p>Formula:C29H35N5O5Color and Shape:SolidMolecular weight:533.62Adenosine receptor agonist 1
<p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>Formula:C12H14ClN5O2SeColor and Shape:SolidMolecular weight:374.68
