GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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Sergliflozin etabonate
CAS:Sergliflozin etabonate (KGT-1251) is an inhibitor of SGLT2 and can be used in studies about type 2 diabetes and obesity.Formula:C23H28O9Purity:97.88%Color and Shape:SolidMolecular weight:448.46Ref: TM-T28757
1mg87.00€5mg215.00€10mg321.00€25mg518.00€50mg692.00€100mg944.00€1mL*10mM (DMSO)212.00€L-693,403 maleate
CAS:L-693,403 maleate has analgesic activity.Formula:C24H27NO4Purity:99.88%Color and Shape:SolidMolecular weight:393.48Ref: TM-T22899
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Formula:C21H24Cl2N2O2Purity:98.58%Color and Shape:SolidMolecular weight:407.33N6-(2-Phenylethyl)adenosine
CAS:N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM forFormula:C18H21N5O4Purity:99.83%Color and Shape:SolidMolecular weight:371.39Milveterol HCl
CAS:Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).Formula:C25H30ClN3O4Purity:99.9%Color and Shape:SolidMolecular weight:471.98Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Formula:C25H19F3N4O5SPurity:98.60% - 98.97%Color and Shape:SolidMolecular weight:544.5U 99194 maleate
CAS:U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.Formula:C21H31NO6Purity:99.45%Color and Shape:SolidMolecular weight:393.47Faxeladol
CAS:Faxeladol: adrenergic, serotonin inhibitor & opioid agonist for neurological studies.Formula:C15H23NOPurity:98.77% - 99.67%Color and Shape:SolidMolecular weight:233.35RS 42358-197
CAS:RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Formula:C19H23ClN2OPurity:99.70%Color and Shape:SolidMolecular weight:330.85Ref: TM-T20739
1mg158.00€5mg351.00€10mg527.00€25mg783.00€50mg1,054.00€100mg1,414.00€200mg1,908.00€1mL*10mM (DMSO)349.00€A-437203
CAS:A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.Formula:C20H27F3N6OSPurity:98.80%Color and Shape:SolidMolecular weight:456.53Ref: TM-T10213
1mg94.00€5mg188.00€10mg264.00€25mg411.00€50mg532.00€100mg740.00€200mg982.00€1mL*10mM (DMSO)215.00€SB-215505
CAS:SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).Formula:C19H16ClN3OPurity:98.33%Color and Shape:SolidMolecular weight:337.8Sarizotan HCl
CAS:Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.Formula:C22H22ClFN2OPurity:96%Color and Shape:SolidMolecular weight:384.87Runcaciguat
CAS:Runcaciguat, a soluble guanylate cyclase stimulator, aids in cardiovascular and renal research.Formula:C23H22Cl2F3NO3Purity:99.17%Color and Shape:SolidMolecular weight:488.33Goxalapladib
CAS:Goxalapladib（GSK 677116） is a small molecule compound that can be used to treat cardiovascular risks associated with atherosclerosis.Formula:C40H39F5N4O3Purity:99.64% - 99.93%Color and Shape:SolidMolecular weight:718.75Torbafylline
CAS:Torbafylline is a xanthine-based PDE inhibitor reducing protein breakdown via PDE4/cAMP/EPAC/PI3K/Akt in rats with burns, cancer, or sepsis.Formula:C16H26N4O4Purity:99.96% - 99.97%Color and Shape:SoildMolecular weight:338.4Ref: TM-T67965
1mg81.00€5mg172.00€10mg259.00€25mg424.00€50mg583.00€100mg800.00€1mL*10mM (DMSO)178.00€cis-Urocanic acid
CAS:cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).Formula:C6H6N2O2Purity:99.81%Color and Shape:SolidMolecular weight:138.12(R)-ZINC-3573
CAS:<p>ZINC-3573: Potent, selective MRGPRX2 activator; triggers mast cell degranulation and calcium release.</p>Formula:C18H21N5Purity:99.75%Color and Shape:SolidMolecular weight:307.39Thiethylperazine dimaleate
CAS:Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor.Formula:C30H37N3O8S2Purity:99.88%Color and Shape:SolidMolecular weight:631.76CV-6209
CAS:CV-6209 is a potent antagonist of the platelet-activating factor (PAF) receptor.Formula:C34H60ClN3O6Purity:>99.99% - >99.99%Color and Shape:SolidMolecular weight:642.31TASP0390325
CAS:<p>TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in rodents.</p>Formula:C25H30Cl2FN5O4Purity:98.62%Color and Shape:SolidMolecular weight:554.44
