
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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Masupirdine free base
CAS:Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formula:C21H24BrN3O3SPurity:98.36% - 99.65%Color and Shape:SolidMolecular weight:478.4CL 316243
CAS:CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.Formula:C20H18ClNNa2O7Purity:98.00% - 99.68%Color and Shape:SolidMolecular weight:465.79RO3244794
CAS:RO3244794 is a selective prostacyclin (IP) receptor antagonist that can be used to study liver injury.Formula:C25H19F2NO5Purity:99.36%Color and Shape:SolidMolecular weight:451.42Lesopitron
CAS:Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.Formula:C15H21ClN6Purity:99.33% - 99.46%Color and Shape:SolidMolecular weight:320.82Ref: TM-T25672
1mg133.00€5mg324.00€10mg477.00€25mg773.00€50mg1,063.00€100mg1,431.00€500mg2,872.00€1mL*10mM (DMSO)323.00€Liafensine
CAS:Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.Formula:C24H22N4Purity:99.91%Color and Shape:SolidMolecular weight:366.46LX-2931
CAS:LX-2931(LX-3305) is a sphingosine-1-phosphate cleavage enzyme (S1P) inhibitor for the treatment of rheumatoid arthritis.Formula:C9H15N3O5Purity:98.85% - 99.83%Color and Shape:SolidMolecular weight:245.23(S)-(+)-Niguldipine hydrochloride
CAS:(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.Formula:C36H40ClN3O6Purity:98.27%Color and Shape:SolidMolecular weight:646.17CP 316311
CAS:CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression.Formula:C21H29NO2Purity:99.71% - >99.99%Color and Shape:SolidMolecular weight:327.46Pavinetant
CAS:Pavinetant (MLE-4901) is an orally available neurokinin-3 receptor (NK3R) antagonist used to improve menopausal symptoms.Formula:C26H25N3O3SPurity:99.8%Color and Shape:SolidMolecular weight:459.56Ref: TM-T16114
1mg77.00€2mg99.00€5mg166.00€10mg245.00€25mg326.00€50mg409.00€100mg590.00€1mL*10mM (DMSO)169.00€N6-(2-Phenylethyl)adenosine
CAS:N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM forFormula:C18H21N5O4Purity:99.83%Color and Shape:SolidMolecular weight:371.39SCH-336
CAS:SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.Formula:C23H25NO8S3Purity:97.00%Color and Shape:SolidMolecular weight:539.64Ref: TM-T24771
5mg49.00€10mg73.00€25mg152.00€50mg213.00€100mg309.00€200mg444.00€1mL*10mM (DMSO)60.00€BP14979
CAS:BP14979 is D3R-selective partial agonist.Formula:C23H34N4O2Purity:98.29% - 99.73%Color and Shape:SolidMolecular weight:398.54SK609 HCl
CAS:SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.Formula:C10H15Cl2NPurity:99.02%Color and Shape:SolidMolecular weight:220.14UNC0006
CAS:UNC0006 is a β-arrestin-biased dopamine D2 ligand.
Formula:C24H29Cl2N3O2Purity:99.35% - 99.97%Color and Shape:SolidMolecular weight:462.41Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formula:C23H26N2OPurity:98.03% - 98.93%Color and Shape:SolidMolecular weight:346.47Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Formula:C25H19F3N4O5SPurity:98.60% - 98.97%Color and Shape:SolidMolecular weight:544.5Itriglumide
CAS:Itriglumide, a CCK2 receptor antagonist, is used potentially for the treatment of peptic ulcers, dyspepsia, and gastroesophageal reflux disease (GERD).Formula:C33H38N2O4Purity:99.95%Color and Shape:SolidMolecular weight:526.67PNU-282987 free base
CAS:PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.
Formula:C14H17ClN2OPurity:99.64%Color and Shape:SolidMolecular weight:264.75Dimethindene maleate
CAS:Dimethindene maleate (SU 6518) is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.Formula:C24H28N2O4Purity:99.79%Color and Shape:SolidMolecular weight:408.49Ref: TM-T21472
1mg34.00€5mg71.00€10mg105.00€25mg236.00€50mg313.00€100mg409.00€200mg582.00€1mL*10mM (DMSO)82.00€7-Hydroxy-DPAT hydrobromide
CAS:7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.Formula:C16H26BrNOPurity:99.73%Color and Shape:SolidMolecular weight:328.29
