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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • Masupirdine free base

    CAS:
    Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.
    Formula:C21H24BrN3O3S
    Purity:98.36% - 99.65%
    Color and Shape:Solid
    Molecular weight:478.4

    Ref: TM-T11948

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
    1mL*10mM (DMSO)
    424.00€
  • CL 316243

    CAS:
    CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.
    Formula:C20H18ClNNa2O7
    Purity:98.00% - 99.68%
    Color and Shape:Solid
    Molecular weight:465.79

    Ref: TM-T10830

    1mg
    50.00€
    5mg
    105.00€
    10mg
    160.00€
    25mg
    313.00€
    50mg
    500.00€
    100mg
    To inquire
    500mg
    To inquire
  • RO3244794

    CAS:
    RO3244794 is a selective prostacyclin (IP) receptor antagonist that can be used to study liver injury.
    Formula:C25H19F2NO5
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:451.42

    Ref: TM-T69360

    1mg
    161.00€
    5mg
    384.00€
    10mg
    482.00€
    25mg
    712.00€
    50mg
    954.00€
    100mg
    1,288.00€
    200mg
    1,738.00€
  • Lesopitron

    CAS:
    Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.
    Formula:C15H21ClN6
    Purity:99.33% - 99.46%
    Color and Shape:Solid
    Molecular weight:320.82

    Ref: TM-T25672

    1mg
    133.00€
    5mg
    324.00€
    10mg
    477.00€
    25mg
    773.00€
    50mg
    1,063.00€
    100mg
    1,431.00€
    500mg
    2,872.00€
    1mL*10mM (DMSO)
    323.00€
  • Liafensine

    CAS:
    Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.
    Formula:C24H22N4
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:366.46

    Ref: TM-T32737

    1mg
    349.00€
    5mg
    830.00€
    10mg
    1,134.00€
    25mg
    1,684.00€
    50mg
    2,268.00€
  • LX-2931

    CAS:
    LX-2931(LX-3305) is a sphingosine-1-phosphate cleavage enzyme (S1P) inhibitor for the treatment of rheumatoid arthritis.
    Formula:C9H15N3O5
    Purity:98.85% - 99.83%
    Color and Shape:Solid
    Molecular weight:245.23

    Ref: TM-T27864

    1mg
    233.00€
    5mg
    577.00€
    10mg
    822.00€
    25mg
    1,234.00€
    50mg
    1,665.00€
  • (S)-(+)-Niguldipine hydrochloride

    CAS:
    (S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.
    Formula:C36H40ClN3O6
    Purity:98.27%
    Color and Shape:Solid
    Molecular weight:646.17

    Ref: TM-T23301

    1mg
    78.00€
    5mg
    167.00€
    10mg
    236.00€
    25mg
    557.00€
    50mg
    973.00€
    100mg
    1,305.00€
    500mg
    2,602.00€
  • CP 316311

    CAS:
    CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression.
    Formula:C21H29NO2
    Purity:99.71% - >99.99%
    Color and Shape:Solid
    Molecular weight:327.46

    Ref: TM-T15008

    1mg
    264.00€
    5mg
    480.00€
    10mg
    615.00€
    25mg
    835.00€
    50mg
    1,134.00€
    100mg
    1,513.00€
  • Pavinetant

    CAS:
    Pavinetant (MLE-4901) is an orally available neurokinin-3 receptor (NK3R) antagonist used to improve menopausal symptoms.
    Formula:C26H25N3O3S
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:459.56

    Ref: TM-T16114

    1mg
    77.00€
    2mg
    99.00€
    5mg
    166.00€
    10mg
    245.00€
    25mg
    326.00€
    50mg
    409.00€
    100mg
    590.00€
    1mL*10mM (DMSO)
    169.00€
  • N6-(2-Phenylethyl)adenosine

    CAS:
    N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for
    Formula:C18H21N5O4
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:371.39

    Ref: TM-T12163

    10mg
    33.00€
    25mg
    59.00€
    50mg
    104.00€
    100mg
    177.00€
    200mg
    316.00€
    1mL*10mM (DMSO)
    33.00€
  • SCH-336

    CAS:
    SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.
    Formula:C23H25NO8S3
    Purity:97.00%
    Color and Shape:Solid
    Molecular weight:539.64

    Ref: TM-T24771

    5mg
    49.00€
    10mg
    73.00€
    25mg
    152.00€
    50mg
    213.00€
    100mg
    309.00€
    200mg
    444.00€
    1mL*10mM (DMSO)
    60.00€
  • BP14979

    CAS:
    BP14979 is D3R-selective partial agonist.
    Formula:C23H34N4O2
    Purity:98.29% - 99.73%
    Color and Shape:Solid
    Molecular weight:398.54

    Ref: TM-T26890

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
  • SK609 HCl

    CAS:
    SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.
    Formula:C10H15Cl2N
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:220.14

    Ref: TM-T24797

    1mg
    69.00€
    5mg
    147.00€
    10mg
    212.00€
    25mg
    356.00€
    50mg
    510.00€
    100mg
    712.00€
    200mg
    982.00€
  • UNC0006

    CAS:

    UNC0006 is a β-arrestin-biased dopamine D2 ligand.

    Formula:C24H29Cl2N3O2
    Purity:99.35% - 99.97%
    Color and Shape:Solid
    Molecular weight:462.41

    Ref: TM-T29061

    1mg
    279.00€
    5mg
    685.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€
  • Roxindole

    CAS:
    Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.
    Formula:C23H26N2O
    Purity:98.03% - 98.93%
    Color and Shape:Solid
    Molecular weight:346.47

    Ref: TM-T26126

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • Opigolix

    CAS:
    Opigolix is a Gonadotropin-releasing hormone receptor antagonist.
    Formula:C25H19F3N4O5S
    Purity:98.60% - 98.97%
    Color and Shape:Solid
    Molecular weight:544.5

    Ref: TM-T17301

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
    50mg
    1,063.00€
    100mg
    1,485.00€
  • Itriglumide

    CAS:
    Itriglumide, a CCK2 receptor antagonist, is used potentially for the treatment of peptic ulcers, dyspepsia, and gastroesophageal reflux disease (GERD).
    Formula:C33H38N2O4
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:526.67

    Ref: TM-T27640

    1mg
    264.00€
    2mg
    393.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • PNU-282987 free base

    CAS:

    PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.

    Formula:C14H17ClN2O
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:264.75

    Ref: TM-T60437

    1mg
    55.00€
    5mg
    111.00€
    10mg
    202.00€
    25mg
    394.00€
    50mg
    732.00€
    100mg
    1,026.00€
    500mg
    2,052.00€
  • Dimethindene maleate

    CAS:
    Dimethindene maleate (SU 6518) is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.
    Formula:C24H28N2O4
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:408.49

    Ref: TM-T21472

    1mg
    34.00€
    5mg
    71.00€
    10mg
    105.00€
    25mg
    236.00€
    50mg
    313.00€
    100mg
    409.00€
    200mg
    582.00€
    1mL*10mM (DMSO)
    82.00€
  • 7-Hydroxy-DPAT hydrobromide

    CAS:
    7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.
    Formula:C16H26BrNO
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:328.29

    Ref: TM-T22531

    1mg
    49.00€
    5mg
    94.00€
    10mg
    153.00€
    25mg
    246.00€
    50mg
    370.00€