GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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JP1302
CAS:JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.Formula:C24H24N4Purity:99.96%Color and Shape:SolidMolecular weight:368.47(±)-Fabesetron hydrochloride
CAS:FK1052 hydrochloride is a potent 5-HT3 and 5-HT4 receptor dual antagonist.Formula:C18H20ClN3OPurity:98%Color and Shape:SolidMolecular weight:329.82BMS-604992
CAS:EX-1314 (BMS-604992) is a growth hormone secretagogue receptor (GHSR) agonist.Formula:C24H32ClN7O5Color and Shape:SolidMolecular weight:534.01Ciprostene (calcium salt)
CAS:Ciprostene, a PGI2 stable analog, is less potent, induces hypotension, tachycardia, and inhibits platelet aggregation in monkeys.Formula:C44H74CaO8Color and Shape:SolidMolecular weight:771.146Celiprolol hydrochloride
CAS:Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.Formula:C20H33N3O4·HClColor and Shape:White Crystalline SolidMolecular weight:415.96DG-041
CAS:DG-041: EP3 receptor antagonist, high affinity (IC50: 4.6 & 8.1 nM), inhibits PGE2 in platelets, blood-brain barrier permeable.Formula:C23H15Cl4FN2O3S2Purity:99.77%Color and Shape:SolidMolecular weight:592.32Ref: TM-T15108
1mg48.00€2mg63.00€5mg92.00€10mg150.00€25mg284.00€50mg512.00€100mg737.00€500mg1,521.00€1mL*10mM (DMSO)104.00€Lazuvapagon
CAS:Lazuvapagon is a vasopressin V2 receptor agonist that can be used to study enuresis.Formula:C27H32N4O3Color and Shape:SolidMolecular weight:460.57Fiduxosin
CAS:Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with KiFormula:C30H29N5O4SPurity:99.73%Color and Shape:SolidMolecular weight:555.65Maropitant citrate anhydrous
CAS:Maropitant citrate anhydrous is a neurokinin (NK1) receptor antagonist.Formula:C38H48N2O8Color and Shape:SolidMolecular weight:660.8PW0464
CAS:PW0464 ((Rac)-Razpipadon) is a non-catechol D1R agonist and potent omplete G protein biased ligand with an EC50 (Gs-cAMP)=5.8 nM for neurological disorders.Formula:C19H17F2N3O4Purity:98.78%Color and Shape:SolidMolecular weight:389.35Ref: TM-T36946
1mg160.00€5mg386.00€10mg635.00€25mg1,228.00€50mg1,839.00€100mg2,470.00€1mL*10mM (DMSO)425.00€S1p receptor agonist 2
CAS:S1P5-selective agonist; less so for S1P1/S1P3; useful for CNS disorders.Formula:C24H23ClN2O4Color and Shape:SolidMolecular weight:438.9IIIM-8
CAS:IIIM-8 is a melanogenesis inhibitor that suppresses pigment production in both in vitro and in vivo settings, exhibiting no cytotoxic effects on Human AdultFormula:C14H17NO4Purity:98%Color and Shape:SolidMolecular weight:263.29GLP-1R agonist 12
CAS:GLP-1R agonist 12 (Compound 123) 是一种 GLP-1R 激动剂，能够用于研究糖尿病。Formula:C34H36N6O4Color and Shape:SolidMolecular weight:592.695-HT2 agonist-1
CAS:Compound 24, a 5-HT2 agonist-1, selectively activates 5-HT2A, 5-HT2B, and 5-HT2C receptors with IC50 values of 10 nM, 8.3 nM, and 1.6 nM, respectively.Formula:C19H23ClN2O2Purity:98%Color and Shape:SolidMolecular weight:346.85Prostaglandin E2-1-glyceryl ester
CAS:Prostaglandin E2-1-glyceryl ester, a member of the Prostaglandin Glycerol Ester family, serves as an endocannabinoid ligand targeting the CB1 receptor. This compound triggers a swift and transient surge in intracellular free calcium levels [1] [2].Formula:C23H38O7Color and Shape:SolidMolecular weight:426.55RXFP1 receptor agonist-7
CAS:RXFP1 receptor agonist-7 (Example 2) serves as an RXFP1 receptor agonist, effectively inhibiting cAMP production in HEK293 cells that stably express the humanFormula:C40H32F5N3O7Color and Shape:SolidMolecular weight:761.69FAUC-312
CAS:FAUC-312 is a potent and selective agonist of the dopamine D4 receptor.Formula:C21H26N4Purity:98%Color and Shape:SolidMolecular weight:334.46Y1R probe-1
CAS:Compound 39, or Y1R probe-1, is a fluorescent probe for Neuropeptide Y Y1 Receptor used in cancer research.Formula:C64H71F3N10O12Color and Shape:SolidMolecular weight:1229.3Veldoreotide TFA
CAS:Veldoreotide (DG3173) TFA, a somatostatin analogue, effectively binds to and activates somatostatin receptors (SSTR) 2, 4, and 5. This compound demonstrates a higher efficacy in inhibiting growth hormone (GH) secretion in adenomas than Octreotide, showcasing its potential as a pain modulating agent [1].Formula:C62H75F3N12O12Color and Shape:SolidMolecular weight:1237.33BU-E 75
CAS:BU-E 75 is an agonist of the histamine H2.Formula:C21H24F2N6Color and Shape:SolidMolecular weight:398.45
