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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • 5α-Pregnane-3α,20α-diol

    CAS:
    5α-Pregnane-3α,20α-diol, an active metabolite of progesterone, is synthesized through intermediates 5α-pregnane-20α-ol-3-one and 5α-pregnane-3α-ol-20-one from
    Formula:C21H36O2
    Color and Shape:Solid
    Molecular weight:320.51

    Ref: TM-T83859

    1mg
    140.00€
    10mg
    733.00€
  • PZ-1190

    CAS:
    PZ-1190, a multitarget ligand for serotonin and dopamine receptors, exhibits potential antipsychotic activity in rodents [1].
    Formula:C27H30N4O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:506.68

    Ref: TM-T81336

    5mg
    To inquire
    50mg
    To inquire
  • Desethoxy Quetiapine hydrochloride

    CAS:
    Desethoxy quetiapine, an active metabolite of the atypical antipsychotic quetiapine, primarily forms through the action of the cytochrome P450 (CYP) isoform CYP3A5. This compound binds to dopamine D2 receptors with an IC50 value of 1,330 nM. In vivo, desethoxy quetiapine at dosages of 20 and 40 mg/kg mitigates dopamine receptor agonist apomorphine-induced climbing behavior and ameliorates swimming deficits in mice, showcasing its potential modulatory effects on dopamine-mediated behaviors.
    Formula:C19H21N3OSHCl
    Color and Shape:Solid
    Molecular weight:412.38

    Ref: TM-T84947

    10mg
    To inquire
    50mg
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  • Maropitant citrate anhydrous

    CAS:
    Maropitant citrate anhydrous is a neurokinin (NK1) receptor antagonist.
    Formula:C38H48N2O8
    Color and Shape:Solid
    Molecular weight:660.8

    Ref: TM-T68519

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • SB 649915

    CAS:
    SB 649915 is a serotonin reuptake inhibitor and 5-HT1A and 5-HT1B receptor antagonist.
    Formula:C26H29N3O3
    Color and Shape:Solid
    Molecular weight:431.53

    Ref: TM-T28678

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • 5-HT2 agonist-1

    CAS:
    Compound 24, a 5-HT2 agonist-1, selectively activates 5-HT2A, 5-HT2B, and 5-HT2C receptors with IC50 values of 10 nM, 8.3 nM, and 1.6 nM, respectively.
    Formula:C19H23ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:346.85

    Ref: TM-T79804

    5mg
    To inquire
    50mg
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  • AR-08

    CAS:
    AR-08 is a potent α2-adrenergic receptor agonist for the study of ADHD and attention deficit.
    Formula:C12H12N6
    Purity:99.7%
    Color and Shape:Solid
    Molecular weight:240.26

    Ref: TM-T10052

    1mg
    630.00€
    5mg
    1,620.00€
  • PD 160170

    CAS:
    neuropeptide Y1 receptor antagonist
    Formula:C18H17N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:371.41

    Ref: TM-T23126

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • L 659837

    CAS:
    L 659837 is an antagonist of ANC-2, lactam, and tackykinin.
    Formula:C40H52N8O7S
    Color and Shape:Solid
    Molecular weight:788.96

    Ref: TM-T24312

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • IIIM-8

    CAS:
    IIIM-8 is a melanogenesis inhibitor that suppresses pigment production in both in vitro and in vivo settings, exhibiting no cytotoxic effects on Human Adult
    Formula:C14H17NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:263.29

    Ref: TM-T79378

    5mg
    To inquire
    50mg
    To inquire
  • Capeserod HCl

    CAS:
    Capeserod HCl, a 5-hydroxytriptamine 4 (5-HT4) receptor agonist, is used potentially for the treatment of Alzheimer's disease.
    Formula:C23H26Cl2N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:493.38

    Ref: TM-T26944

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • LBT 999

    CAS:
    LBT 999 is used as a dopamine reuptake inhibitor.
    Formula:C20H26FNO2
    Color and Shape:Solid
    Molecular weight:331.42

    Ref: TM-T25647

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • LY 53857

    CAS:
    LY 53857 is a potent and selective antagonist of 5-HT2 serotonin receptor.
    Formula:C27H36N2O7
    Color and Shape:Solid
    Molecular weight:500.592

    Ref: TM-T27921

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • PAC1R antagonist 1

    CAS:
    PAC1R antagonist 1 is a PAC1 receptor antagonist that inhibits the activation of peptides by pituitary adenylate cyclase and can be used to study tumours.
    Formula:C17H17ClN6O2
    Purity:98.43% - 99.56%
    Color and Shape:Solid
    Molecular weight:372.81

    Ref: TM-T78105

    1mg
    87.00€
    5mg
    To inquire
    10mg
    To inquire
    25mg
    To inquire
    50mg
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    100mg
    To inquire
    1mL*10mM (DMSO)
    To inquire
  • Apelin agonist 1

    CAS:
    Apelin agonist 1 is an orally available APJ receptor agonist with an EC50 value of 3.2 nM. Apelin agonist 1 is used in the study of cardiovascular disease.
    Formula:C23H20FN5O5S
    Purity:97.69% - 99.07%
    Color and Shape:Solid
    Molecular weight:497.5

    Ref: TM-T10346

    1mg
    1,071.00€
    5mg
    2,178.00€
    10mg
    2,943.00€
  • Brilaroxazine

    CAS:
    Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.
    Formula:C22H25Cl2N3O3
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:450.36

    Ref: TM-T14782

    1mg
    100.00€
    5mg
    236.00€
    10mg
    385.00€
    25mg
    663.00€
    50mg
    954.00€
    100mg
    1,305.00€
    200mg
    1,738.00€
    1mL*10mM (DMSO)
    268.00€
  • TG6-129

    CAS:
    TG6-129 is an EP2 receptor antagonist, blocking PGE2 effects, reducing inflammatory markers with 1.6 µM IC50.
    Formula:C20H18FN5O3S3
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:491.58

    Ref: TM-T28958

    1mg
    114.00€
    5mg
    227.00€
    10mg
    404.00€
    25mg
    665.00€
    50mg
    888.00€
    100mg
    1,251.00€
    500mg
    2,538.00€
    1mL*10mM (DMSO)
    321.00€
  • CCG-63802

    CAS:
    CCG-63802 is a reversible small-molecule inhibitor of regulator of G protein signaling (RGS) proteins.
    Formula:C26H18N4O2S
    Purity:90%
    Color and Shape:Solid
    Molecular weight:450.51

    Ref: TM-T14897

    2mg
    40.00€
    5mg
    59.00€
    10mg
    90.00€
    25mg
    170.00€
  • BMY-42393

    CAS:
    BMY-42393 is an oral prostacyclin agonist and platelet aggregation inhibitor with IC50 of 0.3-2μM and stimulates adenylate cyclase (EC50 = 25nM).
    Formula:C25H21NO4
    Color and Shape:Solid
    Molecular weight:399.44

    Ref: TM-T70865

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • CB1 antagonist 1

    CAS:
    CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and metabolic syndrome, neuroinflammatory disorders, cognitive disorders, and
    Formula:C26H22Cl2N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:461.39

    Ref: TM-T10510

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€