GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,024 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
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S1PL-IN-31
CAS:S1PL-IN-31 is a dual-function chemical compound acting as an inhibitor of sphingosine-1-phosphate (S1P) lyase with an IC50 value of 210 nM and as an antagonistFormula:C26H23ClN6Color and Shape:SolidMolecular weight:454.95Quinpirole dihydrochloride
CAS:Quinpirole dihydrochloride is an agonist of the D2-like dopamine receptor.Formula:C13H23Cl2N3Purity:98%Color and Shape:SolidMolecular weight:292.25Uridine 5'-diphosphate
CAS:Uridine 5'-diphosphate acts as a P2Y6 receptor agonist, exhibiting an EC50 value of 0.013 μM for the human P2Y6 receptor [1].Formula:C9H14N2O12P2Purity:98%Color and Shape:SolidMolecular weight:404.16PSB-SB1202
CAS:PSB-SB1202 (Compound 21a), a phenyl coumarin compound, acts as a CB1/CB2 agonist. It demonstrates EC50 values of 56 and 14 nM and K i values of 32 and 49 nM for CB1 and CB2 receptors, respectively [1].Formula:C23H26O4Color and Shape:SolidMolecular weight:366.45Brilaroxazine
CAS:Brilaroxazine (RP5063): multimodal dopamine/5-HT modulator, partial agonist at D2/D3/D4, 5-HT1A/2A, and antagonist at 5-HT2B/7.Formula:C22H25Cl2N3O3Purity:99.36%Color and Shape:SolidMolecular weight:450.36Ref: TM-T14782
1mg100.00€5mg236.00€1mL*10mM (DMSO)268.00€10mg385.00€25mg663.00€50mg954.00€100mg1,305.00€200mg1,738.00€5-HT2C agonist-3
CAS:5-HT2C agonist-3 ((+)-19), a selective 5-HT2C agonist (EC 50: 24 nM, Ki: 78 nM), exhibits antipsychotic-like activity by blocking amphetamine-inducedFormula:C19H23ClFNO2Purity:98%Color and Shape:SolidMolecular weight:351.84(S)-Bexicaserin
CAS:(S)-Bexcaserin (compound 2) serves as a 5-HT2C receptor agonist, presenting research possibilities in obesity and psychiatric disorders [1].Formula:C15H19F2N3OPurity:98%Color and Shape:SolidMolecular weight:295.33Mocravimod hydrochloride
CAS:Mocravimod hydrochloride (KRP-203) is an effecitive and orally active agonist of sphingosine 1-phosphate receptor type 1(S1PR1).Formula:C24H27Cl2NO3SPurity:90%Color and Shape:SolidMolecular weight:480.45Ref: TM-T12086
1mg66.00€5mg160.00€1mL*10mM (DMSO)169.00€10mg250.00€25mg507.00€50mg785.00€100mg1,054.00€TCS 2510
CAS:TCS 2510 (CAY10598) 是一种选择性 PGE2 和 EP4 受体激动剂，可增强细胞内 cAMP 浓度和活性 β-caten 的丰度。TCS 2510 抑制TNF-α 产生，可用于研究代谢紊乱带来的疾病。Formula:C21H29N5O2Purity:98%Color and Shape:SolidMolecular weight:383.49KUC-7322
CAS:Ritobegron is used as a selective β3-adrenoceptor agonist and the prodrug of the active compound, KUC-7322.Formula:C21H27NO5Color and Shape:SolidMolecular weight:373.44LY-368975
CAS:LY-368975 is a potent and selective inhibitor of the norepinephrine (NE) reuptake site. LY-368975 reduces food consumption in rodents.Formula:C17H21NOSColor and Shape:SolidMolecular weight:287.42AH13205
CAS:AH13205 is an agonist of EP2 prostanoid receptor.Formula:C24H36O4Purity:98%Color and Shape:SolidMolecular weight:388.54Cenerimod
CAS:Cenerimod (ACT-334441) is an S1P1 agonist used in the study of murine experimental autoimmune encephalomyelitis (EAE) and murine scleroderma.Formula:C25H31N3O5Purity:97.43% - 99.97%Color and Shape:SolidMolecular weight:453.53FR-181157
CAS:FR-181157, a novel prostaglandin (PG) mimetic, shows high potency and agonist efficacy at the IP receptor and has good bioavailability.Formula:C30H27NNaO4Purity:98%Color and Shape:SolidMolecular weight:488.539SDZ-216525
CAS:SDZ-216525, a 5-HT1A receptor antagonist, inhibits the tracheal contractions induced both by NKA (10 nM-3 microM) and 5-HT (10 nM-10 microM) (n=4-10).Formula:C25H28N4O5SColor and Shape:SolidMolecular weight:496.58Cipralisant maleate
CAS:Cipralisant maleate is a potent, selective Histamine H3 receptor antagonist.Formula:C18H24N2O4Color and Shape:SolidMolecular weight:332.39Epinephrine HCl
CAS:Epinephrine HCl is a hormone and neurotransmitter secreted by the adrenal medulla, agonist of α-adrenergic and β-adrenergic receptor.Formula:C9H14ClNO3Purity:99.48%Color and Shape:SolidMolecular weight:219.67RR-RJW100
RR-RJW100: potent LRH-1 & SF-1 agonist; studies metabolic disorders, diabetes, liver disease, IBD.Formula:C28H34OColor and Shape:SolidMolecular weight:386.57NVP-SAA164
CAS:NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.Formula:C36H45N5O5SPurity:98%Color and Shape:SolidMolecular weight:659.84PD 160170
CAS:neuropeptide Y1 receptor antagonistFormula:C18H17N3O4SPurity:98%Color and Shape:SolidMolecular weight:371.41
