GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 18 more subcategories

Found 5378 products of "GPCR/G-Protein"

Purity (%)

100

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Spiroglumide
CAS:
- 137795-35-8
Spiroglumide, a CCKB-gastrin antagonist that inhibits dose-dependent pentagastrin-induced acid hypersecretion with an ID50 of 20.1 (8.67-46.4) mg / kg, could be
Formula:C₂₁H₂₆Cl₂N₂O₄
Purity:98.23%
Color and Shape:Soild
Molecular weight:441.35
Ref: TM-T68016
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Survodutide TFA
Survodutide TFA (BI 456906 TFA) is a GCGR/GLP-1R dual agonist, a peptide compound used in obesity research.
Formula:C₁₉₂H₂₈₉N₄₇O₆₁·xC₂HF₃OC₂
Purity:99.29% - 99.96%
Color and Shape:Solid
Molecular weight:4231.62 (free base)
Ref: TM-T78098
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Human growth hormone-releasing factor
CAS:
- 83930-13-6
GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.
Formula:C₂₁₅H₃₅₈N₇₂O₆₆S
Purity:98%
Color and Shape:Solid
Molecular weight:5039.65
Ref: TM-TP1155
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Albenatide
CAS:
- 1031700-39-6
Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.
Formula:C₂₆H₄₇N₇O₉S
Purity:98%
Color and Shape:Solid
Molecular weight:633.76
Ref: TM-TP2368
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Lobeline sulfate
CAS:
- 134-64-5
Lobeline sulfate, an alkaloid like nicotine, aids in smoking cessation, insomnia, and respiratory issues. Less potent on nicotinic receptors.
Formula:C₂₂H₂₉NO₆S
Purity:98%
Color and Shape:White Powder
Molecular weight:435.54
Ref: TM-T22357
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Lisuride maleate
CAS:
- 19875-60-6
Lisuride maleate is a non-selective dopamine agonist and G-protein-biased 5-HT2A receptor agonist capable of blocking prolactin release.
Formula:C₂₄H₃₀N₄O₅
Purity:99.85%
Color and Shape:Solid
Molecular weight:454.52
Ref: TM-T8775
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SB 201146
CAS:
- 141311-11-7
SB 201146 is a leukotriene B4 antagonist with high affinity.
Formula:C₃₀H₃₅LiN₂O₅S
Color and Shape:Solid
Molecular weight:542.61
Ref: TM-T28667
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L-796,778
CAS:
- 217480-25-6
L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.
Formula:C₂₉H₄₀N₆O₇
Purity:96.20%
Color and Shape:Solid
Molecular weight:584.66
Ref: TM-T32511
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YM 16638
CAS:
- 104073-72-5
YM 16638 is an LT antagonist that can be used to study antigen-induced early and late airway responses in allergic sheep.
Formula:C₁₈H₂₂N₂O₅S₃
Purity:99.18%
Color and Shape:Solid
Molecular weight:442.57
Ref: TM-T35258
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LCKLSL acetate
LCKLSL acetate is a potent AnxA2 inhibitor, blocking tPA binding and plasmin production, with anti-angiogenic effects.
Formula:C₃₂H₆₁N₇O₁₀S
Purity:99.9%
Color and Shape:Solid
Molecular weight:735.93
Ref: TM-TP2482
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Parstatin(human)
CAS:
- 1065755-99-8
Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.
Formula:C₁₉₁H₃₃₀N₆₄O₅₃S₃
Purity:98%
Color and Shape:Solid
Molecular weight:4467.29
Ref: TM-TP1965
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Galantide acetate
Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P.
Formula:C₁₀₆H₁₅₅N₂₅O₂₈S
Purity:97.8% - 97.91%
Color and Shape:Solid
Molecular weight:2259.58
Ref: TM-T15368L
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WAY-620645
CAS:
- 742116-45-6
WAY-620645 is a CCK antagonist with antitumor and analgesic activities.
Formula:C₂₂H₂₂N₄O₂
Purity:99.89%
Color and Shape:Solid
Molecular weight:374.44
Ref: TM-T9991
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[D-Trp34]-Neuropeptide Y Acetate
[D-Trp34]-Neuropeptide Y Acetate is a potent Y5 receptor agonist that increases rat food intake; less potent at Y1, Y2, Y4, Y6.
Formula:C₁₉₈H₂₉₃N₅₅O₅₈
Purity:99.73%
Color and Shape:Soild
Molecular weight:4371.78
Ref: TM-TP1984L
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Neuropeptide S(Rat)
CAS:
- 412938-75-1
Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM).
Formula:C₉₅H₁₆₀N₃₄O₂₇
Purity:98%
Color and Shape:Solid
Molecular weight:2210.52
Ref: TM-TP1982
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CB2 receptor agonist 2
CAS:
- 1314230-75-5
CB2 receptor agonist 2 (ZINC72105556): potent, Ki=8.5 nM, high selectivity for CB2.
Formula:C₃₀H₃₆N₂O₄
Purity:99.75%
Color and Shape:Solid
Molecular weight:488.62
Ref: TM-T22009
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α-CGRP(human) TFA
α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as a
Formula:C₁₆₅H₂₆₈F₃N₅₁O₅₁S₂
Color and Shape:Solid
Molecular weight:3903.33
Ref: TM-T75788
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Neuropeptide Y (3-36) (human, rat)
CAS:
- 150138-78-6
Neuropeptide Y (3-36) is a Y2 receptor agonist that limits norepinephrine release, produced by DPP4 from NPY.
Formula:C₁₇₅H₂₆₉N₅₃O₅₄S
Color and Shape:Solid
Molecular weight:4011.5
Ref: TM-T36445
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Endothelin 1 (swine, human), Alexa Fluor 488-labeled
Synthetic human/swine Endothelin 1 peptide, tagged with Alexa Fluor 488, acts as a strong vasoconstrictor via ET A/B receptors.
Color and Shape:Solid
Molecular weight:2848.4
Ref: TM-T76081
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Amylin (IAPP), feline TFA
Amylin (IAPP), feline TFA: 37-amino acid peptide; inhibits insulin/glucagon; secreted by pancreatic β-cells.
Formula:C₁₆₇H₂₇₁F₃N₅₂O₅₆S₂
Color and Shape:Solid
Molecular weight:4024.47
Ref: TM-T76028