CymitQuimica logo
GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 18 more subcategories

Found 5378 products of "GPCR/G-Protein"

Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • CymitQuimica logo
    Targetmol
    + Info

    CCG258208 hydrochloride

    <p>GRKs-IN-1 HCl (14as) strongly inhibits GRK2 (IC50=130nM) &amp; GRK5 (IC50=7.1μM), is a paroxetine derivative with 100x cardiac boost.</p>
    Color and Shape:Solid

    Ref: TM-T35875

  • SHU 9119
    Targetmol
    + Info

    SHU 9119

    CAS:
    <p>SHU 9119 is a potent antagonist for human MC3R/MC4R and partial agonist for MC5R with IC50 values of 0.23, 0.06, 0.09 nM.</p>
    Formula:C54H71N15O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1074.258

    Ref: TM-T16879

  • L-803087 TFA
    Targetmol
    + Info

    L-803087 TFA

    CAS:
    <p>L-803087 TFA: potent sst4 agonist, Ki=0.7 nM, &gt;280x selective vs other somatostatin receptors; boosts AMPA, heightens seizures.</p>
    Formula:C27H30F5N5O5
    Color and Shape:Solid
    Molecular weight:599.55

    Ref: TM-T39207

  • Octodrine
    Targetmol
    + Info

    Octodrine

    CAS:
    <p>Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.</p>
    Formula:C8H19N
    Purity:99.98%
    Color and Shape:Clear Colorless To Light Yellow Liquid
    Molecular weight:129.24

    Ref: TM-T0043

  • 15(R)-17-phenyl trinor Prostaglandin F2α
    Targetmol
    + Info

    15(R)-17-phenyl trinor Prostaglandin F2α

    CAS:
    <p>17-phenyl trinor Prostaglandin F2α N-ethyl amide (17-phenyl trinor PGF2α) is an F-series prostaglandin analog which has been approved for use as an ocular</p>
    Formula:C23H32O5
    Color and Shape:Solid
    Molecular weight:388.5

    Ref: TM-T37930

  • RFRP-3(human)
    Targetmol
    + Info

    RFRP-3(human)

    CAS:
    <p>NPFF1 receptor agonist, IC50 0.7 nM, blocks cAMP by forskolin. A GnIH homolog, it inhibits GnRH neuron activity.</p>
    Formula:C45H72N14O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:969.15

    Ref: TM-TP1936

  • Semaglutide TFA
    Targetmol
    + Info

    Semaglutide TFA

    <p>Semaglutide TFA is a glucagon-like peptide-1 congener that induces weight loss, lowers blood glucose levels and reduces cardiovascular risk in diabetic patients</p>
    Formula:C189H290F3N45O61
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:4225.6482

    Ref: TM-T12878

  • EB1002
    Targetmol
    + Info

    EB1002

    CAS:
    <p>EB1002 is a selective NK2R agonist that has demonstrated significant enhancements in the expression levels of genes associated with mitochondrial biogenesis (such as PGC-1α) in obese mice. This suggests that EB1002 promotes energy expenditure by enhancing mitochondrial activity. Additionally, EB1002 has improved insulin sensitivity and glucose-lipid metabolism in mice. Therefore, EB1002 holds potential for research into obesity and type 2 diabetes.</p>
    Formula:C73H124N12O23
    Color and Shape:Solid
    Molecular weight:1537.83

    Ref: TM-T201621

  • Neurokinin Receptor (393-407), rat
    Targetmol
    + Info

    Neurokinin Receptor (393-407), rat

    CAS:
    <p>Rat NK1R fragment (393-407) binds SP, enabling endocytosis and plasma membrane recycling; key in neurogenic inflammation research.</p>
    Formula:C72H113N17O26S2
    Color and Shape:Solid
    Molecular weight:1696.9

    Ref: TM-T76429

  • CymitQuimica logo
    Targetmol
    + Info

    [His1,Nle27] GHRF (1-32), amide, human

    CAS:
    <p>[His1,Nle27] GHRF (1-32), amide, human is a potent GHRH analog with high GHRHR affinity.</p>
    Formula:C159H265N51O46
    Color and Shape:Solid
    Molecular weight:3627.12

    Ref: TM-T76317

  • ANP [Des18-22] 4-23 amide rat
    Targetmol
    + Info

    ANP [Des18-22] 4-23 amide rat

    CAS:
    <p>ANP [Des18-22] 4-23 amide rat is a peptide fragment of rat atrial natriuretic peptide (ANP) that specifically binds to NPR-C.</p>
    Formula:C64H107N25O19S2
    Color and Shape:Solid
    Molecular weight:1594.82

    Ref: TM-TP3030

  • CymitQuimica logo
    Targetmol
    + Info

    Selepressin acetate

    <p>Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.</p>
    Formula:C48H77N13O13S2
    Color and Shape:Solid
    Molecular weight:1108.33

    Ref: TM-T73654

  • [Ala2] Endothelin-3, human
    Targetmol
    + Info

    [Ala2] Endothelin-3, human

    CAS:
    <p>[Ala2] Endothelin-3, a linear ET-3 analog with Ala replacing Cys, stimulates endothelial cell migration.</p>
    Formula:C120H166N26O32S4
    Color and Shape:Solid
    Molecular weight:2613.02

    Ref: TM-T76305

  • Dotanoc
    Targetmol
    + Info

    Dotanoc

    CAS:
    <p>Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.</p>
    Formula:C69H94N14O17S2
    Color and Shape:Solid
    Molecular weight:1455.71

    Ref: TM-T24014

  • Gastrin I, rat
    Targetmol
    + Info

    Gastrin I, rat

    CAS:
    <p>Gastrin I, rat is a peptide hormone that effectively stimulates gastric acid secretion.</p>
    Formula:C94H128N22O31S2
    Color and Shape:Solid
    Molecular weight:2126.3

    Ref: TM-T38203

  • CymitQuimica logo
    Targetmol
    + Info

    Neuropeptide Y (3-36) (porcine)

    CAS:
    <p>Neuropeptide Y (3-36) (porcine) is a potent, selective agonist at NPY Y2 receptors, increasing feeding in rats.</p>
    Formula:C176H271N53O54
    Color and Shape:Solid
    Molecular weight:3993.36

    Ref: TM-T76355

  • CymitQuimica logo
    Targetmol
    + Info

    TAK-683 acetate

    <p>TAK-683 acetate: potent KISS1R agonist (IC50=170 pM), stable, nonapeptide. Affects GnRH, FSH, LH, testosterone; potential in prostate cancer research.</p>
    Formula:C66H87N17O15
    Color and Shape:Solid
    Molecular weight:1358.5

    Ref: TM-T76048

  • CymitQuimica logo
    Targetmol
    + Info

    Baloncibart

    CAS:
    <p>Baloncibart is a human IgG4K monoclonal antibody that targets NPR1.</p>
    Color and Shape:Liquid

    Ref: TM-T9901A-888

  • Acetyl-Amylin (8-37) (human)
    Targetmol
    + Info

    Acetyl-Amylin (8-37) (human)

    CAS:
    <p>Acetyl-Amylin (8-37) (human) is a specific amylin antagonist [1] .</p>
    Formula:C140H218N42O46
    Color and Shape:Solid
    Molecular weight:3225.48

    Ref: TM-T76645

  • CymitQuimica logo
    Targetmol
    + Info

    Human glucagon-like peptide-1-(7-36)-Lys(Biotin) amide

    <p>Biotin-labeled GLP-1-(7-36) amide; a gut peptide that enhances insulin release.</p>
    Formula:C165H252N44O48S
    Color and Shape:Solid
    Molecular weight:3652.1

    Ref: TM-T76330