
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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Conessine hydrobromide
CAS:<p>Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.</p>Formula:C24H41BrN2Color and Shape:SolidMolecular weight:437.51α-CGRP (mouse, rat) TFA
<p>α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions and</p>Formula:C162H262N50O52S2·C2HF3O2Purity:98%Color and Shape:Solid5-methoxy-α-Ethyltryptamine
CAS:<p>5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects. </p>Formula:C13H18N2OPurity:98.25%Color and Shape:SolidMolecular weight:218.29HTR2A antagonist 1
<p>HTR2A antagonist 1 (Compound 15f) is an HTR2A antagonist with an IC50 of 42.79 nM. It induces sub-G1 cell cycle arrest and apoptosis in colorectal cancer cells by activating the p53/p21/caspase 3 signaling pathway. HTR2A antagonist 1 exhibits good liver microsomal stability and is useful for colorectal cancer research.</p>Formula:C35H43Cl2F2N5O4Color and Shape:SolidMolecular weight:706.65Tamuzimod
CAS:<p>Tamuzimod, an effective immunomodulator, exhibits modulatory activity on S1P Receptors with EC50 values below 1 μM [1] [2].</p>Formula:C21H13Cl3F3N5O3Color and Shape:SolidMolecular weight:546.71Sarafotoxin S6a
CAS:Endothelin receptor agonist (EC50 values are 7.5 and > 150 nM for contraction of pig coronary artery and guinea pig aorta respectively). Nociceptive in vivo.Formula:C105H156N28O34S5Purity:98%Color and Shape:SolidMolecular weight:2514.85CGRP antagonist 6
<p>CGRP Antagonist 6 (Compound 23) is a potent CGRP receptor antagonist (Ki: 0.84 nM). It is utilized in the study of migraines.</p>Color and Shape:Odour SolidHTL22562
CAS:<p>HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.</p>Formula:C40H49N11O5Color and Shape:SolidMolecular weight:763.904Mosliciguat
CAS:<p>Mosliciguat is a guanylate cyclase activator.</p>Formula:C41H36ClF3N2O5Color and Shape:SolidMolecular weight:729.19RXFP3/4 agonist 1
CAS:<p>RXFP3/4 agonist 1 is a relaxin family peptide 3/4 receptor (RXFP3/4) agonist(EC50s of 82/2 nM, respectivley).</p>Formula:C20H22ClN5OPurity:98%Color and Shape:SolidMolecular weight:383.88Fasitibant chloride
CAS:<p>Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.</p>Formula:C36H49Cl3N6O6SColor and Shape:SolidMolecular weight:800.23Tezusomant
CAS:Tezusomant is an antagonist of the growth hormone receptor (growth hormone receptor). It is being investigated for potential use in conditions like acromegaly, which are caused by excessive secretion of growth hormone.Formula:C120H171N23O32SColor and Shape:SolidMolecular weight:2479.84Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:<p>Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.</p>Formula:C47H66N12O11Purity:98%Color and Shape:SolidMolecular weight:975.11Methdilazine
CAS:<p>Methdilazine: oral antibiotic, histamine antagonist, fights mycobacterium (MIC 5-15 μg/mL) for infectious disease research.</p>Formula:C18H20N2SColor and Shape:SolidMolecular weight:296.43Maceneolignan H
CAS:<p>Maceneolignan H, a neolignane from Myristica fragrans, selectively blocks CCR3 (EC50=1.4μM) with allergy research potential.</p>Formula:C24H30O7Color and Shape:SolidMolecular weight:430.49Zicronapine fumarate
CAS:<p>Zicronapine fumarate, an antipsychotic, targets D1/D2 & 5-HT2A receptors; may treat neuropsychiatric conditions.</p>Formula:C26H31ClN2O4Color and Shape:SolidMolecular weight:470.99Ghrelin receptor full agonist-2
CAS:<p>Ghrelin receptor full agonist-2 is a highly potent Ghrelin receptor full agonist.</p>Formula:C26H28ClN5O5SColor and Shape:SolidMolecular weight:558.05Neuropeptide Y (human)
CAS:<p>Neuropeptide Y (29-64), amide, human is a biologically active 36-amino acid peptide.</p>Formula:C189H285N55O57SPurity:98%Color and Shape:SolidMolecular weight:4271.68Cloprostenol isopropyl ester
CAS:<p>(+)-Chloprostol is a PGF2α agonist, mimics prostaglandin F2α, induces luteal dissolution in mares without side effects or stress.</p>Formula:C25H35ClO6Color and Shape:SolidMolecular weight:466.99Seglitide
CAS:<p>Peptide agonist targets sst2/sst5 receptors. IC50/Kd: sst1 >1000, sst2 = 0.2-1.5, sst3 = 27-36, sst4 >127, sst5 = 0.06-23 nM.</p>Formula:C44H56N8O7Purity:98%Color and Shape:SolidMolecular weight:808.98

