GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 18 more subcategories

Found 5378 products of "GPCR/G-Protein"

Purity (%)

100

products per page.

+ Info
α-helical CRF 9-41 acetate
α-helical CRF 9-41 acetate is a competitive antagonist of CRF2 (KB = 100 nM) and a partial agonist of CRF1 (EC50 = 140 nM).
Purity:96.60%
Color and Shape:Solid
Molecular weight:#N/A
Ref: TM-TP2048L
+ Info
Ghrelin receptor full agonist-2
CAS:
- 2602452-73-1
Ghrelin receptor full agonist-2 is a highly potent Ghrelin receptor full agonist.
Formula:C₂₆H₂₈ClN₅O₅S
Color and Shape:Solid
Molecular weight:558.05
Ref: TM-T40234
+ Info
Melanostatin, frog TFA
Melanostatin, frog TFA is an α-MSH release inhibitor, a 36 amino acid peptide isolated from the frog brain.
Purity:99.23%
Color and Shape:Odour Solid
Ref: TM-TP2603L
+ Info
ELA-11(human)
CAS:
- 1784687-32-6
Apelin receptor agonist with high affinity (Ki = 14 nM). Blocks cAMP production and promotes β-arrestin activation; derived from ELA-32.
Formula:C₅₈H₉₀N₁₆O₁₃S₂
Purity:98%
Color and Shape:Solid
Molecular weight:1283.57
Ref: TM-TP1922
+ Info
ARL 15849XX
CAS:
- 152548-39-5
ARL 15849XX, a CCK-8 analog, is a novel anti-obesity agent.
Formula:C₄₇H₆₀N₈O₁₃S
Purity:98%
Color and Shape:Solid
Molecular weight:977.09
Ref: TM-T25108
+ Info
Satoreotide
CAS:
- 1801415-23-5
Satoreotide (JR11) is an SSTR2 antagonist, typically conjugated with radiolabeled chelators for use in neuroendocrine tumor imaging [1].
Formula:C₅₈H₇₂ClN₁₅O₁₄S₂
Color and Shape:Solid
Molecular weight:1302.87
Ref: TM-TP2620
+ Info
Dexbrompheniramine
CAS:
- 132-21-8
Dexbrompheniramine: oral H1 antagonist, antihistamine for hay fever and urticaria research.
Formula:C₁₆H₁₉BrN₂
Color and Shape:Solid
Molecular weight:319.24
Ref: TM-T75276
+ Info
LMN-NKA acetate
LMN-NKA acetate is a modified Neurokinin A (4-10) and selective NK2R (Neurokinin 2 receptor) agonist induces bladder contraction smooth muscle contraction.
Formula:C₄₁H₆₈N₈O₁₂
Color and Shape:Solid
Molecular weight:865.03
Ref: TM-T76426L
+ Info
Nadolol
CAS:
- 42200-33-9
Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities.
Formula:C₁₇H₂₇NO₄
Purity:99.87% - 99.92%
Color and Shape:White To Off-White Crystalline Powder Solid
Molecular weight:309.40
Ref: TM-T1203
+ Info
15(S)-15-methyl Prostaglandin D2
CAS:
- 85280-90-6
15(S)-15-methyl PGD2 is a stable PGD2 analog that induces vasoconstriction, raises blood pressure, and shows strong antifertility effects.
Formula:C₂₁H₃₄O₅
Color and Shape:Solid
Molecular weight:366.49
Ref: TM-T36153
+ Info
OXA(17-33) TFA
OXA(17-33) TFA: Potent OX1 agonist, ~23x more selective for OX1 (EC50=8.29nM) than OX2 (187nM).
Formula:C₈₁H₁₂₆F₃N₂₃O₂₄
Color and Shape:Solid
Molecular weight:1863
Ref: TM-T75922
+ Info
MRS2500 tetraammonium
CAS:
- 630103-23-0
Highly potent and selective antagonist of the platelet P2Y1 receptor
Formula:C₁₃H₂₁IN₆O₈P₂
Purity:98%
Color and Shape:Solid
Molecular weight:578.19
Ref: TM-T23023
+ Info
[Asu1,6-Arg8]Vasopressin
CAS:
- 40944-53-4
[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.
Formula:C₄₈H₆₈N₁₄O₁₂
Color and Shape:Solid
Molecular weight:1033.14
Ref: TM-T76510
+ Info
Cyclic SSTR agonist octreotide
Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .
Formula:C₅₃H₇₁N₁₁O₁₄S₂
Color and Shape:Solid
Molecular weight:1150.33
Ref: TM-T76544
+ Info
Melanostatin, frog
CAS:
- 134709-16-3
Melanostatin, frog, is an inhibitor of α-melanocyte-stimulating hormone (α-MSH) release, with an IC50 of 60 nM [1] [2].
Formula:C₁₈₉H₂₈₅N₅₃O₅₇S
Color and Shape:Solid
Molecular weight:4243.67
Ref: TM-TP2603
+ Info
Israpafant
CAS:
- 117279-73-9
Israpafant: PAF receptor blocker, IC50 0.84nM, hinders platelet aggregation, eosinophil activation, boosts calcium transit, anti-nephrotoxic.
Formula:C₂₈H₂₉ClN₄S
Color and Shape:Solid
Molecular weight:489.07
Ref: TM-T27638
+ Info
Bradykinin (1-6)
CAS:
- 23815-88-5
Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.
Formula:C₃₀H₄₅N₉O₈
Purity:98%
Color and Shape:Solid
Molecular weight:659.73
Ref: TM-TP1747
+ Info
Pasireotide
CAS:
- 396091-73-9
Pasireotide (SOM 230) is a cyclohexapeptide, mimicking somatostatin with high affinity for sst1/2/3/4/5 receptors (pKi=8.2/9.0/9.1/<7.0/9.9).
Formula:C₅₈H₆₆N₁₀O₉
Purity:98%
Color and Shape:Solid
Molecular weight:1047.21
Ref: TM-T12370
+ Info
Semaglutide, FITC labeled
Semaglutide (FITC-labeled Semaglutide) is a long-acting analog of human glucagon-like peptide-1, functioning as an agonist of the GLP-1 receptor. It shows potential for research related to type 2 diabetes.
Formula:C₂₀₉H₃₀₄N₄₆O₆₃S
Molecular weight:4498.17191
Ref: TM-TP3655
+ Info
GLP-1(7-37)
CAS:
- 106612-94-6
GLP-1 (7-37) is a truncated, bioactive form of GLP-1 that is the product of proglucagon processing in intestinal endocrine L cells.
Formula:C₁₅₁H₂₂₈N₄₀O₄₇
Purity:98%
Color and Shape:Solid
Molecular weight:3355.67
Ref: TM-TP1306