GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(53 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5980 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
MrgprX2 antagonist-2
CAS:MrgprX2 antagonist-2, from patent WO2021092262A1 E163, is potent for skin inflammation studies.Formula:C17H16F5N3O3Color and Shape:SolidMolecular weight:405.325Cetirizine Impurity D
CAS:Cetirizine Impurity D, an antihistamine derivative, acts as a long-lasting H1-receptor antagonist with antiallergic effects.Formula:C30H28Cl2N2Color and Shape:SolidMolecular weight:487.46AMTG-DA1
AMTG-DA1 is a ligand for the gastrin-releasing peptide receptor (GRPR), and it can be utilized in cancer research.Formula:C101H149IN22O25Color and Shape:SolidMolecular weight:2197.0109Cortistatin-8 acetate
<p>Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.</p>Formula:C49H72N12O11S2Purity:99.01%Color and Shape:SoildMolecular weight:1069.3Ref: TM-TP2236L
1mg229.00€5mg560.00€10mg800.00€25mg1,216.00€50mg1,644.00€100mg2,213.00€500mg4,436.00€VIP36
VIP36 is an agonist of the cannabinoid type 1 receptor (CB1) with analgesic properties. It reduces the recruitment of inhibitory proteins, thereby exerting its pain-relieving effects, and is applicable in research related to chronic pain.Formula:C27H35FN6O4Color and Shape:SolidMolecular weight:526.60312-epi Leukotriene B4
CAS:LTB4 is made enzymatically (12(R)-specific) and non-enzymatically (6-trans-12-epi mix). 12-epi LTB4 has low receptor activity.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.472TRPV1/CB2 agonist 1
<p>TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.</p>Color and Shape:Odour SolidSRA880 malonate
CAS:SRA880: non-peptide sst(1) antagonist, low affinity for other sst receptors, binds dopamine D4, boosts SRIF, antidepressant-like effects.Formula:C29H36N4O8Purity:98%Color and Shape:SolidMolecular weight:568.62(R,R)-Palonosetron Hydrochloride
CAS:(R,R)-Palonosetron Hydrochloride is the active enantiomer of PalonosetronFormula:C19H25ClN2OPurity:98%Color and Shape:SolidMolecular weight:332.87Senktide TFA
Senktide TFA is a potent and selective neurokinin 3 (NK3) receptor agonist with an EC50 of 0.5-3 nM, while showing significantly weaker activity on NK1 receptors (EC50=35 µM). It is a promising candidate for research in neurological disorders.Color and Shape:Odour SolidSSTR4 agonist-1
CAS:SSTR4agonist-1 (Compound 47) is a selective agonist of the somatostatin receptor 4 (SSTR4), with an EC50 of 4.7 nM. It has a half-life of over 130 minutes in human liver microsomes.Formula:C16H23N3O2Color and Shape:SolidMolecular weight:289.37Meluadrine tartrate
CAS:Meluadrine tartrate is an endogenous metabolite.Formula:C16H24ClNO8Purity:98%Color and Shape:SolidMolecular weight:393.82PHM-27 (human)
CAS:<p>Human-derived peptide, VIP/PHM 27 analog, boosts insulin by targeting calcitonin receptor with an EC50 of 11 nM.</p>Formula:C135H214N34O40SPurity:98%Color and Shape:SolidMolecular weight:2985.44Atrial natriuretic factor (1-28) (rat) TFA
ANP (1-28), rat (TFA) inhibits Ang II-induced endothelin-1 secretion; main circulating ANP form in rats.Formula:C130H206N45F3O41S2Purity:98%Color and Shape:SolidMolecular weight:3176.43Cetirizine D8 dihydrochloride
CAS:Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.Formula:C21H26Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:433.4Anthramycin
CAS:Anthramycin: a PBD family antibiotic with antitumor effects and CNS cholecystokinin antagonist properties in mice.Formula:C16H17N3O4Color and Shape:SolidMolecular weight:315.32Albenatide
CAS:<p>Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.</p>Formula:C26H47N7O9SPurity:98%Color and Shape:SolidMolecular weight:633.76NPC 567
CAS:NPC 567 is an antagonist of the bradykinin receptor.Formula:C60H87N19O13Purity:98%Color and Shape:SolidMolecular weight:1282.48L-threo Lysosphingomyelin (d18:1)
CAS:L-threo Lysosphingomyelin, a natural S1P receptor agonist, has EC50s: 19.3 nM (hS1P1), 131.8 nM (hS1P3), 313.3 nM (hS1P2).Formula:C23H49N2O5PColor and Shape:SolidMolecular weight:464.62Haloperidol D4
CAS:<p>Haloperidol D4 is deuterium-labeled haloperidol.</p>Formula:C21H23ClFNO2Purity:98%Color and Shape:SolidMolecular weight:379.89
