GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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S1R agonist 2
CAS:S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for S2R and 1.1 nM for S1R and is protective against ROS and NMDA-induced neurotoxicity.Formula:C21H27NOPurity:99.66%Color and Shape:SolidMolecular weight:309.45Fpl 14294
CAS:Fpl 14294 is a novel CCK-8 agonist with effective intranasal anorectic activity in the rat.Formula:C45H56N8O13S3Purity:98%Color and Shape:SolidMolecular weight:1013.17NI-203
NI-203 is a monoclonal antibody inhibitor that targets amylin and shows potential for research in type 2 diabetes.Color and Shape:Odour Liquid5-HT2A receptor agonist-6
CAS:5-HT2A receptor agonist-6 (compound 47) is a selective agonist of the 5-HT2A receptor with a pEC50 value of 6.58.Formula:C18H19N3O3Color and Shape:SolidMolecular weight:325.36MM 07
CAS:Biased agonist for apelin/G protein pathway, enhances eNOS and cell growth, reduces apoptosis, improves heart function, and dilates vessels.Formula:C67H106N22O14S3Purity:98%Color and Shape:SolidMolecular weight:1539.9Ularitide
CAS:Ularitide is a 32-amino acid peptide from ANP prohormone, resistant to dog kidney cortex peptidase.Formula:C145H234N52O44S3Purity:98%Color and Shape:SolidMolecular weight:3505.97Eledoisin Related Peptide
CAS:Eledoisin Related Peptide (Eledoisin RP) is a tachykinin receptor ligand.Formula:C34H58N8O6SPurity:98%Color and Shape:SolidMolecular weight:706.94HPP-9
HPP-9, a Proteolysis-Targeting Chimera (PROTAC) derived from Hedgehog Pathway Inhibitor-1 (HPI-1) with a pIC50 value of 6.71, is designed to degrade BETFormula:C49H52N6O11Color and Shape:SolidMolecular weight:900.97ONO-0300302
CAS:ONO-0300302: LPA1 antagonist, treats Benign Prostatic Hyperplasia, IC50 = 0.16 nM, reduces IUP in rats and dogs for 12h.Formula:C29H35NO5Purity:98%Color and Shape:SolidMolecular weight:477.59GR 82334
CAS:Tachykinin NK1 receptor antagonist.Formula:C69H91N15O16Purity:98%Color and Shape:SolidMolecular weight:1386.57Azaline
CAS:Azaline is a gonadorelin antagonist.Formula:C74H106ClN23O12Purity:98%Color and Shape:SolidMolecular weight:1545.26CB2R/FAAH modulator-2
CAS:CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH.Formula:C24H33NO2Purity:99.15%Color and Shape:SoildMolecular weight:367.52Mirtazapine N-oxide
CAS:Mirtazapine N-oxide, a mirtazapine metabolite, is produced by CYP1A2 and CYP3A4 in human liver.Formula:C17H19N3OColor and Shape:SolidMolecular weight:281.359[Lys4] Sarafotoxin S6c
CAS:[Lys4] Sarafotoxin S6c: potent partial endothelin receptor agonist; causes pig coronary contraction, EC50=1.5 nM.Formula:C105H153N27O36S5Color and Shape:SolidMolecular weight:2529.82GRK2i
CAS:GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. Corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.Formula:C153H256N50O41SPurity:98%Color and Shape:SolidMolecular weight:3484.08Mitemcinal fumarate
CAS:Mitemcinal fumarate is a erythromycin derivative that is used to treat gastroesophageal reflux disease.
Formula:C84H142N2O28Color and Shape:SolidMolecular weight:1628.02Neuronostatin-13 (human)
CAS:Neuronostatin-13: human-conserved, 13-amino-acid peptide with amidated C-terminus.Formula:C64H110N20O16Purity:98%Color and Shape:SolidMolecular weight:1415.68LHRH
CAS:Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and hasFormula:C55H74N16O14Purity:98%Color and Shape:SolidMolecular weight:1183.27AC-178335
CAS:AC-178335: SRIF antagonist, Ki=172 nM, inhibits SRIF's adenylate cyclase effects (IC50=5.1 µM), triggers GH release in rats.Formula:C49H63N13O7Color and Shape:SolidMolecular weight:946.11[Tyr11]-Somatostatin
CAS:[Tyr11]-Somatostatin, a neuroactive peptide, aids proteomics research and modulates retinal function.Formula:C76H104N18O20S2Color and Shape:SolidMolecular weight:1653.89
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