GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,997 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5957 products of "GPCR/G-Protein"
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Casopitant
CAS:Casopitant (GW679769) is an orally active neurokinin-1 (NK1) receptor antagonist, researched for its potential use in managing chemotherapy-induced nausea and vomiting (CINV) and postoperative nausea and vomiting (PONV).Formula:C30H35F7N4O2Color and Shape:SolidMolecular weight:616.61Cisapride hydrate
CAS:Cisapride acts directly as a selective agonist of serotonin 5-HT4 receptor with IC50 value of 0.483 μM. And It also acts indirectly as a parasympathomimetic.Formula:C23H31ClFN3O5Purity:98%Color and Shape:SolidMolecular weight:483.96Kisspeptin-10, human
CAS:Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.Formula:C63H83N17O14Purity:98%Color and Shape:SolidMolecular weight:1302.462SAG dihydrochloride
CAS:SAG dihydrochloride: potent Smo agonist, activates Hedgehog pathway, counters Cyclopamine. EC50=3 nM, Kd=59 nM.Formula:C28H30Cl3N3OSPurity:99.57%Color and Shape:SoildMolecular weight:562.988β-Hydroxy-exo-THC
CAS:8β-Hydroxy-exo-THC, a cannabinoid ether analog, exhibits weak affinity for receptor sites with an IC50 of 1.2 μM.Formula:C21H30O3Color and Shape:SolidMolecular weight:330.46Mosliciguat
CAS:Mosliciguat is a guanylate cyclase activator.Formula:C41H36ClF3N2O5Color and Shape:SolidMolecular weight:729.1913,14-dihydro-15-keto Prostaglandin F1α
CAS:13,14-dihydro-15-keto Prostaglandin F1α (13,14-dihydro-15-keto PGF1α) is a metabolite of PGF1α that has been reported in the rat stomach.Formula:C20H36O5Color and Shape:SolidMolecular weight:356.5TGR5 agonist 2
TGR5 agonist 2 (compound 19) serves as a highly potent agonist of TGR5, demonstrating an EC50 value of 0.27 µM [1].Formula:C29H50NNaO6SColor and Shape:SolidMolecular weight:563.77Imnopitant dihydrochloride
CAS:Imnopitant dihydrochloride is a neurokinin NK1 receptor antagonist [1] .Formula:C28H30Cl2F6N4OColor and Shape:SolidMolecular weight:623.46Methdilazine
CAS:Methdilazine: oral antibiotic, histamine antagonist, fights mycobacterium (MIC 5-15 μg/mL) for infectious disease research.Formula:C18H20N2SColor and Shape:SolidMolecular weight:296.43LY 293284
CAS:LY 293284 is a potent, selective full agonist of 5-HT1A receptor with anxiogenic effects in animal studies.Formula:C19H26N2OColor and Shape:SolidMolecular weight:298.42PACAP (6-38), human, ovine, rat
CAS:PACAP (6-38) in humans, sheep, rats: a strong inhibitor of PACAP 38, outperforms PACAP (6-27) in blocking PACAP-27-induced adenylate cyclase.Formula:C182H300N56O45SPurity:98%Color and Shape:SolidMolecular weight:4024.74Lys-γ3-MSH(human)
CAS:Pro-opiomelanocortin (POMC) derived peptide that stimulates lipolysisFormula:C128H193N45O39SPurity:98%Color and Shape:SolidMolecular weight:3018.25MEN 11270
CAS:B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.Formula:C60H90N20O11SPurity:98%Color and Shape:SolidMolecular weight:1299.56Linzagolix choline
CAS:Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.Formula:C27H28F3N3O8SPurity:99.64%Color and Shape:SolidMolecular weight:611.59α-CGRP(human)
CAS:Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.Formula:C163H267N51O49S2Purity:98%Color and Shape:SolidMolecular weight:3789.33Obestatin(rat)
CAS:Endogenous peptide that suppresses food intake and body weight-gainFormula:C114H174N34O31Purity:98%Color and Shape:SolidMolecular weight:2516.81GLP-1 receptor agonist 9 citrate
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
Formula:C38H39ClFN3O12Purity:98.76%Color and Shape:SolidMolecular weight:784.18Dexbrompheniramine
CAS:Dexbrompheniramine: oral H1 antagonist, antihistamine for hay fever and urticaria research.Formula:C16H19BrN2Color and Shape:SolidMolecular weight:319.24CCR4 antagonist 3 hydrochloride
CAS:Orally active CCR4 antagonist 3 hydrochloride with potent selectivity, IC50s: 22/50 nM; has antitumor properties.Formula:C24H27Cl2N7O·xHClColor and Shape:Solid
