GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,997 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5957 products of "GPCR/G-Protein"
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ANP [Des18-22] 4-23 amide rat
CAS:ANP [Des18-22] 4-23 amide rat is a peptide fragment of rat atrial natriuretic peptide (ANP) that specifically binds to NPR-C.
Formula:C64H107N25O19S2Color and Shape:SolidMolecular weight:1594.82Selepressin acetate
Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.Formula:C48H77N13O13S2Color and Shape:SolidMolecular weight:1108.33[Ala2] Endothelin-3, human
CAS:[Ala2] Endothelin-3, a linear ET-3 analog with Ala replacing Cys, stimulates endothelial cell migration.Formula:C120H166N26O32S4Color and Shape:SolidMolecular weight:2613.02Dotanoc
CAS:Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.Formula:C69H94N14O17S2Color and Shape:SolidMolecular weight:1455.71Gastrin I, rat
CAS:Gastrin I, rat is a peptide hormone that effectively stimulates gastric acid secretion.Formula:C94H128N22O31S2Color and Shape:SolidMolecular weight:2126.3Protease-Activated Receptor-1, PAR-1 Agonist TFA
PAR-1 Agonist TFA: Selective peptide, mimics thrombin, activates PAR-1 receptor.Color and Shape:Liquid15-keto Latanoprost
CAS:Latanoprost, a PG analog for ocular pressure, metabolizes into 15-keto latanoprost, a less potent variant reducing intraocular pressure and pupil size.Formula:C26H38O5Color and Shape:SolidMolecular weight:430.58(Trp7,β-Ala8)-Neurokinin A (4-10)
CAS:(Trp7,β-Ala8)-Neurokinin A (4-10) is a potent neurokinin-3 (NK3) antagonist [1] .Formula:C41H57N9O10SColor and Shape:SolidMolecular weight:868.01MDL 29913
CAS:NK2 tachykinin receptor selective antagonist.Formula:C40H56N8O6Purity:98%Color and Shape:SolidMolecular weight:745Vatinoxan
CAS:Vatinoxan is a peripheral α2 adrenoreceptor antagonist.Formula:C20H26N4O4SPurity:98%Color and Shape:SolidMolecular weight:418.51Prepro-ANF (56-92), human
CAS:Human prepro-ANF (56-92) activates renal guanylate cyclase and boosts its activity.Formula:C173H270N44O57Color and Shape:SolidMolecular weight:3878.26Cyclosomatostatin TFA
Cyclosomatostatin TFA blocks SST receptor, reduces CRC cell growth, ALDH+ size, and sphere-formation.Formula:C46H58F3N7O8Color and Shape:SolidMolecular weight:893.99BMS-604992 free base
CAS:BMS-604992 (EX-1314), a selective GHSR agonist, binds strongly (ki=2.3 nM), is orally active, and increases rodent food intake.Formula:C24H31N7O5Color and Shape:SolidMolecular weight:497.556ARC 239 dihydrochloride
CAS:ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).Formula:C24H31Cl2N3O3Purity:99.72%Color and Shape:SolidMolecular weight:480.43Conessine hydrobromide
CAS:Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.Formula:C24H41BrN2Color and Shape:SolidMolecular weight:437.51[Des-His1,Glu9]-Glucagon amide
CAS:Glucagon blocker with pA2 of 7.2; no agonist effect. Boosts insulin; prevents glucagon-driven hyperglycemia in rabbits and diabetic rats.Formula:C148H221N41O47SPurity:98%Color and Shape:SolidMolecular weight:3358.68Bombinakinin M
CAS:Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.Formula:C100H159N31O24Purity:98%Color and Shape:SolidMolecular weight:2179.55Luseogliflozin
CAS:Luseogliflozin inhibits SGLT2 for glucose uptake with 1.10 nM potency.Formula:C23H30O6SColor and Shape:SolidMolecular weight:434.55CCR4 antagonist 3
CAS:Orally active CCR4 antagonist with piperidinyl-azetidine; IC50: 22 nM (calcium flux), 50 nM (CTX); antitumor effects.Formula:C24H27Cl2N7OColor and Shape:SolidMolecular weight:500.43Sauvagine TFA
Sauvagine TFA: frog-derived, 40-amino-acid CRF agonist; stimulates ACTH release, affects diuresis, cardiovascular system, endocrine glands.Formula:C204H347F3N56O65S1Color and Shape:SolidMolecular weight:4713.33
![ANP [Des18-22] 4-23 amide rat](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP3030.webp&w=3840&q=75)
![[Ala2] Endothelin-3, human](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76305.webp&w=3840&q=75)
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