GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,995 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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ELA-21 (human)
CAS:Apelin receptor agonist with high affinity for normal/PAH hearts (pKi 9.31/9.46). Blocks cAMP, promotes β-arrestin in vitro. Part of ELA-32.Formula:C112H184N40O25S3Purity:98%Color and Shape:SolidMolecular weight:2587.12Phenylethanolamine A
CAS:Phenylethanolamine A is a β-adrenergic agonist and a byproduct of the Ractopamine synthesis process.Formula:C19H24N2O4Color and Shape:SolidMolecular weight:344.40RF9 acetate
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.Formula:C28H42N6O5Purity:99.77%Color and Shape:SolidMolecular weight:542.67Ref: TM-T16738L
1mg65.00€5mg125.00€10mg182.00€25mg325.00€50mg467.00€100mg645.00€200mg868.00€1mL*10mM (DMSO)167.00€Hydroxybupropion
CAS:Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).Formula:C13H18ClNO2Purity:99.73%Color and Shape:Off-White SolidMolecular weight:255.74Ref: TM-T11588
1mg89.00€5mg204.00€10mg331.00€25mg545.00€50mg777.00€100mg1,063.00€1mL*10mM (DMSO)232.00€Lisuride maleate
CAS:Lisuride maleate is a non-selective dopamine agonist and G-protein-biased 5-HT2A receptor agonist capable of blocking prolactin release.Formula:C24H30N4O5Purity:99.85%Color and Shape:SolidMolecular weight:454.52Ref: TM-T8775
1mg204.00€5mg627.00€10mg898.00€25mg1,346.00€50mg1,745.00€100mg2,382.00€1mL*10mM (DMSO)627.00€[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
CAS:Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.Formula:C50H75N15O10Purity:98%Color and Shape:SolidMolecular weight:1046.2311-deoxy Prostaglandin E1
CAS:11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and causeFormula:C20H34O4Color and Shape:SolidMolecular weight:338.48Spantide acetate
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.
Formula:C77H112N20O15Purity:98.9200%Color and Shape:SolidMolecular weight:1557.84PEN (human)
CAS:PEN (human) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.Formula:C97H159N27O32Purity:98%Color and Shape:SolidMolecular weight:2215.49Navafenterol saccharinate
CAS:AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).Formula:C45H47N7O9S3Color and Shape:SolidMolecular weight:926.09MK-7246 S enantiomer
MK-7246 S enantiomer is a potent and selective CRTH2 antagonist.Formula:C21H21FN2O4SPurity:98%Color and Shape:SolidMolecular weight:416.47Sch 202596
CAS:Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.Formula:C25H22Cl2O12Color and Shape:SolidMolecular weight:585.34P2Y6R antagonist 1
P2Y6R antagonist 1 (compound 5ab) is a selective, orally active antagonist of P2Y6R, featuring an IC50 value of 19.6 nM. This compound also exhibits anti-inflammatory properties.Color and Shape:Odour SolidGLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Formula:C165H254N44O55SPurity:98%Color and Shape:SolidMolecular weight:3766.19NESS 0327
CAS:NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.Formula:C24H23Cl3N4OPurity:99.78%Color and Shape:SolidMolecular weight:489.82SB234551
CAS:SB234551 is a selective antagonist of endothelin ETA receptor.Formula:C34H34N2O9Color and Shape:SolidMolecular weight:614.645-HT7R antagonist 1 free base
CAS:5-HT7R antagonist 1 (free base) is a G protein-biased antagonist for the 5-HT 7 R receptor, with a dissociation constant (K i) of 6.5 nM.Formula:C14H17ClN4Color and Shape:SolidMolecular weight:276.77K-(D-1-Nal)-FwLL-NH2
CAS:Potent ghrelin receptor inverse agonist with Ki of 4.9/31 nM in COS7/HEK293T; blocks Gq/G13 signaling.Formula:C51H67N9O6Purity:98%Color and Shape:SolidMolecular weight:902.13Dulaglutide
CAS:Dulaglutide (LY2189265) is a GLP-1 receptor agonist for studying type 2 diabetes mellitus (T2DM).Color and Shape:SolidSpns2-IN-2
Spns2-IN-2 (compound 3a) is an inhibitor of SPNS2.Formula:C22H30ClN3O2Color and Shape:SolidMolecular weight:403.95
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