GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5964 products of "GPCR/G-Protein"
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[Nle11]-Substance P
CAS:'[Nle11]-Substance P is a gut and brain peptide, resisting methionine oxidation and causing excitatory neural effects.'
Formula:C64H100N18O13Purity:98%Color and Shape:SolidMolecular weight:1329.59BMS-196085
CAS:BMS-196085 is an effective and selective human β( 3) All agonists of adrenergic receptors, in β( 1) Partial agonist activity was 45%.Formula:C24H26F2N2O5SColor and Shape:SolidMolecular weight:492.547-Hydroxy-PIPAT maleate
CAS:7-Hydroxy-PIPAT maleate is a D3R agonist.Formula:C16H22INOColor and Shape:SolidMolecular weight:371.262TAK-615
CAS:TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of LPA1 receptors.Formula:C25H22FNO4Purity:99.73%Color and Shape:SolidMolecular weight:419.44Ref: TM-T9699
1mg72.00€5mg160.00€10mg245.00€25mg405.00€50mg572.00€100mg772.00€500mg1,539.00€1mL*10mM (DMSO)172.00€ABT-702
CAS:ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.Formula:C22H19BrN6OPurity:99.57%Color and Shape:SoildMolecular weight:463.33Cortistatin-8 acetate
Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.
Formula:C49H72N12O11S2Purity:99.01%Color and Shape:SoildMolecular weight:1069.3Ref: TM-TP2236L
1mg229.00€5mg560.00€10mg800.00€25mg1,216.00€50mg1,644.00€100mg2,213.00€500mg4,436.00€GR 64349
CAS:Potent NK2 agonist, EC50=3.7 nM in rat colon; >1000x selectivity over NK1, >300x over NK3; effective in vivo.Formula:C42H68N10O11SPurity:98%Color and Shape:SolidMolecular weight:921.12K41498
CAS:Potent CRF2α/β antagonist; Ki: 0.66/0.62 nM, weak for CRF1 (425 nM). Blocks sauvagine in hCRF2 cells and urocortin hypotension in rats.Formula:C162H276N48O46Purity:98%Color and Shape:SolidMolecular weight:3632.26Danshenol B
Danshenol B is a natural product that can be used as a reference standard.Formula:C22H26O4Color and Shape:SolidMolecular weight:354.446IRAK inhibitor 4 trans
IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.Formula:C33H35F3N6O3Purity:98%Color and Shape:SolidMolecular weight:620.66GLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Formula:C165H254N44O55SPurity:98%Color and Shape:SolidMolecular weight:3766.19Thielavin A
CAS:Thielavin A, from T. terricola, inhibits COX and glucose-6-phosphatase; non-competitive α-glucosidase inhibitor.Formula:C29H30O10Color and Shape:SolidMolecular weight:538.549Urocortin, rat
CAS:Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.Formula:C206H338N62O64Purity:98%Color and Shape:SolidMolecular weight:4707.2612-epi Leukotriene B4
CAS:LTB4 is made enzymatically (12(R)-specific) and non-enzymatically (6-trans-12-epi mix). 12-epi LTB4 has low receptor activity.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.472PG106
CAS:Selective hMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5 receptors.Formula:C51H69N13O9Purity:98%Color and Shape:SolidMolecular weight:1008.19Hydroxybupropion
CAS:Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).Formula:C13H18ClNO2Purity:99.73%Color and Shape:Off-White SolidMolecular weight:255.74Ref: TM-T11588
1mg89.00€5mg204.00€10mg331.00€25mg545.00€50mg777.00€100mg1,063.00€1mL*10mM (DMSO)232.00€JMV 449
CAS:Potent neurotensin agonist; IC50=0.15 nM, EC50=1.9 nM. Causes hypothermia, neuroprotection, analgesia in mice.Formula:C38H66N8O7Purity:98%Color and Shape:SolidMolecular weight:746.96Spantide acetate
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.
Formula:C77H112N20O15Purity:98.9200%Color and Shape:SolidMolecular weight:1557.8411-deoxy Prostaglandin E1
CAS:11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and causeFormula:C20H34O4Color and Shape:SolidMolecular weight:338.48Pasireotide
CAS:Pasireotide (SOM 230) is a cyclohexapeptide, mimicking somatostatin with high affinity for sst1/2/3/4/5 receptors (pKi=8.2/9.0/9.1/<7.0/9.9).Formula:C58H66N10O9Purity:98%Color and Shape:SolidMolecular weight:1047.21
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