GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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BM213 acetate
BM213 acetate is a selective C5aR1 agonist with antitumor activity that induces C5aR1-mediated calcium mobilization and pERK1/2 signaling.
Formula:C45H74N12O12Purity:99.88%Color and Shape:SolidMolecular weight:975.14RS 56812
CAS:RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive disorders.Formula:C18H21N3O2Purity:99.38%Color and Shape:SoildMolecular weight:311.38Orexin A (human, rat, mouse)
CAS:Orexin A, a 33 AA neuropeptide in humans, rats, mice, influences various processes, studied in pancreatic function and as an OX1R antagonist.Formula:C152H243N47O44S4Purity:98%Color and Shape:SolidMolecular weight:3561.1BAM (8-22) acetate
BAM (8-22) acetate, a proenkephalin A derivative, stimulates MrgprC11, hMrgprX1, and causes scratching in mice.Formula:C93H131N25O25SPurity:98.85%Color and Shape:SolidMolecular weight:2031.25Xanthine amine congener dihydrochloride
CAS:XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.Formula:C21H30Cl2N6O4Color and Shape:SolidMolecular weight:501.41cAC 253 acetate
cAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin binding, with an IC50 of 25 nM.
Formula:C128H206N42O42S2Purity:98.16% - 99.99%Color and Shape:SoildMolecular weight:3069.39Tirzepatide
CAS:Tirzepatide (LY-3298176) is a dual glucose-dependent polypeptide (GIP) (EC50=0.042 nM) and glucagon-like peptide-1 (GLP-1) (EC50=0.086 nM) receptor agonist.Formula:C225H348N48O68Purity:99.52% - 99.99%Color and Shape:SolidMolecular weight:4813.45Donetidine
CAS:Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Formula:C20H25N5O3SPurity:99.32%Color and Shape:SolidMolecular weight:415.51R 50595
CAS:R 50595 is a selective non-competitive cisapride antagonist.Formula:C30H35Cl2F2N3O3Purity:98%Color and Shape:SolidMolecular weight:594.52Zebrafish Kisspeptin-1
CAS:Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.Formula:C58H84N16O15Color and Shape:SolidMolecular weight:1245.39AZ7976
CAS:AZ7976 (Compound 42), a potent and highly selective agonist for Relaxin Family Peptide Receptor 1 (RXFP1) with a pEC 50 value greater than 10.5, operates through an allosteric mechanism to enhance RXFP1's cAMP signaling, which physiologically elevates heart rate. This property makes AZ7976 a valuable tool in cardiovascular disease research [1].Formula:C30H33F7N2O6SColor and Shape:SolidMolecular weight:682.65Anthramycin
CAS:Anthramycin: a PBD family antibiotic with antitumor effects and CNS cholecystokinin antagonist properties in mice.Formula:C16H17N3O4Color and Shape:SolidMolecular weight:315.32Esprolol
CAS:Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.Formula:C17H27NO4Purity:71.58% - 99.16%Color and Shape:SoildMolecular weight:309.4Ref: TM-T27286L
1mg80.00€2mg105.00€5mg172.00€10mg253.00€25mg414.00€50mg583.00€100mg783.00€200mg1,054.00€A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.Formula:C34H34N6O6Purity:98%Color and Shape:SolidMolecular weight:622.67Nadolol
CAS:Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities.Formula:C17H27NO4Purity:99.87% - 99.92%Color and Shape:White To Off-White Crystalline Powder SolidMolecular weight:309.40[D-Pro2] Spantide I TFA
[D-Pro2] Spantide I TFA is an analog of Spantide I, a selective antagonist of the NK1 receptor [1].Formula:C75H108N20O13·xC2HF3O2Purity:98%Color and Shape:Solid5-HT2A receptor agonist-6
CAS:5-HT2A receptor agonist-6 (compound 47) is a selective agonist of the 5-HT2A receptor with a pEC50 value of 6.58.Formula:C18H19N3O3Color and Shape:SolidMolecular weight:325.36Tetrapeptide-1
CAS:Tetrapeptide-1 is a bioactive peptide renowned for its antioxidant properties and has been cited as an ingredient in cosmetics [1].Formula:C20H36N4O6Purity:98%Color and Shape:SolidMolecular weight:428.52α-CGRP(human) TFA
α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as aFormula:C165H268F3N51O51S2Color and Shape:SolidMolecular weight:3903.33PSB-SB-1203
CAS:PSB-SB-1203 (Compound 25b) is a dual CB1/CB2 ligand that blocks the CB1 receptor and activates the CB2 receptor with a CB1 Ki of 0.244 μM, a CB2 Ki of 0.210 μM, and an EC50 of 0.054 μM. It shows potential for research in obesity and cancer.Formula:C25H30O4Color and Shape:SolidMolecular weight:394.5
